Bulletin 2010/15 - European Patent Office
Bulletin 2010/15 - European Patent Office
Bulletin 2010/15 - European Patent Office
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(A61K) II.1(1)<br />
A61K 33/24 A61P 35/00<br />
A61L 27/18 A61L 27/54<br />
(25) En (26) En<br />
(21) 01930891.5 (22) 27.04.2001<br />
(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />
LU MC NL PT SE TR<br />
(43) 26.03.2003<br />
(86) US 2001/013730 27.04.2001<br />
(87) WO 2001/082780 2001/45 08.11.2001<br />
(30) 29.04.2000 CN 01101092<br />
<strong>15</strong>.09.2000 US 663559<br />
12.10.2000 US 687342<br />
13.11.2000 CN 00129316<br />
(54) • BEHANDLUNG VON KREBS UNTER VER-<br />
WENDUNG VON ORGANELLKRISTALLI-<br />
SIERENDEN VERBINDUNGEN<br />
• TREATING CANCER USING ORGANELLE<br />
CRYSTALLIZING AGENTS<br />
• TRAITEMENT DU CANCER PAR UTILISA-<br />
TION D'AGENTS DE CRISTALLISATION<br />
D'ORGANITE<br />
(73) Kong, Qingzhong, Shandong Lanjim Pharmaceuticals<br />
Co. Ltd Tian-Chen Road 1750<br />
Jinan Hi-tech Zone, Jinan, CN<br />
(72) Kong, Qingzhong, Jinan, CN<br />
(74) Evens, Paul Jonathan, et al, Maguire Boss 24<br />
East Street, St. Ives Cambridgeshire PE27<br />
5PD, GB<br />
A61K 31/41 → (51) C07D 231/54<br />
A61K 31/4<strong>15</strong>5 → (51) C07D 209/18<br />
A61K 31/4166 → (51) C07D 401/14<br />
A61K 31/4178 → (51) C07D 209/18<br />
A61K 31/422 → (51) C07D 209/18<br />
(51) A61K 31/426 (11) 1 629 842 B1<br />
A61K 31/427 A61K 9/06<br />
A61P 31/12<br />
(25) De (26) De<br />
(21) 05024999.4 (22) 10.06.2002<br />
(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />
LU MC NL PT SE TR<br />
(43) 01.03.2006<br />
(30) 22.06.2001 DE 10129714<br />
(54) • Topische Anwendung von Thiazolylamiden<br />
• Topical application of thiazolyl amides<br />
• Utilisation topique d'amides de thiazolyle<br />
(73) AiCuris GmbH & Co. KG, Friedrich-Ebert-<br />
Strasse 475, 42117 Wuppertal, DE<br />
(72) Betz, Ulrich, Dr., 64354 Reinheim, DE<br />
Laich, Tobias, Dr., 51069 Köln, DE<br />
Bender, Wolfgang, Dr., 42113 Wuppertal, DE<br />
Fischer, Rüdiger, Dr., 50259 Pulheim, DE<br />
Hendrix, Martin, Dr., 5<strong>15</strong>19 Odenthal, DE<br />
Kleymann, Gerald, Dr., 32107 Bad Salzuflen,<br />
DE<br />
(74) Findeisen, Marco, et al, Witte, Weller &<br />
Partner <strong>Patent</strong>anwälte Postfach 10 54 62,<br />
70047 Stuttgart, DE<br />
(62) 02743172.5 / 1 401 435<br />
A61K 31/427 → (51) A61K 31/41<br />
A61K 31/427 → (51) A61K 31/426<br />
A61K 31/427 → (51) C07D 209/18<br />
A61K 31/433 → (51) C07D 209/18<br />
A61K 31/438 → (51) C07D 401/14<br />
A61K 31/44 → (51) C07D 403/02<br />
Europäisches <strong>Patent</strong>blatt<br />
<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />
<strong>Bulletin</strong> européen des brevets<br />
(51) A61K 31/4439 (11) 1 656 141 B1<br />
A61K 31/403 C07D 401/04<br />
C07D 209/86 C07D 209/88<br />
A61P 25/28<br />
(25) En (26) En<br />
(21) 04767944.4 (22) 29.07.2004<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />
TR<br />
LT LV<br />
(43) 17.05.2006<br />
(86) GB 2004/003286 29.07.2004<br />
(87) WO 2005/013985 2005/07 17.02.2005<br />
(30) 07.08.2003 GB 0318552<br />
08.04.2004 GB 0408100<br />
(54) • BEHANDLUNG VON ALZHEIMER-KRANK-<br />
HEIT UND VERWANDTEN ZUSTÄNDEN<br />
• TREATMENT FOR ALZHEIMER S DISEASE<br />
AND RELATED CONDITIONS<br />
• PROCEDE POUR TRAITER LA MALADIE<br />
D'ALZHEIMER ET DES PATHOLOGIES<br />
LIEES<br />
(73) MERCK SHARP & DOHME LTD., Hertford<br />
Road, Hoddesdon, Hertfordshire EN11 9BU,<br />
GB<br />
(72) BEHER, Dirk, Harlow Essex CM20 2QR, GB<br />
BETTATI, Michela, Harlow Essex CM20 2QR,<br />
GB<br />
CHECKSFIELD, Graham David, Harlow Essex<br />
CM20 2QR, GB<br />
CHURCHER, Ian, Harlow Essex CM20 2QR,<br />
GB<br />
DOUGHTY, Victoria Alexandra, Harlow Essex<br />
CM20 2QR, GB<br />
OAKLEY, Paul Joseph, Harlow Essex CM20<br />
2QR, GB<br />
QUDDUS, Abdul, Harlow Essex CM20 2QR,<br />
GB<br />
