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Bulletin 2010/15 - European Patent Office

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(C07D) II.1(1)<br />

(74) Cornish, Kristina Victoria Joy, et al, Kilburn &<br />

Strode LLP 20 Red Lion Street, London<br />

WC1R 4PJ, GB<br />

C07D 401/04 → (51) A61K 31/4439<br />

C07D 401/04 → (51) C07D 209/12<br />

C07D 401/06 → (51) C07D 209/12<br />

C07D 401/12 → (51) C07D 209/18<br />

C07D 401/12 → (51) C07D 231/54<br />

(51) C07D 401/14 (11) 1 796 678 B1<br />

C07D 471/10 A61K 31/553<br />

A61K 31/55 A61K 31/438<br />

A61K 31/4166 A61P 25/06<br />

(25) En (26) En<br />

(21) 05795301.0 (22) 09.09.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 20.06.2007<br />

(86) US 2005/032036 09.09.2005<br />

(87) WO 2006/031606 2006/12 23.03.2006<br />

(30) 13.09.2004 US 609436 P<br />

(54) • CARBOXAMID-SPIROLACTAM-CGRP-<br />

REZEPTOR-ANTAGONISTEN<br />

• CARBOXAMIDE SPIROLACTAM CGRP<br />

RECEPTOR ANTAGONISTS<br />

• CARBOXAMIDE SPIROLACTAM CGRP<br />

RECEPTOR ANTAGONISTS<br />

(73) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) WILLIAMS, Theresa, M., Rahway, New<br />

Jersey 07065-0907, US<br />

BURGEY, Christopher, S., Rahway, New<br />

Jersey 07065-0907, US<br />

TUCKER, Thomas, J., Rahway, New Jersey<br />

07065-0907, US<br />

STUMP, Craig, A., Rahway, New Jersey<br />

07065-0907, US<br />

BELL, Ian, M., Rahway, New Jersey 07065-<br />

0907, US<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

C07D 401/14 → (51) C07D 231/12<br />

(51) C07D 403/02 (11) 1 797 073 B1<br />

C07D 221/02 C07D 401/00<br />

C07D 239/00 C07D 241/00<br />

A61K 31/4965 A61K 31/44<br />

A61K 31/517<br />

(25) En (26) En<br />

(21) 05795448.9 (22) 09.09.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 20.06.2007<br />

(86) US 2005/032041 09.09.2005<br />

(87) WO 2006/031610 2006/12 23.03.2006<br />

(30) 13.09.2004 US 609292 P<br />

(54) • BICYCLISCHE ANILIDSPIROLACTAME ALS<br />

ANTAGONISTEN DES CGRP-REZEPTORS<br />

• BICYCLIC ANILIDE SPIROLACTAM CGRP<br />

RECEPTOR ANTAGONISTS<br />

• ANTAGONISTES DES RECEPTEURS DU<br />

CGRP DE SPIROLACTAME ANILIDE BICY-<br />

CLIQUE<br />

(73) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) BELL, Ian, M., Rahway, New Jersey 07065-<br />

0907, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

THEBERGE, Cory, R., Rahway, New Jersey<br />

07065-0907, US<br />

STUMP, Craig, A., Rahway, New Jersey<br />

07065-0907, US<br />

ZHANG, Xufang, Rahway, New Jersey<br />

07065-0907, US<br />

GALLICCHIO, Steven, N., Rahway, New<br />

Jersey 07065-0907, US<br />

ZARTMAN, C., Blair, Rahway, New Jersey<br />

07065-0907, US<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

C07D 403/12 → (51) C07D 209/12<br />

C07D 403/12 → (51) C07D 209/18<br />

C07D 403/12 → (51) C07D 231/54<br />

C07D 403/14 → (51) C07D 231/12<br />

C07D 405/06 → (51) C07D 209/12<br />

C07D 405/12 → (51) C07D 209/18<br />

C07D 405/12 → (51) C07D 239/96<br />

C07D 405/12 → (51) C07D 409/12<br />

C07D 409/04 → (51) C07D 231/54<br />

(51) C07D 409/12 (11) 1 858 890 B1<br />

C07D 409/14 C07D 405/12<br />

C07D 207/26 A61K 31/40<strong>15</strong><br />

A61K 31/4025 A61P 7/02<br />

(25) De (26) De<br />

(21) 06724863.3 (22) 22.02.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 28.11.2007<br />

