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Bulletin 2011/31 - European Patent Office

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(C07D) I.1(1)<br />

RAO, Ashwin, U., Avenel New Jersey 07001,<br />

US<br />

CHEN, Xiao, Edison New Jersey 08820, US<br />

LEE, Yoon, Joo, Scotch Plains New Jersey<br />

07076, US<br />

DEGRADO, Sylvia, Scotch Plains New Jersey<br />

07076, US<br />

SHAO, Ning, Clark New Jersey 07066, US<br />

HUANG, Ying, R., Berkeley Heights New<br />

Jersey 07922, US<br />

LIU, Zhidan, Edison New Jersey 08820, US<br />

(74) Buchan, Gavin MacNicol, et al, Merck & Co.,<br />

Inc. <strong>European</strong> <strong>Patent</strong> Department Hertford<br />

Road, Hoddesdon, Hertfordshire EN11 9BU,<br />

GB<br />

(51) C07D 401/12 (11) 2 350 049 A2*<br />

C07D 403/12 A61K <strong>31</strong>/415<br />

A61P 11/00 A61P 29/00<br />

(25) En (26) En<br />

(21) 09785724.7 (22) 02.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) GB 2009/051304 02.10.2009<br />

(87) WO 2010/038086 2010/14 08.04.2010<br />

(88) 24.06.2010<br />

(30) 02.10.2008 GB 0818033<br />

11.12.2008 GB 0822609<br />

(54) • P38-MAP-KINASE-INHIBITOREN<br />

• P38 MAP KINASE INHIBITORS<br />

• NOUVEAUX COMPOSÉS<br />

(71) Respivert Limited, 50-100 Holmers Farm<br />

Way, High Wycombe Buckinghamshire HP12<br />

4EG, GB<br />

(72) ITO, Kazuhiro, London SW7 2AZ, GB<br />

STRONG, Peter, London SW7 2AZ, GB<br />

RAPEPORT, William, Garth, London SW7<br />

2AZ, GB<br />

MURRAY, Peter, John, London SW7 2AZ,<br />

GB<br />

KING-UNDERWOOD, John, Worcestershire<br />

GL19 3PW, GB<br />

WILLIAMS, Jonathan, Gareth, Nottingham<br />

NG1 1GF, GB<br />

ONIONS, Stuart ,Thomas, Nottingham NG1<br />

1GF, GB<br />

HIRST, Simon, Christopher, Nottingham NG1<br />

1GF, GB<br />

TADDEI, David, Michel, Adrien, Nottingham<br />

NG1 1GF, GB<br />

CHARRON, Catherine, Elizabeth, London<br />

SW7 2AZ, GB<br />

(74) Teuten, Andrew John, et al, Sagittarius IP<br />

Taylor House 39 High Street, Marlow, Bucks<br />

SL7 1AF, GB<br />

(51) C07D 401/12 (11) 2 350 050 A1*<br />

A61K <strong>31</strong>/44 A61P 1/04<br />

(25) En (26) En<br />

(21) 09820279.9 (22) 13.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2009/063<strong>31</strong>4 13.10.2009<br />

(87) WO 2010/043601 2010/16 22.04.2010<br />

(30) 14.10.2008 EP 08166571<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

ENANTIOMERENANGEREICHERTEN PRO-<br />

TONENPUMPENHEMMERN<br />

• PROCESS FOR THE PREPARATION OF<br />

ENANTIOMERICALLY ENRICHED PROTON<br />

PUMP INHIBITORS<br />

• PROCÉDÉ POUR LA PRÉPARATION D'IN-<br />

HIBITEURS DE LA POMPE À PROTONS<br />

ENRICHIS DU POINT DE VUE DES ÉNAN-<br />

TIOMÈRES<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(71) LEK Pharmaceuticals d.d., Verovskova 57,<br />

1526 Ljubljana, SI<br />

(72) MOHAR, Barbara, 1526 Ljubljana, SI<br />

TOPLAK CASAR, Renata, 1526 Ljubljana, SI<br />

(74) Prüfer & Partner GbR <strong>European</strong> <strong>Patent</strong><br />

Attorneys, Sohnckestraße 12, 81479<br />

München, DE<br />

(51) C07D 401/12 (11) 2 350 051 A1*<br />

A61P 5/50 C07D 215/16<br />

A61K <strong>31</strong>/14 A61P 7/00<br />

C07D 401/14 A61K <strong>31</strong>/4427<br />

A61P 9/00 C07D 403/14<br />

A61K <strong>31</strong>/47 A61P 17/00<br />

C07D 405/12 A61K <strong>31</strong>/4709<br />

A61P 25/00 C07D 405/14<br />

A61K <strong>31</strong>/4995 A61P 27/00<br />

C07D 413/12 A61K <strong>31</strong>/506<br />

A61P 29/00 C07D 413/14<br />

(25) En (26) En<br />

(21) 09826554.9 (22) 29.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) US 2009/062649 29.10.2009<br />