TEALL, Martin Richard, Harlow Essex CM20<br />
2QR, GB<br />
WRIGLEY, Jonathan David, Harlow Essex<br />
CM20 2QR, GB<br />
(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />
& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />
Hertford Road, Hoddesdon Hertfordshire<br />
EN11 9BU, GB<br />
A61K 31/4439 → (51) C07D 401/04<br />
A61K 31/4468 → (51) C07D 453/02<br />
A61K 31/451 → (51) C07D 211/14<br />
A61K 31/4545 → (51) C07D 211/14<br />
(51) A61K 31/485 (11) 1 663 229 B1<br />
A61K 9/00 A61K 9/22<br />
A61P 25/36<br />
(25) En (26) En<br />
(21) 04788669.2 (22) 09.09.2004<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />
TR<br />
AL HR LT LV MK<br />
(43) 07.06.2006<br />
(86) US 2004/029521 09.09.2004<br />
(87) WO 2005/032555 2005/<strong>15</strong> 14.04.2005<br />
(30) 25.09.2003 US 506222 P<br />
(54) • PHARMAZEUTISCHE KOMBINATIONEN<br />
VON HYDROCODON UND NALTREXON<br />
• PHARMACEUTICAL COMBINATIONS OF<br />
HYDROCODONE AND NALTREXONE<br />
• COMBINAISONS PHARMACEUTIQUES<br />
D'HYDROCODONE ET DE NALTREXONE<br />
(73) EURO-CELTIQUE S.A., 2, avenue Charles de<br />
Gaulle, 1653 Luxembourg, LU<br />
(72) OSHLACK, Benjamin, Boca Raton, FL 33432,<br />
US<br />
530<br />
<strong>Patent</strong>e<br />
<strong>Patent</strong>s<br />
Brevets (<strong>15</strong>/<strong>2010</strong>) 14.04.<strong>2010</strong><br />
WRIGHT, Curtis, Rockport, MA 01966, US<br />
BREDER, Chris, Greenwich, CT 06830, US<br />
(74) Bühler, Dirk, Maiwald <strong>Patent</strong>anwalts GmbH<br />
Elisenhof Elisenstraße 3, 80335 München,<br />
DE<br />
A61K 31/495 → (51) C07D 211/14<br />
(51) A61K 31/496 (11) 1 419 776 B1<br />
C07D 2<strong>15</strong>/22 A61P 25/18<br />
(25) En (26) En<br />
(21) 04002427.5 (22) 25.09.2002<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR IE IT LI LU MC NL PT SE SK TR<br />
LT LV RO SI<br />
(43) 19.05.2004<br />
(30) 25.09.2001 JP 2001290645<br />
14.11.2001 JP 2001348276<br />
27.03.2002 CA 2379005<br />
(54) • Aripiprazole Wirkstoff mit niedriger Hygroskopie<br />
und Verfahren zu ihrer Herstellung<br />
• Low hygroscopic aripiprazole drug substance<br />
and processes for the preparation<br />
thereof<br />
• Substance pharmaceutique d'aripiprazole<br />
faiblement hygroscopique et méthodes de<br />
préparation associées<br />
(73) OTSUKA PHARMACEUTICAL CO., LTD., 9,<br />
Kandatsukasa-cho 2-chome, Chiyoda-ku<br />
Tokyo 101-8535, JP<br />
(72) Bando, Takuji, Tokushima-shi, Tokushima,<br />
JP<br />
Aoki, Satoshi, Naruto-shi, Tokushima, JP<br />
Kawasaki, Junichi, Itano-gun, Tokushima, JP<br />
Ishigami, Makoto, Itano-gun, Tokushima, JP<br />
Taniguchi, Youichi, Tokushima-shi, Tokushima,<br />
JP<br />
Yabuuchi, Tsuyoshi, Tokushima-shi,<br />
Tokushima, JP<br />
Fujimoto, Kiyoshi, Naruto-shi, Tokushima,<br />
JP<br />
Nishioka, Yoshihiro, Matsushige-cho, Itanogun,<br />
Tokushima, JP<br />
Kobayashi, Noriyuki, Tokushima-shi,<br />
Tokushima, JP<br />
Fujimura, Tsutomu, Naruto-shi, Tokushima,<br />
JP<br />
Takahashi, Masanori, Tokushima-shi,<br />
Tokushima, JP<br />
Abe, Kaoru, Tokushima-shi, Tokushima, JP<br />
Nakagawa, Tomonori, Matsushige-cho,<br />
Itano-gun,Tokushima, JP<br />
Shinhama, Koichi, Tokushima-shi, Tokushima,<br />
JP<br />
Utsumi, Naoto, Muyachotateiwa, Naruto-shi,<br />
Tokushima, JP<br />
Tominaga, Michiaki, Itano-gun, Tokushima,<br />
JP<br />
Oi, Yoshihiro, Tokushima-shi, Tokushima, JP<br />
Yamada, Shohei, Itano-gun, Tokushima, JP<br />
Tomikawa, Kenji, Tokushima-shi, Tokushima,<br />
JP<br />
(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />
Arabellastrasse 4, 81925 München, DE<br />
(60) 08000357.7 / 1 927 355<br />
08000358.5 / 1 925 308<br />
08000359.3 / 1 927 356<br />
08000360.1 / 1 927 357<br />
(62) 02782507.4 / 1 330 249<br />
A61K 31/496 → (51) C07D 231/12<br />
A61K 31/4965 → (51) C07D 403/02<br />
(51) A61K 31/501 (11) 1 363 636 B1<br />
A61K 33/06 A61P 9/04<br />
A61P 9/10<br />
(25) En (26) En