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Bulletin 2010/15 - European Patent Office

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(A61K) I.1(1)<br />

(74) Suarez-Miles, Ana Sanchiz, Eli Lilly and<br />

Company Limited <strong>European</strong> <strong>Patent</strong> Operations<br />

Lilly Research Centre, Erl Wood Manor<br />

Sunninghill Road, Windlesham, Surrey GU20<br />

6PH, GB<br />

(51) A61K 31/4745 (11) 2 173 349 A2*<br />

A61K 38/16 A61P 35/00<br />

(25) Fr (26) Fr<br />

(21) 08827826.2 (22) 02.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) FR 2008/000943 02.07.2008<br />

(87) WO 2009/024667 2009/09 26.02.2009<br />

(88) 23.04.2009<br />

(30) 05.07.2007 FR 0704868<br />

(54) • ANTITUMOR-KOMBINATIONEN MIT EINEM<br />

VEGF-HEMMENDEN MITTEL UND IRINO-<br />

TECAN<br />

• ANTITUMOUR COMBINATIONS CONTAIN-<br />

ING A VEGF INHIBITING AGENT AND<br />

IRINOTECAN<br />

• COMBINAISONS ANTITUMORALES<br />

CONTENANT UN AGENT INHIBITEUR DE<br />

VEGF ET DE L'IRINOTECAN<br />

(71) Aventis Pharma S.A., 20, avenue Raymond<br />

Aron, 92160 Antony, FR<br />

(72) BISSERY, Marie-Christine, F-75013 Paris, FR<br />

CHIRON-BLONDEL, Marielle, F-75013 Paris,<br />

FR<br />

LEJEUNE, Pascale, F-75013 Paris, FR<br />

VRIGNAUD, Patricia, F-75013 Paris, FR<br />

(74) Le Pennec, Magali, et al, Sanofi-Aventis<br />

Direction Brevets 174 Avenue de France,<br />

75013 Paris, FR<br />

A61K 31/4985 → (51) A61K 31/4745<br />

(51) A61K 31/505 (11) 2 173 350 A2*<br />

C07D 473/00 C07D 405/04<br />

(25) En (26) En<br />

(21) 08782336.5 (22) 24.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/071069 24.07.2008<br />

(87) WO 2009/018106 2009/06 05.02.2009<br />

(88) 12.03.2009<br />

(30) 30.07.2007 US 962550 P<br />

(54) • STEREOSELEKTIVES VERFAHREN ZUR<br />

HERSTELLUNG VON PURINDIOXOLAN-<br />

NUKLEOSIDE-DERIVATEN<br />

• STEREOSELECTIVE PROCESS FOR PRE-<br />

PARING PURINE DIOXOLANE NUCLEO-<br />

SIDE DERIVATIVES<br />

• PROCÉDÉ STÉRÉOSÉLECTIF POUR PRÉ-<br />

PARER DES DÉRIVÉS DE PURINE DIOXO-<br />

LANE NUCLÉOSIDE<br />

(71) RFS Pharma, LLC., 1860 Montreal Road,<br />

Tucker GA 30084, US<br />

(72) COATS, Steven, J., Mcdonough, GA 30252,<br />

US<br />

(74) Harrison Goddard Foote, 106 Hope Street,<br />

Glasgow G2 6PH, GB<br />

(51) A61K 31/506 (11) 2 173 351 A2*<br />

A61K 31/7064 A61P 7/00<br />

A61P 37/06<br />

(25) En (26) En<br />

(21) 08794556.4 (22) 16.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(86) US 2008/008745 16.07.2008<br />

(87) WO 2009/011889 2009/04 22.01.2009<br />

(88) 05.03.2009<br />

(30) 18.07.2007 US 959984 P<br />

(54) • VERBINDUNG UND VERFAHREN ZUR<br />

BEHANDLUNG VON SICHELZELLENANÄ-<br />

MIE ODER DAMIT VERBUNDENEN KOM-<br />

PLIKATIONEN<br />

• COMPOUNDS AND METHODS FOR<br />

TREATMENT OF SICKLE CELL DISEASE<br />

OR COMPLICATIONS ASSOCIATED<br />

THEREWITH<br />

• COMPOSES ET METHODES DE TRAITE-<br />

MENT DE LA DREPANOCYTOSE OU DE<br />

SES COMPLICATIONS<br />

(71) GlycoMimetics, Inc., 101 Orchard Ridge<br />

Drive, Suite 1E, Gaithersburg, MD 20878, US<br />

(72) MAGNANI, John, L., Gaithersburg, MD<br />

20878, US<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

A61K 31/506 → (51) C07D 239/34<br />

A61K 31/506 → (51) C07D 401/04<br />

A61K 31/513 → (51) A61K 31/4745<br />

A61K 31/513 → (51) C07D 403/06<br />

(51) A61K 31/517 (11) 2 173 352 A2*<br />

A61K 31/53 A61K 31/136<br />

C07D 211/00 C07D 239/70<br />

(25) En (26) En<br />

(21) 08772544.6 (22) 14.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/069974 14.07.2008<br />

