Bulletin 2010/15 - European Patent Office

(C07D) I.1(1)
URMANN, Mathias, 65926 Frankfurt am
Main, DE
HALLAND, Nis, 65926 Frankfurt am Main, DE
(74) Then, Johann, et al, Sanofi-Aventis
Deutschland GmbH Patent- und Lizenzabteilung
Industriepark Höchst Gebäude K 801,
65926 Frankfurt am Main, DE
(51) C07D 471/04 (11) 2 173 748 A2*
C07D 487/04 A61K 31/437
A61P 35/04
(25) En (26) En
(21) 08771523.1 (22) 19.06.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) US 2008/067566 19.06.2008
(87) WO 2009/002807 2009/01 31.12.2008
(88) 30.07.2009
(30) 22.06.2007 US 945820 P
(54) • INDOLYLPYRROLIDINE ZUR BEHAND-
LUNG VON KREBS
• INDOLYL PYRROLIDINES FOR THE
TREATMENT OF CANCER
• COMPOSITIONS ET PROCÉDÉS DE TRAI-
TEMENT DU CANCER
(71) ArQule, Inc., 19 Presidential Way, Woburn,
MA 01801, US
(72) WESTLUND, Neil, Groton, MA 01450, US
HILL, Jason, Auburndale, MA 02466, US
ASHWELL, Mark, A., Carlisle, MA 01741, US
NAMDEV, Nivedita, D., Westford, MA 01886,
US
WANG, Jianqiang, Acton, MA 01720, US
ALI, Syed, M., North Andover, MA 01845, US
(74) UEXKÜLL & STOLBERG, Patentanwälte
Beselerstrasse 4, 22607 Hamburg, DE
(51) C07D 471/04 (11) 2 173 749 A1*
A61K 31/437 A01N 43/40
A61P 31/10
(25) En (26) En
(21) 08750663.0 (22) 21.05.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) GB 2008/001738 21.05.2008
(87) WO 2008/145963 2008/49 04.12.2008
(30) 25.05.2007 GB 0710121
(54) • 2-OXO-2-(2-PHENYL-5,6,7,8-TETRAHYD-
ROINDOLIZIN-3-YL)ACETAMIDDERIVATE
UND VERWANDTE VERBINDUNGEN ALS
ANTIPILZMITTEL
• 2-OXO-2- (2-PHENYL-5,6,7,8-TETRAHY-
DRO-INDOLIZIN-3-YL) -ACETAMIDE
DERIVATIVES AND RELATED COM-
POUNDS AS ANTIFUNGAL AGENTS
• DÉRIVÉS DE 2-OXO-2- (2-PHÉNYL-5,6,7,
8-TÉTRAHYDRO-INDOLIZIN-3-YL) -ACÉ-
TAMIDE ET COMPOSÉS ASSOCIÉS UTILI-
SÉS COMME AGENTS ANTIFONGIQUES
(71) F2G Limited, Lankro Way, Eccles Manchester
Greater Manchester M30 0BH, GB
(72) PAYNE, Lloyd, James, Manchester M30 0BH,
GB
DOWNHAM, Robert, Suffolk CB8 0QN, GB
SIBLEY, Graham, Edward, Morris, Manchester
M30 0BH, GB
EDWARDS, Philip, Cheshire SK7 2NW, GB
DAVIES, Gareth, Morse, Cheshire SK10 2EP,
GB
(74) Simons, Amanda Louise, J.A. Kemp & Co.
14 South Square Gray's Inn, London WC1R
5JJ, GB
Europäisches Patentblatt
European Patent Bulletin
Bulletin européen des brevets
C07D 471/04 → (51) A61K 31/4706
C07D 471/04 → (51) C07D 213/127
C07D 471/04 → (51) C07D 213/81
C07D 471/04 → (51) C07D 235/08
C07D 471/04 → (51) C07D 417/14
(51) C07D 471/10 (11) 2 173 750 A1*
A61K 31/444 A61P 3/04
(25) En (26) En
(21) 08771573.6 (22) 20.06.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) US 2008/067637 20.06.2008
(87) WO 2008/157752 2008/52 24.12.2008
(30) 21.06.2007 US 945487 P
(54) • SPIROCYCLEN ALS INHIBITOREN VON 11-
BETA-HYDROXYLSTEROIDDEHYDROGE-
NASE TYP 1
• SPIROCYCLES AS INHIBITORS OF 11-
BETA HYDROXYL STEROID DEHYDRO-
GENASE TYPE 1
• SPIROCYCLES UTILISÉS EN TANT QU'IN-
HIBITEURS DE LA 11- -HYDROXY-STÉ-
ROÏDE DÉSHYDROGÉNASE DE TYPE 1
(71) Incyte Corporation, Experimental Station
Route 141&Henry Clay Road Building E336,
Wilmer Delaware 19880, US
(72) YAO, Wenqing, Kennett Square, Pennsylvania
19348, US
ZHUO, Jincong, Boothwyn, Pennsylvania
19061, US
