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Bulletin 2010/15 - European Patent Office

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(A61K) II.1(1)<br />

A61K 33/24 A61P 35/00<br />

A61L 27/18 A61L 27/54<br />

(25) En (26) En<br />

(21) 01930891.5 (22) 27.04.2001<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 26.03.2003<br />

(86) US 2001/013730 27.04.2001<br />

(87) WO 2001/082780 2001/45 08.11.2001<br />

(30) 29.04.2000 CN 01101092<br />

<strong>15</strong>.09.2000 US 663559<br />

12.10.2000 US 687342<br />

13.11.2000 CN 00129316<br />

(54) • BEHANDLUNG VON KREBS UNTER VER-<br />

WENDUNG VON ORGANELLKRISTALLI-<br />

SIERENDEN VERBINDUNGEN<br />

• TREATING CANCER USING ORGANELLE<br />

CRYSTALLIZING AGENTS<br />

• TRAITEMENT DU CANCER PAR UTILISA-<br />

TION D'AGENTS DE CRISTALLISATION<br />

D'ORGANITE<br />

(73) Kong, Qingzhong, Shandong Lanjim Pharmaceuticals<br />

Co. Ltd Tian-Chen Road 1750<br />

Jinan Hi-tech Zone, Jinan, CN<br />

(72) Kong, Qingzhong, Jinan, CN<br />

(74) Evens, Paul Jonathan, et al, Maguire Boss 24<br />

East Street, St. Ives Cambridgeshire PE27<br />

5PD, GB<br />

A61K 31/41 → (51) C07D 231/54<br />

A61K 31/4<strong>15</strong>5 → (51) C07D 209/18<br />

A61K 31/4166 → (51) C07D 401/14<br />

A61K 31/4178 → (51) C07D 209/18<br />

A61K 31/422 → (51) C07D 209/18<br />

(51) A61K 31/426 (11) 1 629 842 B1<br />

A61K 31/427 A61K 9/06<br />

A61P 31/12<br />

(25) De (26) De<br />

(21) 05024999.4 (22) 10.06.2002<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 01.03.2006<br />

(30) 22.06.2001 DE 10129714<br />

(54) • Topische Anwendung von Thiazolylamiden<br />

• Topical application of thiazolyl amides<br />

• Utilisation topique d'amides de thiazolyle<br />

(73) AiCuris GmbH & Co. KG, Friedrich-Ebert-<br />

Strasse 475, 42117 Wuppertal, DE<br />

(72) Betz, Ulrich, Dr., 64354 Reinheim, DE<br />

Laich, Tobias, Dr., 51069 Köln, DE<br />

Bender, Wolfgang, Dr., 42113 Wuppertal, DE<br />

Fischer, Rüdiger, Dr., 50259 Pulheim, DE<br />

Hendrix, Martin, Dr., 5<strong>15</strong>19 Odenthal, DE<br />

Kleymann, Gerald, Dr., 32107 Bad Salzuflen,<br />

DE<br />

(74) Findeisen, Marco, et al, Witte, Weller &<br />

Partner <strong>Patent</strong>anwälte Postfach 10 54 62,<br />

70047 Stuttgart, DE<br />

(62) 02743172.5 / 1 401 435<br />

A61K 31/427 → (51) A61K 31/41<br />

A61K 31/427 → (51) A61K 31/426<br />

A61K 31/427 → (51) C07D 209/18<br />

A61K 31/433 → (51) C07D 209/18<br />

A61K 31/438 → (51) C07D 401/14<br />

A61K 31/44 → (51) C07D 403/02<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(51) A61K 31/4439 (11) 1 656 141 B1<br />