(86) EP 2006/060182 22.02.2006<br />

(87) WO 2006/089909 2006/35 31.08.2006<br />

(30) 25.02.2005 DE 102005008649<br />

(54) • NEUE SUBSTITUIERTE PYRROLIDINONE<br />

MIT ANTITHROMBOTISCHER WIRKUNG,<br />

DEREN HERSTELLUNG UND DEREN VER-<br />

WENDUNG ALS ARZNEIMITTEL<br />

• NOVEL ANTITHROMBOTIC SUBSTITUTED<br />

PYRROLIDINONES, THE PRODUCTION<br />

AND USE THEREOF IN THE FORM OF<br />

MEDICAMENTS<br />

• NOUVELLES PYRROLIDINONES SUBSTI-<br />

TUEES A EFFET ANTITHROMBOTIQUE,<br />

LEUR PRODUCTION ET LEUR UTILISA-<br />

TION COMME MEDICAMENTS<br />

(73) Boehringer Ingelheim Pharma GmbH & Co.<br />

KG, Binger Strasse 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(84) DE<br />

(73) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(84) AT BE BG CH CY CZ DK EE ES FI FR GB GR<br />

HU IE IS IT LI LT LU LV MC NL PL PT RO SE<br />

SI SK TR<br />

(72) GERLACH, Kai, 88441 Mittelbiberach, DE<br />

PRIEPKE, Henning, 88447 Warthausen, DE<br />

PFAU, Roland, 88400 Biberach, DE<br />

DAHMANN, Georg, 88448 Attenweiler, DE<br />

WIENEN, Wolfgang, 88400 Biberach, DE<br />

SCHULER-METZ, Annette, 89081 Ulm, DE<br />

NAR, Herbert, 88416 Ochsenhausen, DE<br />

(74) Hammann, Heinz, et al, Boehringer Ingelheim<br />

GmbH CD-<strong>Patent</strong>s Binger Straße 173, 55216<br />

Ingelheim am Rhein, DE<br />

576<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>15</strong>/<strong>2010</strong>) 14.04.<strong>2010</strong><br />

C07D 409/12 → (51) C07D 209/40<br />

C07D 409/12 → (51) C07D 231/54<br />

C07D 409/14 → (51) C07D 231/12<br />

C07D 409/14 → (51) C07D 409/12<br />

C07D 409/14 → (51) C07F 5/02<br />

(51) C07D 413/04 (11) 1 805 170 B1<br />

C07D 265/18 A61K 31/535<br />

A61P 29/00<br />

(25) En (26) En<br />

(21) 05798257.1 (22) 19.10.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 11.07.2007<br />

(86) EP 2005/011233 19.10.2005<br />

(87) WO 2006/045505 2006/18 04.05.2006<br />

(30) 21.10.2004 GB 0423405<br />

(54) • MIF-HEMMER<br />

• MIF-INHIBITORS<br />

• INHIBITEURS MIF<br />

(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(84) BE BG CH CY CZ DE DK EE ES FI FR GB GR<br />

HU IE IS IT LI LT LU LV MC NL PL PT RO SE<br />

SI SK TR<br />

(73) Novartis Pharma GmbH, Brunner Strasse 59,<br />

1230 Wien, AT<br />

(84) AT<br />

(72) BILLICH, Andreas, A-2340 Mödling, AT<br />

LEHR, Philipp, A-2340 Mödling, AT<br />

GSTACH, Hubert, A-1070 Wien, AT<br />

(74) Schaller, Hans, Novartis AG Corporate Intellectual<br />

Property, 4002 Basel, CH<br />

C07D 413/04 → (51) C07D 209/12<br />

C07D 413/04 → (51) C07D 401/04<br />

C07D 413/12 → (51) C07D 209/18<br />

C07D 413/14 → (51) C07D 209/18<br />

C07D 413/14 → (51) C07D 231/12<br />

C07D 417/12 → (51) C07D 209/18<br />

C07D 417/14 → (51) C07D 231/12<br />

(51) C07D 453/02 (11) 1 704 146 B1<br />

A61K 31/4468 A61P 1/00<br />

(25) En (26) En<br />

(21) 05705267.2 (22) 07.01.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

AL BA HR LV MK YU<br />

(43) 27.09.2006<br />

(86) US 2005/000510 07.01.2005<br />

(87) WO 2005/068461 2005/30 28.07.2005<br />

(30) 07.01.2004 US 534892 P<br />

09.04.2004 US 560938 P<br />

(54) • STEREOISOMERE VERBINDUNGEN UND<br />

VERFAHREN ZUR BEHANDLUNG VON<br />

ERKRANKUNGEN DES MAGEN-DARM-<br />

TRAKTS UND DES ZENTRALEN NERVEN-<br />

SYSTEMS<br />

• STEREOISOMERIC COMPOUNDS AND<br />

METHODS FOR THE TREATMENT OF<br />

GASTROINTESTINAL AND CENTRAL NER-<br />

VOUS SYSTEM DISORDERS<br />

• COMPOSES STEREO-ISOMERES ET<br />

METHODES DE TRAITEMENT DE TROU-<br />

BLES GASTRO-INTESTINAUX ET DU SYS-<br />

TEME NERVEUX CENTRAL

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