Bulletin 2010/15 - European Patent Office

(C07C) II.1(1)
C07C 209/78 → (51) C07C 209/54
C07C 209/86 → (51) B01D 3/14
C07C 211/21 → (51) C07C 209/62
C07C 211/45 → (51) C07C 209/62
C07C 211/50 → (51) C07C 209/54
(51) C07C 233/57 (11) 1 685 093 B1
(25) En (26) En
(21) 04761978.8 (22) 28.10.2004
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IT LI LU MC NL PL PT RO SE SI SK
TR
(43) 02.08.2006
(86) CH 2004/000646 28.10.2004
(87) WO 2005/049553 2005/22 02.06.2005
(30) 21.11.2003 US 523977 P
(54) • N-SUBSTITUIERTE P-MENTHANCARBON-
SÄUREAMIDE
• N-SUBSTITUTED P-MENTHANE CARBO-
SAMIDED
• CARBOXAMIDES P-MENTHANE A SUB-
STITUTION N
(73) Givaudan SA, Chemin de la Parfumerie 5,
1214 Vernier, CH
(72) GALOPIN, Christophe, Chesterfield, Virginia
23833, US
KRAWEC, Pablo, Victor, Cincinnati, Ohio
45249, US
SLACK, Jay, Patrick, Loveland, Ohio 45140,
US
TIGANI, Lori, Salisbury, MD 21801, US
(74) Givaudan Patents, Ueberlandstrasse 138,
8600 Dubendorf, CH
(51) C07C 235/24 (11) 1 641 745 B1
C07C 255/58 C07D 213/68
A61K 31/395 A61K 31/277
A61K 31/167 A61P 5/26
A61P 15/16
(25) En (26) En
(21) 04742130.0 (22) 24.06.2004
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IT LI LU MC NL PL PT RO SE SI SK
TR
AL LT LV MK
(43) 05.04.2006
(86) FI 2004/000387 24.06.2004
(87) WO 2005/000794 2005/01 06.01.2005
(30) 27.06.2003 US 482713 P
27.06.2003 FI 20030958
(54) • ALS ANDROGENREZEPTORMODULATO-
REN GEEIGNETE PROPIONAMIDDERIVATE
• PROPIONAMIDE DERIVATIVES USEFUL
AS ANDROGEN RECEPTOR MODULATORS
• DERIVES DE PROPIONAMIDE UTILISES
COMME MODULATEURS DU RECEPTEUR
D'ANDROGENES
(73) ORION CORPORATION, Orionintie 1, 02200
Espoo, FI
(72) RATILAINEN, Jari, FI-80910 Kulho, FI
MOILANEN, Anu, FI-20720 Turku, FI
TÖRMÄKANGAS, Olli, FI-20380 Turku, FI
KARJALAINEN, Arja, FI-02210 Espoo, FI
HUHTALA, Paavo, FI-02200 Espoo, FI
WOHLFAHRT, Gerd, FI-00210 Helsinki, FI
KALLIO, Pekka, FI-20720 Turku, FI
(74) Sexton, Jane Helen, J.A. Kemp & Co. 14
South Square Gray's Inn, London WC1R 5JJ,
GB
(51) C07C 253/30 (11) 1 501 788 B1
C07C 255/56
(25) De (26) De
(21) 03720529.1 (22) 25.04.2003
Europäisches Patentblatt
European Patent Bulletin
Bulletin européen des brevets
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IT LI LU MC NL PT RO SE SI SK
TR
(43) 02.02.2005
(86) EP 2003/004327 25.04.2003
(87) WO 2003/091203 2003/45 06.11.2003
(30) 26.04.2002 DE 10218764
(54) • VERFAHREN ZUR HERSTELLUNG VON 3-
TRIFLUORMETHYLPHENYL-4-CYANOBEN-
ZYLKETON
• METHOD FOR PRODUCING 3-TRIFLUOR-
OMETHYLPHENYL-4-CYANOBENZYL
KETONE
• PROCEDE POUR PRODUIRE DE LA
CETONE 3-TRIFLUOROMETHYLE PHE-
NYLE-4-CYANOBENZYLE
(73) BASF SE, 67056 Ludwigshafen, DE
(72) ENGEL, Stefan, 55268 Nieder-Olm, DE
KEIL, Michael, 67251 Freinsheim, DE
OTT, Christian, 67346 Speyer, DE
RACK, Michael, 69123 Heidelberg, DE
C07C 255/56 → (51) C07C 253/30
C07C 255/58 → (51) C07C 235/24
(51) C07C 311/13 (11) 1 694 410 B1
C07D 205/04 C07D 207/48
C07D 209/44 C07D 211/58
C07D 213/18 C07D 217/08
C07D 231/12 C07D 233/64
C07D 237/12 C07D 239/22
C07D 243/08 C07D 257/04
C07D 261/08 C07D 271/06
C07D 277/26 C07D 295/26
C07D 307/79 C07D 333/18
A61K 31/18 A61P 19/02
(25) En (26) En
(21) 04814080.0 (22) 14.12.2004
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IS IT LI LT LU MC NL PL PT RO SE
SI SK TR
AL BA HR LV MK YU
(43) 30.08.2006
(86) US 2004/041852 14.12.2004
(87) WO 2005/058884 2005/26 30.06.2005
(30) 15.12.2003 US 529116 P
(54) • CYCLOPROPANDERIVATE UND IHRE
PHARMAZEUTISCHE VERWENDUNG
• CYCLOPROPANE DERIVATIVES AND
PHARMACEUTICAL USE THEREOF
• DERIVES DE CYCLOPROPANE ET UTILI-
SATION PHARMACEUTIQUE DE CEUX-CI
(73) Japan Tobacco, Inc., 2-1, Toranomon 2chome,
Minato-ku, Tokyo 105-8422, JP
(72) INABA, Takashi, c/o Japan Tobacco Inc.
