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Bulletin 2011/31 - European Patent Office

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(A61K) I.1(2)<br />

(30) 17.10.2008 KR 20080101932<br />

(54) • PHARMAZEUTISCHE ZUSAMMENSET-<br />

ZUNG ZUR PRÄVENTION UND BEHAND-<br />

LUNG VON DIABETES ODER ADIPOSITAS<br />

MIT EINER VERBINDUNG ZUR HEMMUNG<br />

DER DIPEPTIDYLPEPTIDASE-IV-AKTIVI-<br />

TÄT UND ANDEREN ANTIDIABETIKA ODER<br />

ANTIADIPOSITA ALS WIRKSTOFFE<br />

• PHARMACEUTICAL COMPOSITION FOR<br />

PREVENTION AND TREATMENT OF DIA-<br />

BETES OR OBESITY COMPRISING A<br />

COMPOUND THAT INHIBITS ACTIVITY OF<br />

DIPEPTIDYL PEPTIDASE-IV, AND OTHER<br />

ANTIDIABETIC OR ANTIOBESITY AGENTS<br />

AS ACTIVE INGREDIENTS<br />

• COMPOSITION PHARMACEUTIQUE ET<br />

MEDICAMENT POUR LA PREVENTION ET<br />

LE TRAITEMENT DE DIABETES OU DE<br />

L'OBESITE COMPRENANT COMME PRIN-<br />

CIPE ACTIF, UN COMPOSE QUI INHIBE<br />

L'ACTIVATION DE DIPEPTIDYL PEPTI-<br />

DASE-IV<br />

(71) Dong-A Pharmaceutical Co., Ltd., 252<br />

Yongdu-dong Dongdaemun-ku, Seoul 130-<br />

072, KR<br />

(72) SHIN, Chang Yell, Seoul 132-691, KR<br />

CHOI, Song-Hyen, Suwon-si Gyeonggi-do<br />

443-372, KR<br />

CHAE, Yu Na, Yongin-si Gyeonggi-do 448-<br />

130, KR<br />

YANG, Eun Kyoung, Yongin-si Gyeonggi-do<br />

446-905, KR<br />

AHN, Gook Jun, Anseong-si Gyeonggi-do<br />

456-933, KR<br />

SON, Moon-Ho, Suwon-si Gyeonggi-do 442-<br />

070, KR<br />

KIM, Heung Jae, Seongnam-si Gyeonggi-do<br />

463-773, KR<br />

KWAK, Woo Young, Yongin-si Gyeonggi-do<br />

449-827, KR<br />

MIN, Jong Pil, Yongin-si Gyeonggi-do 446-<br />

760, KR<br />

YOON, Tae Hyun, Yongin-si Gyeonggi-do<br />

446-905, KR<br />

KIM, Soon Hoe, Suwon-si Gyeonggi-do 443-<br />

470, KR<br />

YOO, Moohi, Seoul 135-807, KR<br />

(74) Andrews, Timothy Stephen, et al, Marks &<br />

Clerk LLP 66-68 Hills Road, Cambridge CB2<br />

1LA, GB<br />

A61K <strong>31</strong>/498 → (51) A61K <strong>31</strong>/137<br />

A61K <strong>31</strong>/4985 → (51) A61K <strong>31</strong>/40<br />

A61K <strong>31</strong>/4985 → (51) A61K <strong>31</strong>/522<br />

A61K <strong>31</strong>/506 → (51) A61K <strong>31</strong>/551<br />

A61K <strong>31</strong>/506 → (51) C07D 235/16<br />

A61K <strong>31</strong>/517 → (51) C07D 401/14<br />

A61K <strong>31</strong>/519 → (51) A61K <strong>31</strong>/551<br />

A61K <strong>31</strong>/519 → (51) C07D 487/04<br />

A61K <strong>31</strong>/52 → (51) A61K <strong>31</strong>/551<br />

A61K <strong>31</strong>/52 → (51) C07D 401/14<br />

(51) A61K <strong>31</strong>/522 (11) 2 351 568 A2<br />

A61K <strong>31</strong>/4985 A61P 3/10<br />

A61P 9/04<br />

(25) De (26) De<br />

(21) 11156183.3 (22) 03.05.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

AL BA HR MK RS<br />

(27) 03.05.2007 EP 07728723<br />

(30) 04.05.2006 EP 06009203<br />

(54) • Verwendungen von dpp iv Inhibitoren<br />

• Uses of dpp-iv inhibitors<br />

• Utilisations d'inhibiteurs de l'enzyme dpp<br />

iv<br />

(71) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim am<br />

Rhein, DE<br />

Boehringer Ingelheim Pharma GmbH & Co.<br />

KG, Binger Straße 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(72) Dugi, Klaus, 01324, DRESDEN, DE<br />

Himmelsbach, Frank, 88441, MITTELBIBER-<br />

ACH, DE<br />

Mark, Michael, 88400, BIBERACH, DE<br />

(74) Hammann, Heinz, Boehringer Ingelheim<br />

GmbH CD-<strong>Patent</strong>s Binger Straße 173, 55216<br />

Ingelheim am Rhein, DE<br />

(62) 07728723.3 / 2 015 754<br />

A61K <strong>31</strong>/5377 → (51) C07D 235/16<br />

A61K <strong>31</strong>/538 → (51) A61K <strong>31</strong>/137<br />

(51) A61K <strong>31</strong>/551 (11) 2 351 569 A1<br />

A61K <strong>31</strong>/192 A61K <strong>31</strong>/343<br />

A61K <strong>31</strong>/4409 A61K <strong>31</strong>/506<br />

A61K <strong>31</strong>/519 A61K <strong>31</strong>/5578<br />

A61P 9/08 A61P 9/10<br />

A61P 9/12 A61K <strong>31</strong>/52<br />

(25) En (26) En<br />

(21) 11000632.7 (22) 25.10.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(30) 26.10.2005 US 730273 P<br />

