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Bulletin 2011/31 - European Patent Office

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(C07D) I.1(1)<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) SE 2009/051187 19.10.2009<br />

(87) WO 2010/044743 2010/16 22.04.2010<br />

(30) 17.10.2008 SE 0850043<br />

23.10.2008 SE 0850050<br />

(54) • NEUE THIOPHENVERBINDUNGEN FÜR<br />

THERAPEUTISCHE ZWECKE<br />

• NOVEL THIOPHENE COMPOUNDS FOR<br />

USE IN THERAPHY<br />

• NOUVEAUX COMPOSÉS DU THIOPHÈNE<br />

THÉRAPEUTIQUES<br />

(71) BioChromix Pharma AB, Retzius väg 8, 171<br />

65 Solna, SE<br />

(72) ÅSBERG, Peter, S-11330 Stockholm, SE<br />

JOHANSSON, Leif, S-58223 Linköping, SE<br />

HERLAND, Anna, S-58247 Linköping, SE<br />

(74) Rystedt, Per Hampus, BRANN AB P.O. Box<br />

12246, 102 26 Stockholm, SE<br />

C07D 333/56 → (51) C07D 209/18<br />

C07D 333/66 → (51) A61K <strong>31</strong>/4439<br />

C07D 335/02 → (51) C07D 307/12<br />

(51) C07D 345/00 (11) 2 350 043 A1*<br />

C07D 517/00 A61K 9/127<br />

(25) En (26) En<br />

(21) 09819991.2 (22) 09.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/060251 09.10.2009<br />

(87) WO 2010/042877 2010/15 15.04.2010<br />

(30) 09.10.2008 US 104212 P<br />

09.10.2008 US 104219 P<br />

26.06.2009 US 220666 P<br />

(54) • VERBESSERTE AMINOLIPIDE UND VER-<br />

FAHREN ZUR FREISETZUNG VON NUKLE-<br />

INSÄUREN<br />

• IMPROVED AMINO LIPIDS AND METHODS<br />

FOR THE DELIVERY OF NUCLEIC ACIDS<br />

• LIPIDES AMINÉS AMÉLIORÉS ET PROCÉ-<br />

DÉS D'ADMINISTRATION D'ACIDES<br />

NUCLÉIQUES<br />

(71) TEKMIRA Pharmaceuticals Corporation, 100-<br />

8900 Glenlyon Parkway, Burnaby, BC V5J<br />

5J8, CA<br />

The University of British Columbia, 103 -<br />

6190 Agronomy Road, Vancouver, BC V6T<br />

1Z3, CA<br />

(72) HOPE, Michael, J., Vancouver British<br />

Columbia V6R 2K2, CA<br />

SEMPLE, Sean, C., Delta British Columbia<br />

V4E 3L5, CA<br />

CHEN, Jianxin, Vancouver British Columbia<br />

V6S 1B7, CA<br />

MADDEN, Thomas, D., Vancouver British<br />

Columbia V6L 2A1, CA<br />

CULLIS, Pieter, R., Vancouver British<br />

Columbia V6R 1H4, CA<br />

CIUFOLINI, Marco, A., Vancouver British<br />

Columbia V6T 1Z1, CA<br />

MUI, Barbara, British Columbia V5T 2G3, CA<br />

(74) Walker, Ross Thomson, et al, Forrester &<br />

Boehmert Pettenkoferstrasse 20-22, 80336<br />

München, DE<br />

(51) C07D 401/00 (11) 2 350 044 A1*<br />

(25) En (26) En<br />

(21) 09819926.8 (22) 09.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/060108 09.10.2009<br />

(87) WO 2010/042785 2010/15 15.04.2010<br />

(30) 10.10.2008 US 104551 P<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(54) • VERFAHREN ZUR EINLEITUNG VON<br />

NEGATIVER CHEMOTAXIS<br />

• METHOD OF INDUCING NEGATIVE CHE-<br />

MOTAXIS<br />

• PROCÉDÉ D INDUCTION D UN CHIMIO-<br />

TACTISME NÉGATIF<br />

(71) Celtaxsys, INC., ATDC Biosciences Center,<br />

0390 <strong>31</strong>1 Ferst Drive, Atlanta, GA 30332, US<br />

(72) GOODHEW, Erica, Brook, Atlanta GA 30<strong>31</strong>8,<br />

US<br />

(74) Chapman, Paul William, Kilburn & Strode<br />

LLP 20 Red Lion Street, London WC1R 4PJ,<br />

GB<br />

(51) C07D 401/04 (11) 2 350 045 A1*<br />

C07D 401/14 C07D 405/14<br />

C07D 409/14 C07D 451/06<br />

(25) En (26) En<br />

(21) 09744003.6 (22) 20.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/061253 20.10.2009<br />

