Bulletin 2010/15 - European Patent Office
Bulletin 2010/15 - European Patent Office
Bulletin 2010/15 - European Patent Office
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(C07C) II.1(1)<br />
• SYNTHÈSE DES AGENTS DE MASSE DU<br />
TRITHIOCARBONATE ET DE LEURS<br />
SUBSTANCES INTERMÉDIAIRES<br />
(73) E.I. DU PONT DE NEMOURS AND COM-<br />
PANY, 1007 Market Street, Wilmington, DE<br />
19898, US<br />
(72) FARNHAM, William, Brown, Hockessin,<br />
Delaware 19707, US<br />
(74) Towler, Philip Dean, Dehns St Bride's House<br />
10 Salisbury Square, London EC4Y 8JD, GB<br />
(51) C07C 381/00 (11) 1 685 098 B1<br />
(25) De (26) De<br />
(21) 04818381.8 (22) 03.11.2004<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LU MC NL PL PT RO SE SI<br />
SK TR<br />
LT LV MK<br />
(43) 02.08.2006<br />
(86) EP 2004/012394 03.11.2004<br />
(87) WO 2005/047240 2005/21 26.05.2005<br />
(30) 13.11.2003 DE 10353205<br />
(54) • ORTHO-SUBSTITUIERTE PENTAFLUOR-<br />
SULFANYL-BENZOLE, VERFAHREN ZU<br />
IHRER HERSTELLUNG SOWIE IHRE VER-<br />
WENDUNG AIS WERTVOLLE SYNTHESE-<br />
ZWISCHENSTUFEN<br />
• ORTHO-SUBSTITUTED PENTAFLUORIDE<br />
SULFANYL-BENZENES, METHOD FOR THE<br />
PRODUCTION THEREOF AND THE USE<br />
THEREOF IN THE FORM OF VALUABLE<br />
SYNTHESIS INTERMEDIATE STAGES<br />
• PENTAFLUOROSULFANYLBENZENES<br />
ORTHO-SUBSTITUES, LEUR PROCEDE DE<br />
PRODUCTION ET LEUR UTILISATION<br />
COMME INTERMEDIAIRES DE SYNTHESE<br />
PRECIEUX<br />
(73) Sanofi-Aventis Deutschland GmbH,<br />
Brüningstraße 50, 65929 Frankfurt am Main,<br />
DE<br />
(72) KLEEMANN, Heinz-Werner, 65474 Bischofsheim,<br />
DE<br />
WECK, Remo, 65779 Kelkheim, DE<br />
(51) C07D 201/16 (11) 1 167 350 B1<br />
(25) En (26) En<br />
(21) 01114770.9 (22) 25.06.2001<br />
(84) BE DE ES IT NL<br />
(43) 02.01.2002<br />
(30) 27.06.2000 JP 2000192350<br />
(54) • Verfahren zur Herstellung von epsilon-<br />
Caprolactam<br />
• Process for producing epsilon-caprolactam<br />
• Procédé pour la préparation d'epsiloncaprolactame<br />
(73) Sumitomo Chemical Company, Limited, 27-<br />
1, Shinkawa 2-chome, Chuo-ku, Tokyo 104-<br />
8260, JP<br />
(72) Shimazu, Yasumoto, Niihama-shi, Ehime, JP<br />
Umida, Horyuki, Niihama-shi, Ehime, JP<br />
Fukao, Masami, Ritto-cho, Kurita-gun, Shiga,<br />
JP<br />
(74) Vossius & Partner, Siebertstraße 4, 81675<br />
München, DE<br />
C07D 205/04 → (51) C07C 311/13<br />
C07D 207/04 → (51) C07C 317/30<br />
C07D 207/26 → (51) C07D 409/12<br />
C07D 207/48 → (51) C07C 311/13<br />
(51) C07D 209/08 (11) 1 951 668 B1<br />
(25) En (26) En<br />
(21) 06807752.8 (22) 06.11.2006<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />
