Bulletin 2010/15 - European Patent Office
Bulletin 2010/15 - European Patent Office
Bulletin 2010/15 - European Patent Office
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(C07D) I.1(1)<br />
C07D 231/56 → (51) C07D 213/127<br />
(51) C07D 233/06 (11) 2 173 719 A1*<br />
C07D 233/12 C07D 233/22<br />
C07D 233/24 A61K 31/4174<br />
A61P 25/24<br />
(25) En (26) En<br />
(21) 08774237.5 (22) 24.06.2008<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MT NL<br />
NO PL PT RO SE SI SK TR<br />
AL BA MK RS<br />
(86) EP 2008/057980 24.06.2008<br />
(87) WO 2009/003867 2009/02 08.01.2009<br />
(30) 03.07.2007 EP 07111623<br />
(54) • 4-IMIDAZOLINE UND IHRE VERWENDUNG<br />
ALS ANTIDEPRESSIVA<br />
• 4-IMIDAZOLINES AND THEIR USE AS<br />
ANTIDEPRESSANTS<br />
• 4-IMIDAZOLINES ET LEUR UTILISATION<br />
COMME ANTIDÉPRESSEURS<br />
(71) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />
124, 4070 Basel, CH<br />
(72) GALLEY, Guido, 79618 Rheinfelden, DE<br />
GROEBKE ZBINDEN, Katrin, CH-4410 Liestal,<br />
CH<br />
NORCROSS, Roger, CH-4305 Olsberg, CH<br />
STALDER, Henri, CH-4055 Basel, CH<br />
(74) Poppe, Regina, F.Hoffmann-La Roche AG<br />
<strong>Patent</strong> Department Grenzacherstrasse 124,<br />
4070 Basel, CH<br />
(51) C07D 233/10 (11) 2 173 720 A2*<br />
C07D 233/20 C07D 233/22<br />
C07D 233/24 C07D 233/42<br />
C07D 233/50 C07D 233/52<br />
C07D 405/12 A61K 31/4<strong>15</strong><br />
A61K 31/4<strong>15</strong>5 A61P 25/00<br />
(25) En (26) En<br />
(21) 08761316.2 (22) 24.06.2008<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MT NL<br />
NO PL PT RO SE SI SK TR<br />
AL BA MK RS<br />
(86) EP 2008/057989 24.06.2008<br />
(87) WO 2009/003868 2009/02 08.01.2009<br />
(88) 09.04.2009<br />
(30) 02.07.2007 EP 0711<strong>15</strong>58<br />
(54) • 2-IMIDAZOLINE MIT GUTER AFFINITÄT ZU<br />
TRACE-AMINE-ASSOCIATED-REZEPT-<br />
OREN (TAARS)<br />
• 2-IMIDAZOLINES HAVING A GOOD AFFI-<br />
NITY TO THE TRACE AMINE ASSOCIATED<br />
RECEPTORS (TAARS)<br />
• 2-IMIDAZOLINES<br />
(71) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />
124, 4070 Basel, CH<br />
(72) GALLEY, Guido, 79618 Rheinfelden, DE<br />
GROEBKE ZBINDEN, Katrin, CH-4410 Liestal,<br />
CH<br />
NORCROSS, Roger, CH-4305 Olsberg, CH<br />
STALDER, Henri, CH-4055 Basel, CH<br />
(74) Poppe, Regina, F.Hoffmann-La Roche AG<br />
<strong>Patent</strong> Department Grenzacherstrasse 124,<br />
4070 Basel, CH<br />
C07D 233/12 → (51) C07D 233/06<br />
C07D 233/20 → (51) C07D 233/10<br />
C07D 233/22 → (51) C07D 233/06<br />
C07D 233/22 → (51) C07D 233/10<br />
C07D 233/24 → (51) C07D 233/06<br />
