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Bulletin 2010/15 - European Patent Office

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(C07C) II.1(1)<br />

• SYNTHÈSE DES AGENTS DE MASSE DU<br />

TRITHIOCARBONATE ET DE LEURS<br />

SUBSTANCES INTERMÉDIAIRES<br />

(73) E.I. DU PONT DE NEMOURS AND COM-<br />

PANY, 1007 Market Street, Wilmington, DE<br />

19898, US<br />

(72) FARNHAM, William, Brown, Hockessin,<br />

Delaware 19707, US<br />

(74) Towler, Philip Dean, Dehns St Bride's House<br />

10 Salisbury Square, London EC4Y 8JD, GB<br />

(51) C07C 381/00 (11) 1 685 098 B1<br />

(25) De (26) De<br />

(21) 04818381.8 (22) 03.11.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LU MC NL PL PT RO SE SI<br />

SK TR<br />

LT LV MK<br />

(43) 02.08.2006<br />

(86) EP 2004/012394 03.11.2004<br />

(87) WO 2005/047240 2005/21 26.05.2005<br />

(30) 13.11.2003 DE 10353205<br />

(54) • ORTHO-SUBSTITUIERTE PENTAFLUOR-<br />

SULFANYL-BENZOLE, VERFAHREN ZU<br />

IHRER HERSTELLUNG SOWIE IHRE VER-<br />

WENDUNG AIS WERTVOLLE SYNTHESE-<br />

ZWISCHENSTUFEN<br />

• ORTHO-SUBSTITUTED PENTAFLUORIDE<br />

SULFANYL-BENZENES, METHOD FOR THE<br />

PRODUCTION THEREOF AND THE USE<br />

THEREOF IN THE FORM OF VALUABLE<br />

SYNTHESIS INTERMEDIATE STAGES<br />

• PENTAFLUOROSULFANYLBENZENES<br />

ORTHO-SUBSTITUES, LEUR PROCEDE DE<br />

PRODUCTION ET LEUR UTILISATION<br />

COMME INTERMEDIAIRES DE SYNTHESE<br />

PRECIEUX<br />

(73) Sanofi-Aventis Deutschland GmbH,<br />

Brüningstraße 50, 65929 Frankfurt am Main,<br />

DE<br />

(72) KLEEMANN, Heinz-Werner, 65474 Bischofsheim,<br />

DE<br />

WECK, Remo, 65779 Kelkheim, DE<br />

(51) C07D 201/16 (11) 1 167 350 B1<br />

(25) En (26) En<br />

(21) 01114770.9 (22) 25.06.2001<br />

(84) BE DE ES IT NL<br />

(43) 02.01.2002<br />

(30) 27.06.2000 JP 2000192350<br />

(54) • Verfahren zur Herstellung von epsilon-<br />

Caprolactam<br />

• Process for producing epsilon-caprolactam<br />

• Procédé pour la préparation d'epsiloncaprolactame<br />

(73) Sumitomo Chemical Company, Limited, 27-<br />

1, Shinkawa 2-chome, Chuo-ku, Tokyo 104-<br />

8260, JP<br />

(72) Shimazu, Yasumoto, Niihama-shi, Ehime, JP<br />

Umida, Horyuki, Niihama-shi, Ehime, JP<br />

Fukao, Masami, Ritto-cho, Kurita-gun, Shiga,<br />

JP<br />

(74) Vossius & Partner, Siebertstraße 4, 81675<br />

München, DE<br />

C07D 205/04 → (51) C07C 311/13<br />

C07D 207/04 → (51) C07C 317/30<br />

C07D 207/26 → (51) C07D 409/12<br />

C07D 207/48 → (51) C07C 311/13<br />

(51) C07D 209/08 (11) 1 951 668 B1<br />

(25) En (26) En<br />

(21) 06807752.8 (22) 06.11.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(43) 06.08.2008<br />

(86) EP 2006/068128 06.11.2006<br />

(87) WO 2007/057316 2007/21 24.05.2007<br />

(30) 16.11.2005 EP 05110786<br />

(54) • NEUES VERFAHREN ZUR HERSTELLUNG<br />

VON THOC<br />

• NOVEL PROCESS FOR THE PREPARATION<br />

OF THOC<br />

• NOUVEAU PROCEDE DE PREPARATION<br />

DE THOC<br />

(73) F.HOFFMANN-LA ROCHE AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) KNIPP, Bernhard, 5<strong>15</strong><strong>15</strong> Kuerten-Olpe, DE<br />

KUCZNIERZ, Ralf, 67098 Bad Duerkheim, DE<br />

SATTELKAU, Tim, 67065 Ludwigshafen, DE<br />

ZEIBIG, Thomas, 67122 Mutterstadt, DE<br />

(74) Heiroth, Ulrike Hildegard, F. Hoffmann-La<br />

Roche AG <strong>Patent</strong> Department, Grenzacherstrasse<br />

124, CH-4070 Basel, CH<br />

C07D 209/10 → (51) C07D 209/12<br />

(51) C07D 209/12 (11) 1 537 078 B1<br />

A61K 31/404 A61P 3/10<br />

C07D 401/04 C07D 209/36<br />

C07D 413/04 C07D 209/30<br />

C07D 401/06 C07D 405/06<br />

C07D 403/12 C07D 209/10<br />

(25) En (26) En<br />

(21) 03791952.9 (22) 27.08.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

LT LV<br />

(43) 08.06.2005<br />

(86) US 2003/027<strong>15</strong>6 27.08.2003<br />

(87) WO 2004/020409 2004/11 11.03.2004<br />

(30) 29.08.2002 US 406741 P<br />

17.01.2003 US 440672 P<br />

(54) • INDOLE MIT ANTIDIABETISCHER WIR-<br />

KUNG<br />

• INDOLES HAVING ANTI-DIABETIC ACTIV-<br />

ITY<br />

• INDOLES A ACTIVITE ANTIDIABETIQUE<br />

(73) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) ACTON, John, J., III, Rahway, NJ 07065-<br />

