Bulletin 2011/31 - European Patent Office

(A61K) I.1(1)
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) US 2009/057363 17.09.2009
(87) WO 2010/033733 2010/12 25.03.2010
(30) 17.09.2008 US 97655 P
(54) • FOLATREZEPTOR-BINDUNGSKONJUGATE
VON ANTIFOLATEN
• FOLATE RECEPTOR BINDING CONJU-
GATES OF ANTIFOLATES
• CONJUGUÉS D'ANTIFOLATES LIANT LE
RÉCEPTEUR DE FOLATE
(71) Endocyte, Inc., 3000 Kent Avenue, West
Lafayette, IN 47906, US
Purdue Research Foundation, 1281 Win
Hentschel Boulevard, West Lafayette, IN
47096-4182, US
(72) LEAMON, Christopher, Paul, West Lafayette,
IN 47906, US
VLAHOV, Iontcho, Radoslavov, West Lafayette,
IN 47906, US
LOW, Philip, Stewart, West Lafayette, IN
47906, US
(74) Hart, Deborah Mary, et al, Kilburn & Strode
LLP 20 Red Lion Street, London WC1R 4PJ,
GB
A61K 31/517 → (51) C07D 239/91
A61K 31/519 → (51) A01N 43/90
A61K 31/519 → (51) A61K 31/155
A61K 31/519 → (51) A61K 31/195
A61K 31/519 → (51) A61K 31/437
A61K 31/519 → (51) C07D 471/04
A61K 31/519 → (51) C07D 473/34
A61K 31/519 → (51) C07D 487/04
A61K 31/519 → (51) C07D 487/12
A61K 31/519 → (51) C07D 495/04
A61K 31/519 → (51) C07D 513/04
A61K 31/52 → (51) C07D 473/34
A61K 31/522 → (51) A61K 9/22
A61K 31/522 → (51) A61K 31/155
A61K 31/525 → (51) A61K 31/195
A61K 31/535 → (51) C07D 471/22
A61K 31/5375 → (51) A61K 9/16
(51) A61K 31/5377 (11) 2 349 275 A1*
A61P 35/00
(25) En (26) En
(21) 09744391.5 (22) 29.10.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) EP 2009/064274 29.10.2009
(87) WO 2010/049481 2010/18 06.05.2010
(30) 31.10.2008 EP 08168044
(54) • KOMBINATION EINES PHOSPHATIDYLI-
NOSITOL-3-KINASE (PI3K) INHIBITORS
UND EINES MTOR-INHIBITORS
• COMBINATION OF A PHOSPHATIDYLINO-
SITOL-3-KINASE (PI3K) INHIBITOR AND A
MTOR INHIBITOR
Europäisches Patentblatt
European Patent Bulletin
Bulletin européen des brevets
• COMBINAISON D UN INHIBITEUR DE LA
PHOSPHATIDYLINOSITOL-3-KINASE
(PI3K) ET D UN INHIBITEUR DE MTOR
(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH
(72) GARCIA-ECHEVERRIA, Carlos, CH-4002
Basel, CH
MAIRA, Sauveur-Michel, CH-4002 Basel, CH
(74) Gruber, Markus, et al, Novartis Pharma AG
Patent Department, 4002 Basel, CH
A61K 31/5377 → (51) C07D 407/06
A61K 31/55 → (51) A01N 43/00
A61K 31/55 → (51) A61K 31/553
A61K 31/55 → (51) C07D 487/12
A61K 31/551 → (51) A61K 31/575
A61K 31/551 → (51) C07D 407/06
A61K 31/5517 → (51) C07D 487/04
(51) A61K 31/553 (11) 2 349 276 A2*
C07D 487/04 C07D 281/10
A61K 31/55 A61P 31/18
(25) En (26) En
(21) 09740569.0 (22) 02.10.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
AL BA RS
(86) US 2009/059308 02.10.2009
(87) WO 2010/042392 2010/15 15.04.2010
(88) 03.06.2010
(30) 06.10.2008 US 195271 P
(54) • HIV-INTEGRASEHEMMER
• HIV INTEGRASE INHIBITORS
• INHIBITEURS DE L'INTÉGRASE DU VIH
(71) Merck Sharp & Dohme Corp., 126 East
Lincoln Avenue, Rahway, NJ 07065-0907,
US
(72) ISAACS, Richard, C. A., Rahway New Jersey
07065-0907, US