SE SI SK TR<br />
Europäisches <strong>Patent</strong>blatt<br />
<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />
<strong>Bulletin</strong> européen des brevets<br />
(43) 06.08.2008<br />
(86) EP 2006/068128 06.11.2006<br />
(87) WO 2007/057316 2007/21 24.05.2007<br />
(30) 16.11.2005 EP 05110786<br />
(54) • NEUES VERFAHREN ZUR HERSTELLUNG<br />
VON THOC<br />
• NOVEL PROCESS FOR THE PREPARATION<br />
OF THOC<br />
• NOUVEAU PROCEDE DE PREPARATION<br />
DE THOC<br />
(73) F.HOFFMANN-LA ROCHE AG, Grenzacherstrasse<br />
124, 4070 Basel, CH<br />
(72) KNIPP, Bernhard, 5<strong>15</strong><strong>15</strong> Kuerten-Olpe, DE<br />
KUCZNIERZ, Ralf, 67098 Bad Duerkheim, DE<br />
SATTELKAU, Tim, 67065 Ludwigshafen, DE<br />
ZEIBIG, Thomas, 67122 Mutterstadt, DE<br />
(74) Heiroth, Ulrike Hildegard, F. Hoffmann-La<br />
Roche AG <strong>Patent</strong> Department, Grenzacherstrasse<br />
124, CH-4070 Basel, CH<br />
C07D 209/10 → (51) C07D 209/12<br />
(51) C07D 209/12 (11) 1 537 078 B1<br />
A61K 31/404 A61P 3/10<br />
C07D 401/04 C07D 209/36<br />
C07D 413/04 C07D 209/30<br />
C07D 401/06 C07D 405/06<br />
C07D 403/12 C07D 209/10<br />
(25) En (26) En<br />
(21) 03791952.9 (22) 27.08.2003<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IT LI LU MC NL PT RO SE SI SK<br />
TR<br />
LT LV<br />
(43) 08.06.2005<br />
(86) US 2003/027<strong>15</strong>6 27.08.2003<br />
(87) WO 2004/020409 2004/11 11.03.2004<br />
(30) 29.08.2002 US 406741 P<br />
17.01.2003 US 440672 P<br />
(54) • INDOLE MIT ANTIDIABETISCHER WIR-<br />
KUNG<br />
• INDOLES HAVING ANTI-DIABETIC ACTIV-<br />
ITY<br />
• INDOLES A ACTIVITE ANTIDIABETIQUE<br />
(73) Merck Sharp & Dohme Corp., 126 East<br />
Lincoln Avenue, Rahway, NJ 07065, US<br />
(72) ACTON, John, J., III, Rahway, NJ 07065-<br />
0907, US<br />
DEBENHAM, Sheryl, D., Rahway, NJ 07065-<br />
0907, US<br />
LIU, Kun, Rahway, NJ 07065-0907, US<br />
MEINKE, Peter, T., Rahway, NJ 07065-0907,<br />
US<br />
WOOD, Harold, B., Rahway, NJ 07065-0907,<br />
US<br />
BLACK, Regina, M., Rahway, NJ 07065-<br />
0907, US<br />
(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />
& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />
Hertford Road, Hoddesdon Hertfordshire<br />
EN11 9BU, GB<br />
(51) C07D 209/18 (11) 1 919 869 B1<br />
C07D 401/12 C07D 403/12<br />
C07D 405/12 A61K 31/405<br />
A61K 31/4<strong>15</strong>5 A61K 31/4178<br />
A61P 3/00 A61P 25/00<br />
C07D 413/12 C07D 413/14<br />
C07D 417/12 A61K 31/422<br />
A61K 31/427 A61K 31/433<br />
(25) Fr (26) Fr<br />
(21) 06808258.5 (22) 29.08.2006<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />
SE SI SK TR<br />
AL BA HR MK RS<br />