(87) WO 2010/056549 2010/20 20.05.2010<br />

(30) 29.10.2008 US 197595 P<br />

(54) • PYRIDIN, BIZYKLISCHES PYRIDIN UND<br />

DEREN ANALOGE ALS SIRTUINMODULA-<br />

TOREN<br />

• PYRIDINE, BICYCLIC PYRIDINE AND<br />

RELATED ANALOGS AS SIRTUIN MODU-<br />

LATORS<br />

• PYRIDINE, PYRIDINE BICYCLIQUE ET<br />

ANALOGUES ASSOCIÉS EN TANT QUE<br />

MODULATEURS DE SIRTUINE<br />

(71) Sirtris Pharmaceuticals, Inc., 200 Technology<br />

Square, Suite 300, Cambridge, MA<br />

02139, US<br />

(72) NARAYAN, Radha, Cambridge, MA 02139,<br />

US<br />

DISCH, Jeremy, S., Cambridge, MA 02139,<br />

US<br />

PERNI, Robert, B., Cambridge, MA 02139,<br />

US<br />

VU, Chi, B., Cambridge, MA 02139, US<br />

(74) Chapman, Paul Gilmour, Marks & Clerk LLP<br />

Aurora 120 Bothwell Street, Glasgow G2<br />

7JS, GB<br />

C07D 401/12 → (51) A61P 3/10<br />

C07D 401/12 → (51) C07D 207/08<br />

C07D 401/12 → (51) C07D 207/16<br />

C07D 401/12 → (51) C07D 211/76<br />

C07D 401/12 → (51) C07D 211/96<br />

C07D 401/12 → (51) C07D 213/40<br />

C07D 401/12 → (51) C07D 213/81<br />

C07D 401/12 → (51) C07D 217/26<br />

(51) C07D 401/14 (11) 2 350 052 A2*<br />

C07D 413/14 C07D 417/14<br />

C07D 487/04 A61K <strong>31</strong>/4439<br />

A61P 35/00<br />

(25) En (26) En<br />

(21) 09783505.2 (22) 28.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

BA RS<br />

182<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

(86) EP 2009/062551 28.09.2009<br />

(87) WO 2010/034838 2010/13 01.04.2010<br />

(88) 18.11.2010<br />

(30) 29.09.2008 EP 08165437<br />

(54) • ANTIPROLIFERATIVE VERBINDUNGEN<br />

• ANTIPROLIFERATIVE COMPOUNDS<br />

• Composés antiprolifératifs<br />

(71) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(72) STEURER, Steffen, 55216 Ingelheim am<br />

Rhein, DE<br />

ETTMAYER, Peter, 55216 Ingelheim am<br />

Rhein, DE<br />

MANTOULIDIS, Andreas, 55216 Ingelheim<br />

am Rhein, DE<br />

(74) Hammann, Heinz, Boehringer Ingelheim<br />

GmbH CD <strong>Patent</strong>s Binger Strasse 173,<br />

55216 Ingelheim Am Rhein, DE<br />

(51) C07D 401/14 (11) 2 350 053 A2*<br />

C07D 403/14 C07D 487/04<br />

C07D 487/02 A61K <strong>31</strong>/4162<br />

A61P 3/00 A61P 3/04<br />

(25) En (26) En<br />

(21) 09820914.1 (22) 16.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/005656 16.10.2009<br />

(87) WO 2010/044885 2010/16 22.04.2010<br />

(88) 02.09.2010<br />

(30) 10.06.2009 US 185923 P<br />

20.10.2008 US 196772 P<br />

17.10.2008 US 106411 P<br />

(54) • LÖSLICHE MTOR-KOMPLEXE UND<br />

MODULATOREN DARAUS<br />

• SOLUBLE MTOR COMPLEXES AND MOD-<br />

ULATORS THEREOF<br />

• COMPLEXES MTOR SOLUBLES ET<br />

MODULATEURS ASSOCIÉS<br />

(71) Whitehead Institute For Biomedical<br />

Research, Nine Cambridge Center, Cambridge,<br />

MA 02142, US<br />

Dana-Farber Cancer Institute Inc., 44 Binney<br />

Street, Boston, MA 02115, US<br />

(72) GRAY, Nathanael, Boston MA 02130, US<br />

CHANG, Jae, Won, Boston MA 02120, US<br />

ZHANG, Jianming, Cambridge MA 02139, US<br />

THOREEN, Carson, C., Jamaica Plain MA<br />

02130, US<br />

KANG, Seong Woo, Anthony, Cambridge MA<br />

02139, US<br />

SABATINI, David, M., Cambridge MA 02138,<br />

US<br />

LIU, Qingsong, Jamaica Plain MA 02130, US<br />

(74) Chapman, Paul William, Kilburn & Strode<br />

LLP 20 Red Lion Street, GB-London WC1R<br />

4PJ, GB<br />

C07D 401/14 → (51) C07D 207/08<br />

C07D 401/14 → (51) C07D 207/16<br />

C07D 401/14 → (51) C07D 211/76<br />

C07D 401/14 → (51) C07D 211/96<br />

C07D 401/14 → (51) C07D 213/81<br />

C07D 401/14 → (51) C07D 235/02<br />

C07D 401/14 → (51) C07D 401/04<br />

C07D 401/14 → (51) C07D 401/12<br />

C07D 401/14 → (51) C07D 403/04

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