0907, US<br />

DEBENHAM, Sheryl, D., Rahway, NJ 07065-<br />

0907, US<br />

LIU, Kun, Rahway, NJ 07065-0907, US<br />

MEINKE, Peter, T., Rahway, NJ 07065-0907,<br />

US<br />

WOOD, Harold, B., Rahway, NJ 07065-0907,<br />

US<br />

BLACK, Regina, M., Rahway, NJ 07065-<br />

0907, US<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

(51) C07D 209/18 (11) 1 919 869 B1<br />

C07D 401/12 C07D 403/12<br />

C07D 405/12 A61K 31/405<br />

A61K 31/4<strong>15</strong>5 A61K 31/4178<br />

A61P 3/00 A61P 25/00<br />

C07D 413/12 C07D 413/14<br />

C07D 417/12 A61K 31/422<br />

A61K 31/427 A61K 31/433<br />

(25) Fr (26) Fr<br />

(21) 06808258.5 (22) 29.08.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 14.05.2008<br />

573<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>15</strong>/<strong>2010</strong>) 14.04.<strong>2010</strong><br />

(86) FR 2006/050818 29.08.2006<br />

(87) WO 2007/026097 2007/10 08.03.2007<br />

(30) 30.08.2005 FR 0508858<br />

(54) • INDOLDERIVATE ALS PPAR-AKTIVATO-<br />

REN<br />

• INDOLE DERIVATIVES AS PPAR ACTIVA-<br />

TORS<br />

• DÉRIVÉS DE L'INDOLE ACTIVATEURS DES<br />

PPAR<br />

(73) LABORATOIRES FOURNIER SA, 28, Boulevard<br />

Clémenceau, 21000 Dijon, FR<br />

(72) BINET, Jean, F-21121 Fontaine Les Dijon, FR<br />

BOUBIA, Benaïssa, F-21850 Saint Apollinaire,<br />

FR<br />

DODEY, Pierre, F-21121 Fontaine Les Dijon,<br />

FR<br />

LEGENDRE, Christiane, F-21370 Velard Sur<br />

Ouche, FR<br />

BARTH, Martine, F-21380 Asnieres Les<br />

Dijon, FR<br />

POUPARDIN-OLIVIER, Olivia, F-21490 Varois<br />

et Chaignot, FR<br />

(74) Hubert, Philippe, et al, Cabinet Beau de<br />

Loménie <strong>15</strong>8, rue de l'Université, 75340<br />

Paris Cédex 07, FR<br />

C07D 209/30 → (51) C07D 209/12<br />

C07D 209/36 → (51) C07D 209/12<br />

(51) C07D 209/40 (11) 1 335 901 B1<br />

C07D 217/06 C07D 409/12<br />

C07K 5/062 A61K 31/18<br />

A61P <strong>15</strong>/06<br />

(25) En (26) En<br />

(21) 01982432.5 (22) <strong>15</strong>.10.2001<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

AL LT LV RO SI<br />

(43) 20.08.2003<br />

(86) EP 2001/011865 <strong>15</strong>.10.2001<br />

(87) WO 2002/032864 2002/17 25.04.2002<br />

(30) 17.10.2000 EP 00122588<br />

(54) • PHARMAZEUTISCH AKTIVE SULFONAMID-<br />

DERIVATE<br />

• PHARMACEUTICALLY ACTIVE SULFANI-<br />

LIDE DERIVATIVES<br />

• DERIVES DE SULFANILIDE ACTIFS DU<br />

POINT DE VUE PHARMACEUTIQUE<br />

(73) Merck Serono SA, Centre Industriel, 1267<br />

Coinsins, Vaud, CH<br />

(72) QUATTROPANI, Anna, CH-1227 Carouge, CH<br />

SCHWARZ, Matthias, CH-1226 Thônex, CH<br />

JORAND-LEBRUN, Catherine, F-74270 Contamine-Sarzin,<br />

FR<br />

CHURCH, Dennis, CH-1291 Commugny, CH<br />

SCHEER, Alexander, CH-1290 Versoix, CH<br />

(74) Stevens, Ian Edward, et al, Potter Clarkson<br />

LLP Park View House 58 The Ropewalk,<br />

Nottingham NG1 5DD, GB<br />

C07D 209/44 → (51) C07C 311/13<br />

C07D 209/86 → (51) A61K 31/4439<br />

C07D 209/88 → (51) A61K 31/4439<br />

(51) C07D 211/14 (11) 1 627 871 B1<br />

C07D 211/70 C07D 211/62<br />

C07D 295/08 C07D 295/18<br />

C07D 295/22 A61K 31/451<br />

A61K 31/4545 A61K 31/495<br />

A61P 43/00 A61P 35/00<br />

A61P <strong>15</strong>/00 A61P 37/06<br />

A61P 25/28 A61P 17/00<br />

(25) Ja (26) En<br />

(21) 04731745.8 (22) 07.05.2004

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