THOMPSON, Wayne, J., Rahway New Jersey
07065-0907, US
WILLIAMS, Peter, D., Rahway New Jersey
07065-0907, US
SU, Dai-Shi, Rahway New Jersey 07065-
0907, US
VENKATRAMAN, Shankar, Rahway New
Jersey 07065-0097, US
EMBREY, Mark, W., Rahway New Jersey
07065-0907, US
FISHER, Thorsten, E., Rahway New Jersey
07065-0907, US
WAI, John, S., Rahway New Jersey 07065-
0907, US
DUBOST, David, C., Rahway New Jersey
07065-0907, US
BALL, Richard, G., Rahway New Jersey
07065-0907, US
CHOI, Eric, J., Rahway New Jersey 07065-
0907, US
PEI, Tao, Rahway New Jersey 07065-0907,
US
TRICE, Sarah, L., Rahway New Jersey
07065-0907, US
CAMPBELL, Neil, Rahway New Jersey
07065-0907, US
MADDESS, Matthew, Rahway New Jersey
07065-0907, US
MALIGRES, Peter, E., Rahway New Jersey
07065-0907, US
SHEVLIN, Michael, Rahway New Jersey
07065-0907, US
77
Anmeldungen
Applications
Demandes (31/2011) 03.08.2011
SONG, Zhiguo Jake, Rahway New Jersey
07065-0907, US
STEINHUEBEL, Dietrich, P., Rahway New
Jersey 07065-0907, US
STROTMAN, Neil, A., Rahway New Jersey
07065-0907, US
YIN, Jingjun, Rahway New Jersey 07065-
0907, US
(74) Horgan, James Michael Frederic, Merck &
Co., Inc. European Patent Department Hertford
Road, Hoddesdon EN11 9BU, GB
A61K 31/553 → (51) C07D 407/06
A61K 31/555 → (51) A61K 31/167
A61K 31/5575 → (51) A61K 31/155
(51) A61K 31/575 (11) 2 349 277 A2*
A61P 17/06 A61P 37/06
A61P 1/00 A61P 17/00
A61P 29/00 G01N 33/50
A61K 31/551 A61K 31/192
(25) En (26) En
(21) 09740864.5 (22) 28.10.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) EP 2009/007717 28.10.2009
(87) WO 2010/049144 2010/18 06.05.2010
(88) 08.07.2010
(30) 28.10.2008 EP 08018795
28.10.2008 US 108990 P
(54) • VERFAHREN ZUR IDENTIFIZIERUNG VON
NEUEN LIGANDEN ZUR MODULIERUNG
DER AKTIVITÄT VON NR1F3 ( ORPHAN
NUCLEAR RECEPTOR RAR-RELATED
ORPHAN RECEPTOR-GAMMA)
• METHODS OF IDENTIFICATION OF NOVEL
LIGANDS FOR MODULATION OF ORPHAN
NUCLEAR RECEPTOR RAR-RELATED
ORPHAN RECEPTOR-GAMMA (NR1F3)
ACTIVITY
• PROCÉDÉS D'IDENTIFICATION DE NOU-
VEAUX LIGANDS DESTINÉS À LA MODU-
LATION DE L'ACTIVITÉ DU RÉCEPTEUR
ORPHELIN GAMMA (NR1F3) EN FONC-
TION AU RÉCEPTEUR NUCLÉAIRE
ORPHELIN DU RÉCEPTEUR DE L'ACIDE
RÉTINOÏDE (RAR)
(71) Phenex Pharmaceuticals AG, J542N, Werksgelände
BASF, 67056 Ludwigshafen, DE
(72) DEUSCHLE, Ulrich, 67549 Worms, DE
ABEL, Ulrich, 69126 Heidelberg, DE
KREMOSER, Claus, 69121 Heidelberg, DE
SCHLUETER, Thomas, 69123 Heidelberg, DE
HOFFMANN, Thomas, 68519 Viernheim, DE
PEROVIC-OTTSTADT, Sanja, 65462 Ginsheim-Gustavsburg,
DE
(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser
Anwaltssozietät, Leopoldstrasse 4,
80802 München, DE
A61K 31/575 → (51) A61K 8/19
A61K 31/58 → (51) A61K 9/00
A61K 31/66 → (51) A01N 57/00
(51) A61K 31/665 (11) 2 349 278 A1*
A61K 31/7036 A61P 31/04
(25) En (26) En
(21) 09756875.2 (22) 16.10.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) US 2009/061033 16.10.2009
(87) WO 2010/048059 2010/17 29.04.2010
(30) 21.10.2008 US 107242 P