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Bulletin 2010/15 - European Patent Office

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(C07D) I.1(1)<br />

• NOVEL COMPOUNDS 951: A BIPHENY-<br />

LOXYPROPANOIC ACID AS CRTH2 MOD-<br />

ULATOR AND INTERMEDIATES<br />

• NOUVEAUX COMPOSÉS 951: ACIDE<br />

BIPHÉNYLOXYPROPANOÏQUE UTILE<br />

COMME MODULATEUR DE CRTH2 ET<br />

INTERMÉDIAIRES<br />

(71) AstraZeneca AB, <strong>15</strong>1 85 Södertälje, SE<br />

(72) BONNERT, Roger, Victor, Loughborough<br />

Leicestershire LE11 5RH, GB<br />

LUKER, Timothy, Jon, Loughborough Leicestershire<br />

LE11 5RH, GB<br />

PATEL, Anil, Loughborough Leicestershire<br />

LE11 5RH, GB<br />

RIGBY, Aaron, Loughborough Leicestershire<br />

LE11 5RH, GB<br />

(51) C07D 301/12 (11) 2 173 731 A2*<br />

C07D 303/04<br />

(25) En (26) En<br />

(21) 08778059.9 (22) 04.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/062538 04.07.2008<br />

(87) WO 2009/008493 2009/03 <strong>15</strong>.01.2009<br />

(88) 16.04.2009<br />

(30) 10.07.2007 JP 2007180644<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

PROPYLENOXID<br />

• METHOD FOR PRODUCING PROPYLENE<br />

OXIDE<br />

• PROCÉDÉ DE FABRICATION D'OXYDE DE<br />

PROPYLÈNE<br />

(71) Sumitomo Chemical Company, Limited, 27-<br />

1, Shinkawa 2-chome Chuo-ku, Tokyo 104-<br />

8260, JP<br />

(72) MIZUNO, Masahiko, Nara-shi, Nara 630-<br />

8114, JP<br />

NARAHARA, Hideo, Ichihara-shi, Chiba 290-<br />

0142, JP<br />

(74) Vossius & Partner, Siebertstraße 4, 81675<br />

München, DE<br />

C07D 303/04 → (51) C07D 301/12<br />

(51) C07D 305/14 (11) 2 173 732 A2*<br />

A61K 31/33<br />

(25) En (26) En<br />

(21) 08781353.1 (22) 03.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/069192 03.07.2008<br />

(87) WO 2009/006590 2009/02 08.01.2009<br />

(88) 12.03.2009<br />

(30) 04.07.2007 IN CH14422007<br />

22.08.2007 IN CH18802007<br />

07.11.2007 US 986027 P<br />

17.03.2008 US 37162<br />

(54) • HERSTELLUNGSVERFAHREN FÜR DOCE-<br />

TAXEL UND POLYMORPHE<br />

• DOCETAXEL PROCESS AND POLY-<br />

MORPHS<br />

• PROCÉDÉS DE PRÉPARATION DE DOCÉ-<br />

TAXEL ET DE POLYMORPHES<br />

(71) Dr. Reddy's Laboratories Ltd., 7-1-27<br />

Ameerpet, Hyderabad 500 016, Andhra<br />

Pradesh, IN<br />

Dr. Reddy's Laboratories, Inc., 200 Somerset<br />

Corporate Boulevard 7th Floor, Bridgewater,<br />

NJ 08807, US<br />

(72) PALLE, Raghavendracharyulu, Venkata, 500<br />

050, Andhra Pradesh, IN<br />

NARIYAM, Sekhar Munaswamy, 500 072,<br />

Andhra Pradesh, IN<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

KADABOINA, Rajasekhar, Andhra Pradesh,<br />

IN<br />

MATTI, Lankeshwararao, 500 049 Andhra<br />

Pradesh, IN<br />

VASAM, Sridhar, 506 330, Andhra Pradesh,<br />

IN<br />

KOMATI, Shravan, Kumar, 508 205, Andhra<br />

Pradesh, IN<br />

MAKIREDDY, Siva, Reddy, 522 403, Andhra<br />

Pradesh, IN<br />

(74) Bates, Philip Ian, Reddie & Grose 16<br />

Theobalds Road, London WC1X 8PL, GB<br />

C07D 307/92 → (51) C09B 47/00<br />

(51) C07D 313/08 (11) 2 173 733 A2*<br />

C07D 321/10 C07D 327/02<br />

A61K 31/365 A61K 31/39<br />

A61P 25/00 A61P 29/00<br />

A61P 31/04 A61P 35/00<br />

(25) En (26) En<br />

(21) 08807<strong>15</strong>6.8 (22) 05.06.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) IB 2008/002497 05.06.2008<br />