A61K 31/403 C07D 401/04<br />

C07D 209/86 C07D 209/88<br />

A61P 25/28<br />

(25) En (26) En<br />

(21) 04767944.4 (22) 29.07.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

LT LV<br />

(43) 17.05.2006<br />

(86) GB 2004/003286 29.07.2004<br />

(87) WO 2005/013985 2005/07 17.02.2005<br />

(30) 07.08.2003 GB 0318552<br />

08.04.2004 GB 0408100<br />

(54) • BEHANDLUNG VON ALZHEIMER-KRANK-<br />

HEIT UND VERWANDTEN ZUSTÄNDEN<br />

• TREATMENT FOR ALZHEIMER S DISEASE<br />

AND RELATED CONDITIONS<br />

• PROCEDE POUR TRAITER LA MALADIE<br />

D'ALZHEIMER ET DES PATHOLOGIES<br />

LIEES<br />

(73) MERCK SHARP & DOHME LTD., Hertford<br />

Road, Hoddesdon, Hertfordshire EN11 9BU,<br />

GB<br />

(72) BEHER, Dirk, Harlow Essex CM20 2QR, GB<br />

BETTATI, Michela, Harlow Essex CM20 2QR,<br />

GB<br />

CHECKSFIELD, Graham David, Harlow Essex<br />

CM20 2QR, GB<br />

CHURCHER, Ian, Harlow Essex CM20 2QR,<br />

GB<br />

DOUGHTY, Victoria Alexandra, Harlow Essex<br />

CM20 2QR, GB<br />

OAKLEY, Paul Joseph, Harlow Essex CM20<br />

2QR, GB<br />

QUDDUS, Abdul, Harlow Essex CM20 2QR,<br />

GB<br />

TEALL, Martin Richard, Harlow Essex CM20<br />

2QR, GB<br />

WRIGLEY, Jonathan David, Harlow Essex<br />

CM20 2QR, GB<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

A61K 31/4439 → (51) C07D 401/04<br />

A61K 31/4468 → (51) C07D 453/02<br />

A61K 31/451 → (51) C07D 211/14<br />

A61K 31/4545 → (51) C07D 211/14<br />

(51) A61K 31/485 (11) 1 663 229 B1<br />

A61K 9/00 A61K 9/22<br />

A61P 25/36<br />

(25) En (26) En<br />

(21) 04788669.2 (22) 09.09.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

AL HR LT LV MK<br />

(43) 07.06.2006<br />

(86) US 2004/029521 09.09.2004<br />

(87) WO 2005/032555 2005/<strong>15</strong> 14.04.2005<br />

(30) 25.09.2003 US 506222 P<br />

(54) • PHARMAZEUTISCHE KOMBINATIONEN<br />

VON HYDROCODON UND NALTREXON<br />

• PHARMACEUTICAL COMBINATIONS OF<br />

HYDROCODONE AND NALTREXONE<br />

• COMBINAISONS PHARMACEUTIQUES<br />

D'HYDROCODONE ET DE NALTREXONE<br />

(73) EURO-CELTIQUE S.A., 2, avenue Charles de<br />

Gaulle, 1653 Luxembourg, LU<br />

(72) OSHLACK, Benjamin, Boca Raton, FL 33432,<br />

US<br />

530<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>15</strong>/<strong>2010</strong>) 14.04.<strong>2010</strong><br />

WRIGHT, Curtis, Rockport, MA 01966, US<br />

BREDER, Chris, Greenwich, CT 06830, US<br />

(74) Bühler, Dirk, Maiwald <strong>Patent</strong>anwalts GmbH<br />

Elisenhof Elisenstraße 3, 80335 München,<br />

DE<br />

A61K 31/495 → (51) C07D 211/14<br />

(51) A61K 31/496 (11) 1 419 776 B1<br />

C07D 2<strong>15</strong>/22 A61P 25/18<br />

(25) En (26) En<br />

(21) 04002427.5 (22) 25.09.2002<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SK TR<br />

LT LV RO SI<br />

(43) 19.05.2004<br />

(30) 25.09.2001 JP 2001290645<br />

14.11.2001 JP 2001348276<br />

27.03.2002 CA 2379005<br />

(54) • Aripiprazole Wirkstoff mit niedriger Hygroskopie<br />

und Verfahren zu ihrer Herstellung<br />

• Low hygroscopic aripiprazole drug substance<br />

and processes for the preparation<br />

thereof<br />

• Substance pharmaceutique d'aripiprazole<br />

faiblement hygroscopique et méthodes de<br />

préparation associées<br />

(73) OTSUKA PHARMACEUTICAL CO., LTD., 9,<br />

Kandatsukasa-cho 2-chome, Chiyoda-ku<br />

Tokyo 101-8535, JP<br />

(72) Bando, Takuji, Tokushima-shi, Tokushima,<br />

JP<br />

Aoki, Satoshi, Naruto-shi, Tokushima, JP<br />

Kawasaki, Junichi, Itano-gun, Tokushima, JP<br />

Ishigami, Makoto, Itano-gun, Tokushima, JP<br />

Taniguchi, Youichi, Tokushima-shi, Tokushima,<br />

JP<br />

Yabuuchi, Tsuyoshi, Tokushima-shi,<br />

Tokushima, JP<br />

Fujimoto, Kiyoshi, Naruto-shi, Tokushima,<br />

JP<br />

Nishioka, Yoshihiro, Matsushige-cho, Itanogun,<br />

Tokushima, JP<br />

Kobayashi, Noriyuki, Tokushima-shi,<br />

Tokushima, JP<br />

Fujimura, Tsutomu, Naruto-shi, Tokushima,<br />

JP<br />

Takahashi, Masanori, Tokushima-shi,<br />

Tokushima, JP<br />

Abe, Kaoru, Tokushima-shi, Tokushima, JP<br />

Nakagawa, Tomonori, Matsushige-cho,<br />

Itano-gun,Tokushima, JP<br />

Shinhama, Koichi, Tokushima-shi, Tokushima,<br />

JP<br />

Utsumi, Naoto, Muyachotateiwa, Naruto-shi,<br />

Tokushima, JP<br />

Tominaga, Michiaki, Itano-gun, Tokushima,<br />

JP<br />

Oi, Yoshihiro, Tokushima-shi, Tokushima, JP<br />

Yamada, Shohei, Itano-gun, Tokushima, JP<br />

Tomikawa, Kenji, Tokushima-shi, Tokushima,<br />

JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

(60) 08000357.7 / 1 927 355<br />

08000358.5 / 1 925 308<br />

08000359.3 / 1 927 356<br />

08000360.1 / 1 927 357<br />

(62) 02782507.4 / 1 330 249<br />

A61K 31/496 → (51) C07D 231/12<br />

A61K 31/4965 → (51) C07D 403/02<br />

(51) A61K 31/501 (11) 1 363 636 B1<br />

A61K 33/06 A61P 9/04<br />

A61P 9/10<br />

(25) En (26) En

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