(43) 14.05.2008<br />
573<br />
<strong>Patent</strong>e<br />
<strong>Patent</strong>s<br />
Brevets (<strong>15</strong>/<strong>2010</strong>) 14.04.<strong>2010</strong><br />
(86) FR 2006/050818 29.08.2006<br />
(87) WO 2007/026097 2007/10 08.03.2007<br />
(30) 30.08.2005 FR 0508858<br />
(54) • INDOLDERIVATE ALS PPAR-AKTIVATO-<br />
REN<br />
• INDOLE DERIVATIVES AS PPAR ACTIVA-<br />
TORS<br />
• DÉRIVÉS DE L'INDOLE ACTIVATEURS DES<br />
PPAR<br />
(73) LABORATOIRES FOURNIER SA, 28, Boulevard<br />
Clémenceau, 21000 Dijon, FR<br />
(72) BINET, Jean, F-21121 Fontaine Les Dijon, FR<br />
BOUBIA, Benaïssa, F-21850 Saint Apollinaire,<br />
FR<br />
DODEY, Pierre, F-21121 Fontaine Les Dijon,<br />
FR<br />
LEGENDRE, Christiane, F-21370 Velard Sur<br />
Ouche, FR<br />
BARTH, Martine, F-21380 Asnieres Les<br />
Dijon, FR<br />
POUPARDIN-OLIVIER, Olivia, F-21490 Varois<br />
et Chaignot, FR<br />
(74) Hubert, Philippe, et al, Cabinet Beau de<br />
Loménie <strong>15</strong>8, rue de l'Université, 75340<br />
Paris Cédex 07, FR<br />
C07D 209/30 → (51) C07D 209/12<br />
C07D 209/36 → (51) C07D 209/12<br />
(51) C07D 209/40 (11) 1 335 901 B1<br />
C07D 217/06 C07D 409/12<br />
C07K 5/062 A61K 31/18<br />
A61P <strong>15</strong>/06<br />
(25) En (26) En<br />
(21) 01982432.5 (22) <strong>15</strong>.10.2001<br />
(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />
LU MC NL PT SE TR<br />
AL LT LV RO SI<br />
(43) 20.08.2003<br />
(86) EP 2001/011865 <strong>15</strong>.10.2001<br />
(87) WO 2002/032864 2002/17 25.04.2002<br />
(30) 17.10.2000 EP 00122588<br />
(54) • PHARMAZEUTISCH AKTIVE SULFONAMID-<br />
DERIVATE<br />
• PHARMACEUTICALLY ACTIVE SULFANI-<br />
LIDE DERIVATIVES<br />
• DERIVES DE SULFANILIDE ACTIFS DU<br />
POINT DE VUE PHARMACEUTIQUE<br />
(73) Merck Serono SA, Centre Industriel, 1267<br />
Coinsins, Vaud, CH<br />
(72) QUATTROPANI, Anna, CH-1227 Carouge, CH<br />
SCHWARZ, Matthias, CH-1226 Thônex, CH<br />
JORAND-LEBRUN, Catherine, F-74270 Contamine-Sarzin,<br />
FR<br />
CHURCH, Dennis, CH-1291 Commugny, CH<br />
SCHEER, Alexander, CH-1290 Versoix, CH<br />
(74) Stevens, Ian Edward, et al, Potter Clarkson<br />
LLP Park View House 58 The Ropewalk,<br />
Nottingham NG1 5DD, GB<br />
C07D 209/44 → (51) C07C 311/13<br />
C07D 209/86 → (51) A61K 31/4439<br />
C07D 209/88 → (51) A61K 31/4439<br />
(51) C07D 211/14 (11) 1 627 871 B1<br />
C07D 211/70 C07D 211/62<br />
C07D 295/08 C07D 295/18<br />
C07D 295/22 A61K 31/451<br />
A61K 31/4545 A61K 31/495<br />
A61P 43/00 A61P 35/00<br />
A61P <strong>15</strong>/00 A61P 37/06<br />
A61P 25/28 A61P 17/00<br />
(25) Ja (26) En<br />
(21) 04731745.8 (22) 07.05.2004