Central Pharmaceutical Research Institute,
Osaka 569-1125, JP
HAAS, Julia, Boulder, CO 80302, US
SHIOZAKI, Makoto, c/o Japan Tobacco Inc.
Central Pharmaceutical Research Institute,
Osaka 569-1125, JP
LITTMAN, Nicole, M., Erie, CO 08516, US
YASUE, Katsutaka, c/o Japan Tobacco Inc.
Central Pharmaceutical Research Institute,
Osaka 569-1125, JP
ANDREWS, Steven, W., Longmont, CO
80501, US
SAKAI, Atushi, c/o Japan Tobacco Inc.
Central Pharmaceutical Research Institute,
Osaka 569-1125, JP
FRYER, Andrew, M., Erie, CO 80516, US
MATSUO, Takafumi, c/o Japan Tobacco Inc.
Central Pharmaceutical Research Institute,
Osaka 569-1125, JP
LAIRD, Ellen, R., Longmont, CO 80504, US
572
Patente
Patents
Brevets (15/2010) 14.04.2010
SUMA, Akira, c/o Japan Tobacco Inc. Central
Pharmaceutical Research Institute, Osaka
569-1125, JP
SHINOZAKI, Yuichi, c/o Japan Tobacco Inc.
Central Pharmaceutical Research Institute,
Osaka 569-1125, JP
MORI, Yoshikazu, c/o Japan Tobacco Inc.
Central Pharmaceutical Research Institute,
Osaka 569-1125, JP
IMAI, Hiroto, c/o Japan Tobacco Inc. Central
Pharmaceutical Research Institute, Osaka
569-1125, JP
NEGORO, Tamotsu, c/o Japan Tobacco Inc.
Central Pharmaceutical Research Institute,
Osaka 569-1125, JP
(74) Vossius & Partner, Siebertstraße 4, 81675
München, DE
(51) C07C 317/30 (11) 1 551 799 B1
C07D 213/71 C07D 295/10
C07D 207/04 A61K 31/10
A61P 25/28
(25) En (26) En
(21) 03750987.4 (22) 25.09.2003
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IT LI LU MC NL PT RO SE SI SK
TR
LT LV
(43) 13.07.2005
(86) GB 2003/004196 25.09.2003
(87) WO 2004/031139 2004/16 15.04.2004
(30) 04.10.2002 GB 0223038
(54) • CYCLOHEXYL-SULPHONE ALS GAMMA-
SEKRETASE-INHIBITOREN
• CYCLOHEXYL SULPHONES AS GAMMA-
SECRETASE INHIBITORS
• SULFONES CYCLOHEXYLIQUES TELS QUE
DES INHIBITEURS DE GAMMA-SECRE-
TASE
(73) MERCK SHARP & DOHME LTD., Hertford
Road, Hoddesdon, Hertfordshire EN11 9BU,
GB
(72) CHURCHER, Ian, Harlow,Essex CM20 2QR,
GB
HARRISON, Timothy, Harlow, Essex CM20
2QR, GB
KERRAD, Sonia, Harlow,Essex CM20 2QR,
GB
NADIN, Alan John, Harlow, Essex CM20
2QR, GB
OWENS, Andrew, Pate, Harlow, Essex CM20
2QR, GB
SHAW, Duncan Edward, Harlow, Essex
CM20 2QR, GB
THOMSON, Joanne, Harlow, Essex CM20
2QR, GB
WILLIAMS, Susannah, Harlow, Essex CM20
2QR, GB
(74) Buchan, Gavin MacNicol, et al, Merck Sharp
& Dohme Limited European Patent Department
Hertford Road, Hoddesdon Hertfordshire
EN11 9BU, GB
(51) C07C 329/00 (11) 1 745 017 B1
(25) En (26) En
(21) 05750365.8 (22) 11.05.2005
(84) DE FR GB
(43) 24.01.2007
(86) US 2005/016584 11.05.2005
(87) WO 2005/113493 2005/48 01.12.2005
(30) 12.05.2004 US 570150 P
(54) • SYNTHESE VON TRITHIOCARBONAT-
RAFT-AGENTIA UND ZWISCHENPRO-
DUKTE DARAUS
• SYNTHESIS OF TRITHIOCARBONATE
RAFT GENTS AND INTERMEDIATES
THEREOF