Europäisches <strong>Patent</strong>blatt<br />
<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />
<strong>Bulletin</strong> européen des brevets<br />
C07D 233/24 → (51) C07D 233/10<br />
C07D 233/42 → (51) C07D 233/10<br />
C07D 233/50 → (51) C07D 233/10<br />
C07D 233/52 → (51) C07D 233/10<br />
C07D 233/60 → (51) C07D 405/06<br />
C07D 233/90 → (51) C07D 213/81<br />
(51) C07D 235/08 (11) 2 173 721 A1*<br />
C07D 235/16 C07D 235/18<br />
C07D 401/04 C07D 471/04<br />
(25) En (26) En<br />
(21) 08759<strong>15</strong>8.2 (22) 11.06.2008<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MT NL<br />
NO PL PT RO SE SI SK TR<br />
AL BA MK RS<br />
(86) EP 2008/004639 11.06.2008<br />
(87) WO 2009/000413 2009/01 31.12.2008<br />
(30) 26.06.2007 EP 07290800<br />
(54) • REGIOSELEKTIVE, KUPFERKATALYSIERTE<br />
SYNTHESE VON BENZIMIDAZOLEN UND<br />
AZABENZIMIDAZOLEN<br />
• A REGIOSELECTIVE COPPER CATALYZED<br />
SYNTHESIS OF BENZIMIDAZOLES AND<br />
AZABENZIMIDAZOLES<br />
• SYNTHÈSE RÉGIOSÉLECTIVE CATALYSÉE<br />
PAR LE CUIVRE DE BENZIMIDAZOLES ET<br />
D'AZABENZIMIDAZOLES<br />
(71) Sanofi-Aventis, 174 Avenue de France,<br />
75013 Paris, FR<br />
(72) ALONSO, Jorge, 68163 Mannheim, DE<br />
LINDENSCHMIDT, Andreas, 65926 Frankfurt<br />
am Main, DE<br />
NAZARÉ, Marc, 65926 Frankfurt am Main,<br />
DE<br />
URMANN, Matthias, 65926 Frankfurt am<br />
Main, DE<br />
HALLAND, Nis, 65926 Frankfurt am Main, DE<br />
R'KYEK, Omar, Tangier, MA<br />
(74) Then, Johann, et al, Sanofi-Aventis<br />
Deutschland GmbH <strong>Patent</strong>- und Lizenzabteilung<br />
Industriepark Höchst Gebäude K 801,<br />
65926 Frankfurt am Main, DE<br />
C07D 235/16 → (51) C07D 235/08<br />
C07D 235/18 → (51) C07D 235/08<br />
C07D 239/26 → (51) C07D 213/127<br />
(51) C07D 239/34 (11) 2 173 722 A2*<br />
C07D 239/42 C07D 401/12<br />
C07D 403/04 C07D 403/10<br />
C07D 405/10 C07D 419/12<br />
A61K 31/506 A61P 35/00<br />
(25) En (26) En<br />
(21) 08775347.1 (22) 24.07.2008<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MT NL<br />
NO PL PT RO SE SI SK TR<br />
AL BA MK RS<br />
(86) EP 2008/059748 24.07.2008<br />
(87) WO 2009/013348 2009/05 29.01.2009<br />
(88) 23.07.2009<br />
(30) 26.07.2007 EP 07113237<br />
(54) • ZUR BEHANDLUNG VON ENTZÜNDLICHEN<br />
ODER ALLERGISCHEN LEIDEN GEEIG-<br />
NETE PYRIMIDINDERIVATE<br />
• PYRIMIDINE DERIVATIVES USEFUL FOR<br />
THE TREATMENT OF INFLAMMATORY OR<br />
ALLERGIC CONDITIONS<br />
96<br />
Anmeldungen<br />
Applications<br />
Demandes (<strong>15</strong>/<strong>2010</strong>) 14.04.<strong>2010</strong><br />
• DÉRIVÉS DE PYRIMIDINES POUR LE<br />
TRAITEMENT DE MALADIES INFLAMM-<br />
