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Bulletin 2010/31 - European Patent Office

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(C07D) I.1(2)<br />

(62) 05716085.5 / 1 730 138<br />

C07D 405/04 → (51) C07D 401/04<br />

C07D 409/14 → (51) A01N 43/56<br />

C07D 413/12 → (51) C07D 209/42<br />

C07D 413/14 → (51) A61K <strong>31</strong>/553<br />

C07D 417/06 → (51) C07D 405/04<br />

(51) C07D 471/04 (11) 2 213 671 A1<br />

A61K 49/00 A61K 49/04<br />

(25) Ja (26) En<br />

(21) 08841078.2 (22) 24.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/069336 24.10.2008<br />

(87) WO 2009/054497 2009/18 30.04.2009<br />

(30) 26.10.2007 JP 2007278504<br />

(54) • NEUE VERBINDUNG MIT AFFINITÄT ZU<br />

AMYLOID<br />

• NOVEL COMPOUND HAVING AFFINITY<br />

FOR AMYLOID<br />

• NOUVEAU COMPOSÉ PRÉSENTANT UNE<br />

AFFINITÉ POUR L'AMYLOÏDE<br />

(71) Nihon Medi-Physics Co., Ltd., 3-4-10 Shinsuna<br />

Koto-ku, Tokyo 136-0075, JP<br />

(72) TANIFUJI, Shigeyuki, Sodegaura-shi Chiba<br />

299-0266, JP<br />

NAKAMURA, Daisaku, Sodegaura-shi Chiba<br />

299-0266, JP<br />

TAKASAKI, Shinya, Sodegaura-shi Chiba<br />

299-0266, JP<br />

OKUMURA, Yuki, Sodegaura-shi Chiba 299-<br />

0266, JP<br />

(74) Wilhelms · Kilian & Partner <strong>Patent</strong>anwälte,<br />

Eduard-Schmid-Straße 2, 81541 München,<br />

DE<br />

(51) C07D 471/04 (11) 2 213 672 A1<br />

A61K 49/00 A61K 49/04<br />

(25) Ja (26) En<br />

(21) 08842644.0 (22) 24.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/069335 24.10.2008<br />

(87) WO 2009/054496 2009/18 30.04.2009<br />

(30) 24.10.2007 JP 2007276826<br />

(54) • NEUE VERBINDUNG MIT AFFINITÄT ZU<br />

AMYLOID<br />

• NOVEL COMPOUND HAVING AFFINITY<br />

FOR AMYLOID<br />

• NOUVEAU COMPOSÉ POSSÉDANT UNE<br />

AFFINITÉ VIS-À-VIS D'UNE SUBSTANCE<br />

AMYLOÏDE<br />

(71) Nihon Medi-Physics Co., Ltd., 3-4-10 Shinsuna<br />

Koto-ku, Tokyo 136-0075, JP<br />

(72) TANIFUJI, Shigeyuki, Sodegaura-shi Chiba<br />

299-0266, JP<br />

NAKAMURA, Daisaku, Sodegaura-shi Chiba<br />

299-0266, JP<br />

TAKASAKI, Shinya, Sodegaura-shi Chiba<br />

299-0266, JP<br />

OKUMURA, Yuki, Sodegaura-shi Chiba 299-<br />

0266, JP<br />

(74) Wilhelms · Kilian & Partner <strong>Patent</strong>anwälte,<br />

Eduard-Schmid-Straße 2, 81541 München,<br />

DE<br />

(51) C07D 487/04 (11) 2 213 673 A1<br />

A61K <strong>31</strong>/519 A61K 39/395<br />

A61K 45/00 A61P 35/00<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

A61P 35/02 A61P 43/00<br />

C07D 519/00<br />

(25) Ja (26) En<br />

(21) 08842196.1 (22) 20.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/068932 20.10.2008<br />

(87) WO 2009/054332 2009/18 30.04.2009<br />

(30) 23.10.2007 JP 2007275<strong>31</strong>1<br />

(54) • PYRIDONSUBSTITUIERTES DIHYDROPY-<br />

RAZOLOPYRIMIDINONDERIVAT<br />

• PYRIDONE-SUBSTITUTED-DIHYDROPYR-<br />

AZOLOPYRIMIDINONE DERIVATIVE<br />

• DÉRIVÉ DE DIHYDROPYRAZOLOPYRIMI-<br />

DINONE SUBSTITUÉ PAR PYRIDONE<br />

(71) Banyu Pharmaceutical Co., Ltd., Kitanomaru<br />

Square 1-13-12 Kudankita, Chiyoda-ku<br />

Tokyo 102-8667, JP<br />

(72) FRUYAMA, Hidetomo, Tsukuba-shi Ibaraki<br />

300-2611, JP<br />

KAWAMURA, Mikako, Tsukuba-shi Ibaraki<br />

300-2611, JP<br />

SAKAMOTO, Toshihiro, Tsukuba-shi Ibaraki<br />

300-2611, JP<br />

YAMAMOTO, Fuyuki, Tsukuba-shi Ibaraki<br />

300-2611, JP<br />

YOSHIZUMI, Takashi, Tsukuba-shi Ibaraki<br />

300-2611, JP<br />

(74) Hussain, Deeba, Merck Sharp & Dohme<br />

Limited Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

(51) C07D 487/04 (11) 2 213 674 A1<br />

A61K <strong>31</strong>/519 A61P 35/00<br />

(25) Zh (26) En<br />

(21) 08844190.2 (22) 21.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) CN 2008/072758 21.10.2008<br />