(87) WO 2008/149244 2008/50 11.12.2008<br />

(88) 12.03.2009<br />

(30) 05.06.2007 US 933171 P<br />

(54) • ZUSAMMENSETZUNGEN UND VERFAH-<br />

REN MIT ANALOGEN VON RADICICOL A<br />

• COMPOSITIONS AND METHODS COM-<br />

PRISING ANALOGUES OF RADICICOL A<br />

• COMPOSITIONS ET PROCÉDÉS COMPRE-<br />

NANT DES ANALOGUES DE RADICICOL A<br />

(71) WINSSINGER, Nicolas, 30 Rue Jean-Jaques<br />

Rousseau, 67000 Strasbourg, FR<br />

BARLUENGA, Sofia, 30 Rue Jean-Jaques<br />

Rousseau, 67000 Strasburg, FR<br />

(72) WINSSINGER, Nicolas, 67000 Strasbourg,<br />

FR<br />

BARLUENGA, Sofia, 67000 Strasburg, FR<br />

(74) Gallois, Valérie, Cabinet BECKER & ASS-<br />

OCIES 25, rue Louis Le Grand, 75002 Paris,<br />

FR<br />

C07D 321/10 → (51) C07D 313/08<br />

C07D 327/02 → (51) C07D 313/08<br />

C07D 333/08 → (51) C07C 201/12<br />

C07D 333/10 → (51) C07D 263/32<br />

C07D 333/24 → (51) C07D 213/127<br />

(51) C07D 401/04 (11) 2 173 734 A2*<br />

C07D 403/04 C07D 417/04<br />

A61K 31/4192 A61K 31/427<br />

A61K 31/4439 A61K 31/506<br />

A61P 35/00 C07D 401/14<br />

C07D 403/14 C07D 417/14<br />

C07D 487/08<br />

(25) En (26) En<br />

(21) 08774579.0 (22) 01.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/058433 01.07.2008<br />

(87) WO 2009/003999 2009/02 08.01.2009<br />

(88) 16.07.2009<br />

(30) 02.07.2007 EP 0711<strong>15</strong>66<br />

(54) • CHEMISCHE VERBINDUNGEN<br />

• CHEMICAL COMPOUNDS<br />

• COMPOSÉS CHIMIQUES<br />

98<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>15</strong>/<strong>2010</strong>) 14.04.<strong>2010</strong><br />

(71) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim, DE<br />

(72) SAPOUNTZIS, Ioannis, 55216 Ingelheim Am<br />

Rhein, DE<br />

ETTMAYER, Peter, 55216 Ingelheim Am<br />

Rhein, DE<br />

KLEIN, Christian, 55216 Ingelheim Am<br />

Rhein, DE<br />

MANTOULIDIS, Andreas, 55216 Ingelheim<br />

Am Rhein, DE<br />

STEURER, Steffen, 55216 Ingelheim Am<br />

Rhein, DE<br />

WAIZENEGGER, Irene, 55216 Ingelheim Am<br />

Rhein, DE<br />

(74) Hammann, Heinz, Boehringer Ingelheim<br />

GmbH CD-<strong>Patent</strong>s Binger Straße 173, 55216<br />

Ingelheim am Rhein, DE<br />

C07D 401/04 → (51) C07D 235/08<br />

C07D 401/04 → (51) C07D 263/48<br />

(51) C07D 401/06 (11) 2 173 735 A1*<br />

C07D 401/14 C07D 403/06<br />

C07D 405/14 A61K 31/4178<br />

A61K 31/4439 A61P 9/00<br />

(25) En (26) En<br />

(21) 08774212.8 (22) 23.06.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/057934 23.06.2008<br />

(87) WO 2009/003861 2009/02 08.01.2009<br />

(30) 02.07.2007 EP 0711<strong>15</strong>52<br />

(54) • IMIDAZOLDERIVATE ALS CCR2-REZEP-<br />

TOR-ANTAGONISTEN<br />

• IMIDAZOLE DERIVATIVES AS CCR2<br />

RECEPTOR ANTAGONISTS<br />

• DÉRIVÉS IMIDAZOLÉS COMME ANTAGO-<br />

NISTES DU RÉCEPTEUR CCR2<br />

(71) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) AEBI, Johannes, CH-4102 Binningen, CH<br />

BINGGELI, Alfred, CH-4102 Binningen, CH<br />

GREEN, Luke, CH-4057 Basel, CH<br />

HARTMANN, Guido, 79539 Loerrach, DE<br />

MAERKI, Hans P., CH-4059 Basel, CH<br />

MATTEI, Patrizio, CH-4125 Riehen, CH<br />

RICKLIN, Fabienne, F-68490 Hombourg, FR<br />

ROCHE, Olivier, F-68220 Folgensbourg, FR<br />

(74) Heiroth, Ulrike Hildegard, F. Hoffmann-La<br />

Roche AG <strong>Patent</strong> Department, Grenzacherstrasse<br />

124, CH-4070 Basel, CH<br />

(51) C07D 401/06 (11) 2 173 736 A2*<br />

(25) En (26) En<br />

(21) 08793030.1 (22) 04.08.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) KR 2008/004516 04.08.2008<br />

(87) WO 2009/020323 2009/07 12.02.2009<br />

(88) 09.04.2009<br />

(30) 06.08.2007 KR 20070078439<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

VORICONAZOL<br />

• PROCESS FOR PREPARING VORICONA-<br />

ZOLE<br />

• PROCÉDÉ SERVANT À PRÉPARER DU<br />

VORICONAZOLE<br />

(71) Hanmi Pharm. Co., Ltd., 893-5 Hajeo-ri<br />

Paltan-myeon Hwaseong-si, Gyeonggi-do<br />

445-910, KR<br />

(72) MOON, Young Ho, Suwon-si Gyeonggi-do<br />

442-470, KR

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