MATOIRES ET ALLERGIQUES<br />
(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />
(72) BRUCE, Ian, Horsham, West Sussex RH12<br />
5AB, GB<br />
DUNSTAN, Andrew, Horsham, West Sussex<br />
RH12 5AB, GB<br />
HUNT, Thomas Anthony, Horsham, West<br />
Sussex RH12 5AB, GB<br />
HOWSHAM, Catherine, Horsham, West Sussex<br />
RH12 5AB, GB<br />
(74) Vögeli-Lange, Regina, Novartis Pharma AG<br />
<strong>Patent</strong> Department, 4002 Basel, CH<br />
C07D 239/42 → (51) C07D 239/34<br />
(51) C07D 239/70 (11) 2 173 723 A1*<br />
A61K 31/517 A61P 35/00<br />
(25) En (26) En<br />
(21) 08781340.8 (22) 03.07.2008<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MT NL<br />
NO PL PT RO SE SI SK TR<br />
AL BA MK RS<br />
(86) US 2008/069147 03.07.2008<br />
(87) WO 2009/006569 2009/02 08.01.2009<br />
(30) 05.07.2007 US 948147 P<br />
(54) • PYRIMIDYLCYCLOPENTANE ALS INHIBI-<br />
TOREN DER AKT-PROTEINKINASE<br />
• PYRIMIDYL CYCLOPENTANES AS AKT<br />
PROTEIN KINASE INHIBITORS<br />
• PYRIMIDYL CYCLOPENTANES UTILSÉS<br />
COMME INHIBITEURS DE LA PROTÉINE<br />
KINASE AKT<br />
(71) Array Biopharma, Inc., 3200 Walnut Street,<br />
Boulder, CO 80301, US<br />
Genentech, Inc., 1 DNA Way, South San<br />
Francisco CA 94080-4990, US<br />
(72) BENCSIK, Josef, R., Longmont, CO 80501,<br />
US<br />
BLAKE, James, F., Longmont, CO 80504, US<br />
KALLAN, Nicholas, C., Boulder, CO 80301,<br />
US<br />
MITCHELL, Ian, S., Lafayette, CO 80026, US<br />
SPENCER, Keith, L., Lyons, CO 80540, US<br />
XIAO, Dengming, Longmont, CO 80501, US<br />
XU, Rui, Longmont, CO 80501, US<br />
CHABOT, Christine, San Mateo, CA 94402,<br />
US<br />
LIANG, Jun, Palo Alto, CA 94306, US<br />
SAFINA, Brian, S., Redwood City, CA 94061,<br />
US<br />
(74) Bailey, Sam Rogerson, et al, Mewburn Ellis<br />
LLP 33 Gutter Lane, London EC2V 8AS, GB<br />
C07D 239/70 → (51) A61K 31/517<br />
(51) C07D 239/90 (11) 2 173 724 A2*<br />
A61K 31/517 A61P 35/00<br />
(25) En (26) En<br />
(21) 0877<strong>15</strong>27.2 (22) 19.06.2008<br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HR HU IE IS IT LI LT LU LV MC MT NL<br />
NO PL PT RO SE SI SK TR<br />
AL BA MK RS<br />
(86) US 2008/067571 19.06.2008<br />
(87) WO 2009/002808 2009/01 31.12.2008<br />
(88) 23.07.2009<br />
(30) 22.06.2007 US 945838 P<br />
(54) • CHINAZOLINONVERBINDUNGEN UND<br />
VERFAHREN ZU IHRER ANWENDUNG<br />
• QUINAZOLINONE COMPOUNDS AND<br />
METHODS OF USE THEREOF<br />
• COMPOSÉS DE QUINAZOLINONE ET<br />
LEURS MÉTHODES D'UTILISATION<br />
(71) ArQule, Inc., 19 Presidential Way, Woburn,<br />
MA 01801, US
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