(87) WO 2009/056029 2009/19 07.05.2009<br />

(30) 24.10.2007 CN 200710092879<br />

(54) • REINIGUNGSVERFAHREN FÜR PEMETRE-<br />

XEDSALZE, NATRIUMSALZE UND DINAT-<br />

RIUMSALZE<br />

• PURIFICATION METHOD OF PEMETREXED<br />

SALTS,SODIUM SALTS AND DISODIUM<br />

SALTS<br />

• PROCÉDÉ DE PURIFICATION DE SELS,<br />

SELS SODIQUES ET SELS DISSODIQUES<br />

DE PEMETREXED<br />

(71) Chongqing Pharmaceutical Research Institute<br />

Co., Ltd., 565 Tushan Road Nan'an<br />

District, Chongqing 400-061, CN<br />

(72) LUO, Jie, Chongqing 400061, CN<br />

LIN, Meng, Chongqing 400061, CN<br />

LIN, Bo, Chongqing 400061, CN<br />

YE, Wenrun, Chongqing 400061, CN<br />

QIN, Yongmei, Chongqing 400061, CN<br />

DENG, Jie, Chongqing 400061, CN<br />

(74) Epping - Hermann - Fischer, <strong>Patent</strong>anwaltsgesellschaft<br />

mbH Ridlerstrasse 55, 80339<br />

München, DE<br />

C07D 487/04 → (51) C07D 221/18<br />

C07D 493/04 → (51) C07D 405/04<br />

(51) C07D 498/04 (11) 2 213 675 A1<br />

A61K <strong>31</strong>/553 A61P 1/00<br />

A61P 3/04 A61P 13/00<br />

A61P 15/00 A61P 43/00<br />

(25) Ja (26) En<br />

(21) 08849982.7 (22) 14.11.2008<br />

291<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2010</strong>) 04.08.<strong>2010</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/070808 14.11.2008<br />

(87) WO 2009/063991 2009/21 22.05.2009<br />

(30) 15.11.2007 JP 2007297169<br />

(54) • PYRIDOOXAZEPINDERIVAT UND SEINE<br />

VERWENDUNG<br />

• PYRIDOOXAZEPINE DERIVATIVE AND USE<br />

THEREOF<br />

• DÉRIVÉ DE PYRIDOOXAZÉPINE ET SON<br />

UTILISATION<br />

(71) Takeda Pharmaceutical Company Limited, 1-<br />

1, Doshomachi 4-chome Chuo-ku, Osakashi,<br />

Osaka 541-0045, JP<br />

(72) MATSUMOTO, Takahiro, Osaka-shi Osaka<br />

532-8686, JP<br />

KUSUMOTO, Tomokazu, Osaka-shi Osaka<br />

532-8686, JP<br />

(74) Meissner, Bolte & Partner, Anwaltssozietät<br />

GbR Widenmayerstrasse 48, 80538<br />

München, DE<br />

(51) C07D 501/04 (11) 2 213 676 A1<br />

C07D 501/22<br />

(25) En (26) En<br />

(21) 09177637.7 (22) 01.11.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LU MC NL PL PT RO SE SI<br />

SK TR<br />

AL HR LT LV MK YU<br />

(54) • Neuartiges Verfahren zur Herstellung von<br />

Cefprozil<br />

• A Novel process for preparation of cefprozil<br />

• Nouveau procédé de préparation de cefprozil<br />

(71) Hetero Drugs Limited, Hetero House 8-3-<br />

166/7/1, Erragadda, Hyderabad, Andhrapradesh.<br />

Hyderabad 500 018, IN<br />

(72) Reddy, Bandi Parthasaradhi, 500018,<br />

Hyderabad, IN<br />

Reddy, Kura Rathnakar, 500018, Hyderabad,<br />

IN<br />

Reddy, Rapolu Raji, 500018, Hyderabad, IN<br />

Reddy, Dasari Muralidhara, 500018, Hyderabad,<br />

IN<br />

Murali, Nagabelli, 500018, Hyderabad, IN<br />

(74) Thomas, Simon, Urquhart-Dykes & Lord LLP<br />

30 Welbeck Street, London W1G 8ER, GB<br />

(62) 04806740.9 / 1 809 638<br />

C07D 501/22 → (51) C07D 501/04<br />

C07D 519/00 → (51) C07D 487/04<br />

(51) C07F 9/09 (11) 2 213 677 A1<br />

C07F 9/11 C07B 61/00<br />

C08F 4/52<br />

(25) Ja (26) En<br />

(21) 08840734.1 (22) 15.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/068682 15.10.2008<br />

(87) WO 2009/051144 2009/17 23.04.2009<br />

(30) 15.10.2007 JP 2007267991<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

DIALKYLPHOSPHATESTER-SELTENERD-<br />

SALZ ODER DIOLEYLPHOSPHATESTER-<br />

SELTENERDSALZ<br />

• PROCESS FOR PRODUCTION OF DIALKYL<br />

PHOSPHATE ESTER RARE-EARTH SALT<br />

OR DIOLEYL PHOSPHATE ESTER RARE-<br />

EARTH SALT OF

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