(87) WO 2010/0481<strong>31</strong> 2010/17 29.04.2010<br />

(30) 21.10.2008 US 107013 P<br />

(54) • INHIBITOREN VON C-MET-PROTEINKI-<br />

NASE<br />

• C-MET PROTEIN KINASE INHIBITORS<br />

• INHIBITEURS DE LA PROTÉINE KINASE C-<br />

MET<br />

(71) Vertex Pharmaceuticals Incorporated, 130<br />

Waverly Street, Cambridge, MA 02139, US<br />

(72) LAUFFER, David, Stow MA 01775, US<br />

LI, Pan, Lexington MA 02421, US<br />

MCGINTY, Kira, Medford MA 02155, US<br />

RONKIN, Steven, Watertown MA 02472, US<br />

TANG, Qing, Acton MA 01720, US<br />

GRILLOT, Anne-Laure, Somerville MA<br />

02144, US<br />

WAAL, Nathan, Cambridge MA 02141, US<br />

(74) Coles, Andrea Birgit, et al, Kilburn & Strode<br />

LLP 20 Red Lion Street, London WC1R 4PJ,<br />

GB<br />

(51) C07D 401/04 (11) 2 350 046 A1*<br />

(25) En (26) En<br />

(21) 09764118.7 (22) 11.11.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

RS<br />

(86) US 2009/063991 11.11.2009<br />

(87) WO 2010/056720 2010/20 20.05.2010<br />

(30) 14.11.2008 US 114629 P<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINER<br />

NICHTHYDRATISIERBAREN KRISTALL-<br />

FORM<br />

• METHOD FOR PREPARING A NON-<br />

HYDRATABLE CRYSTAL FORM<br />

• PROCÉDÉ DE PRÉPARATION D'UNE<br />

FORME CRISTALLINE NON HYDRATABLE<br />

(71) E. I. du Pont de Nemours and Company,<br />

1007 Market Street, Wilmington, DE 19898,<br />

US<br />

(72) OBERHOLZER, Mathew, Richard, Wilmington<br />

Delaware 19810, US<br />

(74) Beacham, Annabel Rose, et al, Dehns St<br />

Bride's House 10 Salisbury Square, London<br />

EC4Y 8JD, GB<br />

C07D 401/04 → (51) C07D 207/08<br />

C07D 401/04 → (51) C07D 211/96<br />

C07D 401/04 → (51) C07D 213/81<br />

C07D 401/04 → (51) C07D 235/02<br />

181<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

C07D 401/04 → (51) C07D 403/14<br />

C07D 401/06 → (51) C07D 211/76<br />

C07D 401/06 → (51) C07D 217/26<br />

C07D 401/06 → (51) C07D 235/02<br />

C07D 401/10 → (51) C07D 213/40<br />

C07D 401/10 → (51) C07D 213/64<br />

C07D 401/10 → (51) C07D 235/02<br />

(51) C07D 401/12 (11) 2 350 047 A2*<br />

A61K <strong>31</strong>/415 A61P 11/00<br />

A61P 29/00<br />

(25) En (26) En<br />

(21) 09736271.9 (22) 02.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) GB 2009/051303 02.10.2009<br />

(87) WO 2010/038085 2010/14 08.04.2010<br />

(88) 24.06.2010<br />

(30) 02.10.2008 GB 0818033<br />

(54) • P38-MAP-KINASE-INHIBITOREN<br />

• P38 MAP KINASE INHIBITORS<br />

• INHIBITEUR DE LA P38 MAPK KINASE<br />

(71) Respivert Limited, 50-100 Holmers Farm<br />

Way, High Wycombe Buckinghamshire HP12<br />

4EG, GB<br />

(72) ITO, Kazuhiro, London SW7 2AZ, GB<br />

STRONG, Peter, London SW7 2AZ, GB<br />

RAPEPORT, William, Garth, London SW7<br />

2AZ, GB<br />

KING-UNDERWOOD, John, Worcestershire<br />

GL19 3PW, GB<br />

WILLIAMS, Jonathan, Gareth, Nottingham<br />

NG1 1GF, GB<br />

ONIONS, Stuart, Thomas, Nottingham NG1<br />

1GF, GB<br />

MURRAY, Peter, John, London SW7 2AZ,<br />

GB<br />

CHARRON, Catherine, Elisabeth, London<br />

SW7 2AZ, GB<br />

(74) Teuten, Andrew John, et al, Sagittarius IP<br />

Taylor House 39 High Street, Marlow, Bucks<br />

SL7 1AF, GB<br />

(51) C07D 401/12 (11) 2 350 048 A2*<br />

A61K <strong>31</strong>/4427 A61P 7/12<br />

(25) En (26) En<br />

(21) 09744830.2 (22) 14.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/060613 14.10.2009<br />

(87) WO 2010/045306 2010/16 22.04.2010<br />

(88) 15.07.2010<br />

(30) 16.10.2008 US 105968 P<br />

(54) • AZINDERIVATE UND VERFAHREN ZU<br />

DEREN ANWENDUNG<br />

• AZINE DERIVATIVES AND METHODS OF<br />

USE THEREOF<br />

• DÉRIVÉS D'AZINE ET LEURS MÉTHODES<br />

D'UTILISATION<br />

(71) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033-0530, US<br />

(72) PALANI, Anandan, Bridgewater New Jersey<br />

08807, US<br />

XIAO, Dong, Warren New Jersey 07059, US<br />

ASLANIAN, Robert, G., Rockaway New<br />

Jersey 07866, US<br />

BERLIN, Michael, Y., Flemington New Jersey<br />

08822, US

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