ZHANG, Colin, Ambler, Pennsylvania 19002,
US
(74) Howard, Paul Nicholas, et al, Carpmaels &
Ransford 43-45 Bloomsbury Square, London
WC1A 2RA, GB
C07D 471/14 → (51) C07D 471/04
C07D 473/00 → (51) A61K 31/505
C07D 473/18 → (51) C07D 403/06
C07D 473/34 → (51) C07D 403/06
(51) C07D 487/04 (11) 2 173 751 A2*
(25) En (26) En
(21) 08770791.5 (22) 12.06.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) US 2008/066658 12.06.2008
(87) WO 2008/157207 2008/52 24.12.2008
(88) 26.02.2009
(30) 13.06.2007 US 943695 P
(54) • METABOLITEN DES JANUS-KINASE-INHI-
BITORS (R)-3-(4-(7H-PYRROLO[2,3-D]
PYRIMIDIN-4-YL)-1H-PYRAZOL-1-YL)-3-
CYCLOPENTYLPROPANNITRIL
• METABOLITES OF THE JANUS KINASE
INHIBITOR (R)-3-(4-(7H-PYRROLO[2,3-D]
PYRIMIDIN-4-YL)-LH-PYRAZOL-L-YL)-3-
CYCLOPENTYLPROPANENITRILE
• MÉTABOLITES DE L'INHIBITEUR DE
JANUS KINASE (R)-3-(4-(7H-PYRROLO
[2,3-D]PYRIMIDIN-4-YL)-1H-PYRAZOL-1-
YL)-3-CYCLOPENTYLPROPANENITRILE
(71) Incyte Corporation, Experimental Station,
Route 141 & Henry Clay Road, Building
E336, Wilmington, DE 19880, US
101
Anmeldungen
Applications
Demandes (15/2010) 14.04.2010
(72) RODGERS, James D., Landenberg, PA
19350, US
ARVANITIS, Argyrios G., Kennett Square,
Pennsylvania 19348, US
SHI, Jack Guoen, Wilmington, Delaware
19803, US
(74) Howard, Paul Nicholas, et al, Carpmaels &
Ransford 43-45 Bloomsbury Square, London
WC1A 2RA, GB
(51) C07D 487/04 (11) 2 173 752 A2*
A61K 31/519
(25) En (26) En
(21) 08770794.9 (22) 12.06.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) US 2008/066662 12.06.2008
(87) WO 2008/157208 2008/52 24.12.2008
(88) 12.02.2009
(30) 13.06.2007 US 943705 P
(54) • SALZE DES JANUS-KINASE-INHIBITORS
(R)-3-(4-(7H-PYRROLO[2,3-D]PYRIMI-
DIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLO-
PENTYLPROPANNITRIL
• SALTS OF THE JANUS KINASE INHIBITOR
(R)-3-(4-(7H-PYRROLOÝ2,3-D¨PYRIMI-
DIN-4-YL)-1H-PYRAZOL-1-YL)-3-CYCLO-
PENTYLPROPANENITRILE
• SELS DE L'INHIBITEUR (R)-3-(4-(7H-
PYRROLOÝ2,3-D¨PYRIMIDIN-4-YL)-1H-
PYRAZOL-1-YL)-3-CYCLOPENTYLPROPA-
NENITRILE DE LA JANUS KINASE
(71) Incyte Corporation, Experimental Station,
Route 141 & Henry Clay Road, Building
E336, Wilmington, DE 19880, US
(72) LI, Hui-Yin, Hockessin, DE 19707, US
RODGERS, James, D., Landenberg, PA
19350, US
(74) Howard, Paul Nicholas, et al, Carpmaels &
Ransford 43-45 Bloomsbury Square, London
WC1A 2RA, GB
C07D 487/04 → (51) C07D 471/04
(51) C07D 487/08 (11) 2 173 753 A2*
C07B 59/00
(25) En (26) En
(21) 08761135.6 (22) 18.06.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) EP 2008/057659 18.06.2008
(87) WO 2008/155339 2008/52 24.12.2008
(88) 26.02.2009
(30) 20.06.2007 US 945118 P
(54) • MARKIERUNGSVERFAHREN
• LABELLING METHODS
• PROCÉDÉS DE MARQUAGE
(71) GE Healthcare UK Limited, Amersham Place,
Little Chalfont Buckinghamshire HP7 9NA,
GB
(72) JACKSON, Alexander, Amersham Buckinghamshire
HP7 9LL, GB
BHALLA, Rajiv, Amersham Buckinghamshire
HP7 9LL, GB
(74) Canning, Lewis R., GE Healthcare Limited
Pollards Wood Nightingales Lane Chalfont St
Giles, Buckinghamshire HP8 4SP, GB
C07D 487/08 → (51) C07D 401/04
(51) C07D 489/02 (11) 2 173 754 A1*
C07D 489/04
(25) En (26) En
(21) 08772838.2 (22) 30.06.2008