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Bulletin 2011/31 - European Patent Office

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(C07D) I.1(1)<br />

• ISOXAZOLE/ISOXAZOLINE/COMBRETAS-<br />

TATIN LINKED DIHYDROQUINAZOLINONE<br />

HYBRIDS AS POTENTIAL ANTICANCER<br />

AGENTS AND PROCESS FOR THE PREP-<br />

ARATION THEREOF<br />

• HYBRIDES DIHYDROQUINAZOLINONE-<br />

ISOXAZOLE/ISOXAZOLINE/COMBRÉSTA-<br />

TATINE COMME AGENTS ANTICANCÉ-<br />

REUX POTENTIELS, ET PROCÉDÉ DE<br />

PRÉPARATION ASSOCIÉ<br />

(71) Council Of Scientific & Industrial Research,<br />

Anusandhan of Societies Act (Act XXI of<br />

1860) Anusandhan Bhawan 2 Rafi Marg.,<br />

New Delhi 110 001, IN<br />

(72) KAMAL, Ahmed, Andhra Pradesh, IN<br />

BHARATHI, Earla, Vijaya, Andhra Pradesh, IN<br />

REDDY, Jonnala, Surendranadha, Andhra<br />

Pradesh, IN<br />

DASTAGIRI, Dudekula, Andhra Pradesh, IN<br />

VISWANATH, Arutla, Andhra Pradesh, IN<br />

(74) Jönsson, Anneli, Awapatent AB Södra<br />

Hamngatan 37-41 Box 11394, 404 28<br />

Göteborg, SE<br />

C07D 241/08 → (51) A23K 1/16<br />

C07D 241/42 → (51) C07D 239/48<br />

C07D 241/44 → (51) C07D 239/48<br />

C07D 243/08 → (51) A01N 43/50<br />

C07D 249/06 → (51) C07D 2<strong>31</strong>/12<br />

(51) C07D 257/02 (11) 2 350 0<strong>31</strong> A2*<br />

C07D 273/00 A61K <strong>31</strong>/395<br />

A61P 19/02 A61P 25/28<br />

A61P 35/00<br />

(25) En (26) En<br />

(21) 09791736.3 (22) 20.08.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/054487 20.08.2009<br />

(87) WO 2010/022249 2010/08 25.02.2010<br />

(88) 15.04.2010<br />

(30) 22.09.2008 US 98865 P<br />

10.02.2009 US 151245 P<br />

20.08.2008 US 90410 P<br />

(54) • MAKROCYCLISCHE VERBINDUNGEN ZUR<br />

INHIBIERUNG DES TUMORNEKROSEFAK-<br />

TORS ALPHA<br />

• MACROCYCLIC COMPOUNDS FOR INHI-<br />

BITION OF TUMOR NECROSIS FACTOR<br />

ALPHA<br />

• COMPOSÉS DESTINÉS À L INHIBITION DU<br />

FACTEUR DE NÉCROSE TUMORALE<br />

ALPHA<br />

(71) Ensemble Therapeutics Corporation, 99 Erie<br />

Street, Cambridge MA 02139, US<br />

(72) LEE, Jinbo, Andover MA 01810, US<br />

BOND, Julian, F., Weymouth MA 02188, US<br />

TERRETT, Nicholas, Sherborn MA 01770, US<br />

FAVALORO, Frank, G., North Attleboro MA<br />

02760, US<br />

WANG, Daniel, Duxbury MA 02332, US<br />

BRIGGS, Timothy, F., Cambridge MA 02141,<br />

US<br />

SEIGAL, Benjamin, Adam, Watertown MA<br />

02472, US<br />

SUN, Wei-Chuan, Acton MA 01720, US<br />

HALE, Stephen, P., Belmont MA 02478, US<br />

(74) Harris, Jennifer Lucy, et al, Kilburn & Strode<br />

LLP 20 Red Lion Street, London WC1R 4PJ,<br />

GB<br />

C07D 261/08 → (51) C07D 2<strong>31</strong>/12<br />

C07D 263/32 → (51) C07D 213/40<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

C07D 263/32 → (51) C07D 2<strong>31</strong>/12<br />

(51) C07D 263/56 (11) 2 350 032 A1*<br />

C07D 413/12 A61K <strong>31</strong>/423<br />

(25) En (26) En<br />

(21) 09793015.0 (22) 25.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/058398 25.09.2009<br />