(87) WO 2009/009793 2009/03 <strong>15</strong>.01.2009<br />

(88) 26.03.2009<br />

(30) 12.07.2007 US 949365 P<br />

(54) • INHIBITOREN VON AKT/PKB MIT ANTI-<br />

TUMORALER WIRKUNG<br />

• INHIBITORS OF AKT/PKB WITH ANTI-<br />

TUMOR ACTIVITY<br />

• INHIBITEURS DE AKT/PKB À ACTIVITÉ<br />

ANTITUMORALE<br />

(71) University of South Florida, 3802 Spectrum<br />

Blvd., Suite 100, Tampa, FL 33612-9220, US<br />

(72) CHENG, Jin, Q., Tampa, FL 33647, US<br />

SUN, Mei, Tampa, FL 33647, US<br />

SEBTI, Said, M., Tampa, FL 33647, US<br />

(74) Büchel, Edwin, Isenbruck Bösl Hörschler<br />

Wichmann LLP Eastsite One Seckenheimer<br />

Landstrasse 4, 68163 Mannheim, DE<br />

A61K 31/517 → (51) A61K 31/352<br />

A61K 31/517 → (51) C07D 239/70<br />

A61K 31/517 → (51) C07D 239/90<br />

A61K 31/519 → (51) A61K 31/131<br />

A61K 31/519 → (51) A61K 31/4468<br />

A61K 31/519 → (51) C07D 487/04<br />

A61K 31/52 → (51) C07D 403/06<br />

(51) A61K 31/53 (11) 2 173 353 A1*<br />

A01N 1/02<br />

A61P 41/00<br />

A61K 31/167<br />

(25) En (26) En<br />

(21) 08714339.2 (22) 03.03.2008<br />

44<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>15</strong>/<strong>2010</strong>) 14.04.<strong>2010</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) AU 2008/000289 03.03.2008<br />

(87) WO 2008/106724 2008/37 12.09.2008<br />

(30) 02.03.2007 AU 2007901098 P<br />

(54) • TRANSPLANTATE<br />

• TRANSPLANTS<br />

• TRANSPLANTS<br />

(71) Hibernation Therapeutics Limited, 14 Dahl<br />

Cresent, Wulguru, QLD 4811, AU<br />

(72) DOBSON, Geoffrey, Wulguru, Queensland<br />

4811, AU<br />

(74) Hallybone, Huw George, et al, Carpmaels &<br />

Ransford 43-45 Bloomsbury Square, London<br />

WC1A 2RA, GB<br />

A61K 31/53 → (51) A01N 43/64<br />

A61K 31/53 → (51) A61K 31/517<br />

(51) A61K 31/535 (11) 2 173 354 A1*<br />

(25) En (26) En<br />

(21) 08797323.6 (22) 07.08.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/072401 07.08.2008<br />

(87) WO 2009/021083 2009/07 12.02.2009<br />

(30) 09.08.2007 US 954845 P<br />

(54) • CHINOXALINDERIVATE ALS PI3-KINASE-<br />

INHIBITOREN<br />

• QUINOXALINE DERIVATIVES AS PI3<br />

KINASE INHIBITORS<br />

• DÉRIVÉS DES QUINOXALINES UTILISÉS<br />

COMME INHIBITEURS DES PI3-KINASES<br />

(71) GlaxoSmithKline LLC, One Franklin Plaza 200<br />

North 16th Street, Philadelphia, PA 19102,<br />

US<br />

(72) KNIGHT, Steven, David, Collegeville, PA<br />

19426, US<br />

PARISH, Cynthia, A., Collegeville, PA 19426,<br />

US<br />

RIDGERS, Lance, H., Collegeville, PA 19426,<br />

US<br />

SARPONG, Martha, A., Collegeville, PA<br />

19426, US<br />

CHAUDHARI, Amita, M., Collegeville, PA<br />

19426, US<br />

(74) Gladwin, Amanda Rachel, GlaxoSmithKline<br />

Corporate Intellectual Property CN925.1<br />

Great West Road, Brentford, Middlesex TW8<br />

9GS, GB<br />

A61K 31/5377 → (51) C07D 263/48<br />

A61K 31/54 → (51) A61K 31/7<strong>15</strong><br />

A61K 31/54<strong>15</strong> → (51) A61K 31/45<strong>15</strong><br />

(51) A61K 31/551 (11) 2 173 355 A2*<br />

A61K 31/553 A61K 31/554<br />

A61P 25/28<br />

(25) En (26) En<br />

(21) 08774661.6 (22) 02.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/058527 02.07.2008<br />

(87) WO 2009/004038 2009/02 08.01.2009<br />

(88) 26.11.2009<br />

(30) 02.07.2007 EP 07111491<br />

(54) • PIRENZEPIN UND SEINE DERIVATE ALS<br />

ANTI-AMYLOID-MITTEL

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