(54) • Kombinationstherapie mit Fasudil zur<br />

Behandlung von pulmonaler Hypertonie<br />

• Fasudil in combination therapies for the<br />

treatment of pulmonary arterial hypertension<br />

• Fasudil dans des thérapies combinées pour<br />

le traitement de l'hypertension artérielle<br />

pulmonaire<br />

(71) Asahi Kasei Pharma Corporation, 1-105<br />

Kanda Jinbocho Chiyoda-ku, Tokyo 101-<br />

8101, JP<br />

(72) Fong, Benson, Brisbane CA 94005-1846, US<br />

(74) Forstmeyer, Dietmar, et al, BOETERS &<br />

LIECK Oberanger 32, 803<strong>31</strong> München, DE<br />

(62) 09007232.3 / 2 111 863<br />

06826765.7 / 1 951 253<br />

A61K <strong>31</strong>/5578 → (51) A61K <strong>31</strong>/551<br />

A61K <strong>31</strong>/573 → (51) A61K <strong>31</strong>/65<br />

A61K <strong>31</strong>/60 → (51) A61K <strong>31</strong>/05<br />

A61K <strong>31</strong>/64 → (51) A61K <strong>31</strong>/40<br />

(51) A61K <strong>31</strong>/65 (11) 2 351 570 A1<br />

A61K <strong>31</strong>/70 A61K <strong>31</strong>/165<br />

A61K <strong>31</strong>/44 A61K <strong>31</strong>/573<br />

A61P 29/00 A61P <strong>31</strong>/00<br />

(25) En (26) En<br />

(21) 10185616.9 (22) 27.11.2001<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(27) 27.11.2001 PCT/US01/44<strong>31</strong>5<br />

(30) 27.11.2000 US 723064<br />

(54) • Antibiotikum-/Analgesikumformulierung<br />

und Verfahren zur Herstellung dieser<br />

Formulierung<br />

• An Antibiotic/Analgesic Formulation And a<br />

Method of Making This Formulation<br />

383<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

• Formulation antibiotique/analgésique et<br />

son procédé de fabrication<br />

(71) IVX Animal Health, Inc., 3915 South 48th<br />

Street Terrace, St. Joseph MO 64503, US<br />

(72) Mihalik, Richard, St Joseph, MO 64501, US<br />

(74) Turner, Craig Robert, A.A. Thornton & Co.<br />

235 High Holborn, London WC1V 7LE, GB<br />

(62) 01997308.0 / 1 345 611<br />

A61K <strong>31</strong>/661 → (51) A61K <strong>31</strong>/137<br />

A61K <strong>31</strong>/661 → (51) C07C 217/84<br />

(51) A61K <strong>31</strong>/695 (11) 2 351 571 A1<br />

A61P 35/00 A61P 43/00<br />

C07F 7/18<br />

(25) Ja (26) En<br />

(21) 09818941.8 (22) 02.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2009/005128 02.10.2009<br />

(87) WO 2010/041401 2010/15 15.04.2010<br />

(30) 09.10.2008 JP 2008262646<br />

(54) • PROTEINPHOSPHATASEHEMMER<br />

• PROTEIN PHOSPHATASE INHIBITOR<br />

• INHIBITEUR DE PROTÉINE PHOSPHATASE<br />

(71) LSIP, LLC, 7-12, Marunouchi 1-chome,<br />

Chiyoda-ku Tokyo 100-0005, JP<br />

(72) SAKAGUCHI, Kazuyasu, , JP<br />

TANINO, Keiji, , JP<br />

CHUMAN, Yoshiro, , JP<br />

YOSHIMURA, Fumihiko, , JP<br />

YAGI, Hiroaki, , JP<br />

(74) von Kreisler Selting Werner, <strong>Patent</strong>anwälte<br />

Deichmannhaus am Dom Bahnhofsvorplatz<br />

1, 50667 Köln, DE<br />

A61K <strong>31</strong>/70 → (51) A61K <strong>31</strong>/65<br />

A61K <strong>31</strong>/7016 → (51) C12P 19/44<br />

A61K <strong>31</strong>/7024 → (51) C07H 13/06<br />

A61K <strong>31</strong>/7088 → (51) A61K 45/00<br />

A61K <strong>31</strong>/7105 → (51) A61K 45/00<br />

A61K <strong>31</strong>/7115 → (51) A61K 45/00<br />

A61K <strong>31</strong>/713 → (51) C12N 15/00<br />

A61K 35/74 → (51) A23L 1/29<br />

A61K 35/74 → (51) A23L 3/3571<br />

A61K 36/00 → (51) A61K 36/53<br />

A61K 36/18 → (51) A61K <strong>31</strong>/05<br />

(51) A61K 36/53 (11) 2 351 572 A1<br />

A23L 1/30 A61K 36/00<br />

A61P 1/04 A61P <strong>31</strong>/04<br />

A61P 35/00<br />

(25) Ja (26) En<br />

(21) 09823693.8 (22) 30.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2009/068668 30.10.2009<br />

(87) WO 2010/050583 2010/18 06.05.2010<br />

(30) 30.10.2008 JP 2008279358<br />

(54) • MITTEL GEGEN HELICOBACTER PYLORI<br />

• AGENT HAVING ANTI-HELICOBACTER<br />

PYLORI ACTIVITY<br />

• AGENT AYANT UNE ACTIVITÉ ANTI-HELI-<br />

COBACTER PYLORI

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