(87) WO 2010/036905 2010/13 01.04.2010<br />

(30) 26.09.2008 US 100678 P<br />

(54) • BENZOXAZOLVERBINDUNGEN UND<br />

ANWENDUNGSVERFAHREN<br />

• BENZOXAZOLE COMPOUNDS AND METH-<br />

ODS OF USE<br />

• COMPOSÉS BENZOXAZOLE ET PROCÉDÉS<br />

D'UTILISATION<br />

(71) Eisai R&D Management Co., Ltd., 6-10,<br />

Koishikawa 4-chome Bunkyo-ku, Tokyo 112-<br />

8088, JP<br />

(72) ZHENG, Wanjun, Londonderry, New Hampshire<br />

03053-3<strong>31</strong>7, US<br />

SPYVEE, Mark, Hampstead, New Hampshire<br />

03841, US<br />

GUSOVSKY, Fabian, Andover, Massachusetts<br />

01810-5502, US<br />

ISHIZAKA, Sally T., Weston, Massachusetts<br />

02493-1645, US<br />

(74) Harrison Goddard Foote, Belgrave Hall Belgrave<br />

Street, Leeds LS2 8DD, GB<br />

C07D 271/113→ (51) C07D 417/04<br />

C07D 273/00 → (51) C07D 257/02<br />

C07D 277/22 → (51) C07C 213/08<br />

C07D 277/24 → (51) C07D 2<strong>31</strong>/12<br />

C07D 277/28 → (51) C07D 213/40<br />

C07D 277/34 → (51) C07D 213/40<br />

C07D 277/46 → (51) A61P 3/10<br />

C07D 281/10 → (51) A61K <strong>31</strong>/553<br />

C07D 285/06 → (51) C07D 2<strong>31</strong>/12<br />

C07D 285/135→ (51) C07D 417/04<br />

C07D 295/04 → (51) A61K <strong>31</strong>/4025<br />

C07D 295/088→ (51) C07C 39/42<br />

C07D 295/088→ (51) C07C 217/08<br />

C07D 295/10 → (51) A61K <strong>31</strong>/4025<br />

C07D 295/135→ (51) C07C 235/38<br />

C07D 295/135→ (51) C07C <strong>31</strong>1/21<br />

C07D 295/185→ (51) C07D 209/24<br />

(51) C07D 301/10 (11) 2 350 033 A1*<br />

(25) De (26) De<br />

(21) 09783673.8 (22) 02.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2009/062804 02.10.2009<br />

(87) WO 2010/040688 2010/15 15.04.2010<br />

(30) 08.10.2008 EP 08166057<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINES<br />

ALKYLENOXIDS<br />

• METHOD FOR PRODUCING AN ALKYLENE<br />

OXIDE<br />

179<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

• PROCÉDÉ DE FABRICATION D UN OXYDE<br />

D ALKYLÈNE<br />

(71) BASF SE, 67056 Ludwigshafen, DE<br />

(72) GITTER, Markus, Baton Rouge Louisiana<br />

70808, US<br />

(74) Altmann, Andreas, Herzog Fiesser & Partner<br />

<strong>Patent</strong>anwälte Isartorplatz 1, 803<strong>31</strong><br />

München, DE<br />

(51) C07D 307/12 (11) 2 350 034 A1*<br />

C07D 309/06 C07D <strong>31</strong>3/04<br />

C07D <strong>31</strong>7/26 C07D <strong>31</strong>9/06<br />

C07D 335/02 C07D 493/04<br />

C07D 493/10 A01N 43/08<br />

A01N 43/16 A01N 43/28<br />

A01N 43/32<br />

(25) En (26) En<br />

(21) 09783332.1 (22) 23.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

RS<br />

(86) EP 2009/062327 23.09.2009<br />

(87) WO 2010/046194 2010/17 29.04.2010<br />

(30) 20.10.2008 GB 0819205<br />

(54) • NEUE HERBIZIDE<br />

• NOVEL HERBICIDES<br />

• NOUVEAUX HERBICIDES<br />

(71) Syngenta Limited, <strong>European</strong> Regional Centre<br />

Priestley Road Surrey Research Park, Guildford,<br />

Surrey GU2 7YH, GB<br />

(72) MATHEWS, Christopher John, Bracknell<br />

Berkshire RG42 6EY, GB<br />

CLOUGH, John Martin, Bracknell Berkshire<br />

RG42 6EY, GB<br />

BEAUTEMENT, Kevin, Bracknell Berkshire<br />

RG42 6EY, GB<br />

TYTE, Melloney, Bracknell Berkshire RG42<br />

6EY, GB<br />

ROBINSON, Louisa, Bracknell Berkshire<br />

RG42 6EY, GB<br />

JEANMART, Stephane André Marie, Bracknell<br />

Berkshire RG42 6EY, GB<br />

(74) Breen, Anthony Paul, et al, Syngenta Limited<br />

Intellectual Property Department PO Box<br />

3538 Jealott's Hill International Research<br />

Centre, Bracknell Berkshire RG42 6YA, GB<br />

C07D 307/12 → (51) C07C 39/42<br />

(51) C07D 307/20 (11) 2 350 035 A2*<br />

C07D 307/34 C07D 307/24<br />

C07D 307/28<br />

(25) En (26) En<br />

(21) 09829644.5 (22) 30.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/062778 30.10.2009<br />

(87) WO 2010/062689 2010/22 03.06.2010<br />

(88) 22.07.2010<br />

(30) 30.10.2008 US 109634 P<br />

(54) • REDUZIERUNG VON HMF-ETHERN MIT-<br />

HILFE EINES METALLKATALYSATORS<br />

• REDUCTION OF HMF ETHERS WITH<br />

METAL CATALYST<br />

• RÉDUCTION D ÉTHERS D HYDROXYMÉ-<br />

THYLFURFURAL AVEC UN CATALYSEUR<br />

MÉTALLIQUE<br />

(71) Archer Daniels Midland Co., 4666 Faries<br />

Parkway, Decatur, IL 62526, US<br />

(72) BLOOM, Paul, David, Decature, IL 62521, US<br />

SANBORN, Alexandra, J., Lincoln, IL 62656,<br />

US<br />

(74) Hart, Deborah Mary, et al, Kilburn & Strode<br />

LLP 20 Red Lion Street, London WC1R 4PJ,<br />

GB

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