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Bulletin 2011/31 - European Patent Office

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(C07D) II.1(1)<br />

• PIPERIDINE-AMIDE DERIVATIVES<br />

• DÉRIVÉS DE PIPÉRIDINE-AMIDE<br />

(73) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) ANDJELKOVIC, Mirjana, CH-4055 Basel, CH<br />

CECCARELLI, Simona M., CH-4057 Basel,<br />

CH<br />

CHOMIENNE, Odile, F-68130 Altkirch, FR<br />

MATTEI, Patrizio, CH-4125 Riehen, CH<br />

(74) Waschbüsch, Klaus, F. Hoffmann-La Roche<br />

AG <strong>Patent</strong> Department (CLP) Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

C07D 417/06 → (51) C07D 235/26<br />

C07D 417/12 → (51) C07D 235/18<br />

C07D 417/12 → (51) C07D 285/18<br />

C07D 417/14 → (51) C07D 235/26<br />

C07D 417/14 → (51) C07D 401/12<br />

C07D 417/14 → (51) C07D 401/14<br />

(51) C07D 471/04 (11) 1 784 402 B1<br />

(25) En (26) En<br />

(21) 057811<strong>31</strong>.7 (22) 03.09.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 16.05.2007<br />

(86) KR 2005/002924 03.09.2005<br />

(87) WO 2006/025714 2006/10 09.03.2006<br />

(30) 03.09.2004 KR 20040070536<br />

(54) • PYRROLO[3,2-c]PYRIDINDERIVATE UND<br />

HERSTELLUNGSVERFAHREN DAFÜR<br />

• PYRROLO[3,2-c]PYRIDINE DERIVATIVES<br />

AND PROCESSES FOR THE PREPARATION<br />

THEREOF<br />

• DERIVES PYRROLO[3,2-C]PYRIDINE ET<br />

PROCEDES DE PREPARATION DE CES<br />

DERNIERS<br />

(73) Yuhan Corporation, 49-6 Taebang-dong,<br />

Tongjak-gu, Seoul 156-754, KR<br />

(72) KIM, Jae-Gyu, Seoul 152-859, KR<br />

AHN, Byung-Nak, Seoul 121-040, KR<br />

LEE, Hyouk-Woo, 234-701, Hanwha Dreamgrenn<br />

Apt., Hwaseong-si, Gyeonggi-do 445-<br />

735, KR<br />

YOON, Suk-Won, Seoul 156-090, KR<br />

YOON, Young-Ae, 502-1006 Munrae Hyundai<br />

5cha Apt., Seoul 150-959, KR<br />

KIM, Dong-Hoon, Gunpo-city, Kyungki-do<br />

435-839, KR<br />

KEUM, Se-Hoon, Seoul 156-805, KR<br />

SHIN, Young-Ah, 113-103 Samsung Raemian<br />

1cha Apt., Yongin-city, Kyungki-do<br />

449-557, KR<br />

KANG, Heui-Il, Gunpo-city, Kyungki-do 435-<br />

047, KR<br />

CHOI, Ryong, Deceased, KR<br />

(74) Turner, Craig Robert, et al, A.A. Thornton &<br />

Co. 235 High Holborn, London WC1V 7LE,<br />

GB<br />

(51) C07D 471/04 (11) 1 888 579 B1<br />

(25) Fr (26) Fr<br />

(21) 06755509.4 (22) 19.05.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 20.02.2008<br />

(86) FR 2006/001137 19.05.2006<br />

(87) WO 2006/123061 2006/47 23.11.2006<br />

(30) 19.05.2005 FR 0505037<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(54) • NEUE FLUORENDERIVATE, ZUSAMMEN-<br />

SETZUNG MIT DIESEN DERIVATEN UND<br />

VERWENDUNG<br />

• NOVEL FLUORENE DERIVATIVES, COM-<br />

POSITION CONTAINING SAID DERIVA-<br />

TIVES AND THE USE THEREOF<br />

• NOUVEAUX DERIVES DU FLUORENE,<br />

COMPOSITIONS LES CONTENANT ET<br />

UTILISATION<br />

(73) Aventis Pharma S.A., 20, avenue Raymond<br />

Aron, 92160 Antony, FR<br />

(72) MAILLIET, Patrick, F-94120 Fontenay Sous<br />

Bois, FR<br />

BERTIN, Luc, F-91560 Crosnes, FR<br />

GUYON, Thierry, F-91270 Vigneux Sur Seine,<br />

FR<br />

THOMPSON, Fabienne, F-75012 Paris, FR<br />

RUXER, Jean-Marie, F-92130 Issy Les<br />

Moulineaux, FR<br />

PILORGE, Fabienne, F-77220 Tournan En<br />

Brie, FR<br />

BENARD, Didier, F-95560 Montsoult, FR<br />

MINOUX, Hervé, F-94320 Thiais, FR<br />

CARREZ, Chantal, F-94320 Thiais, FR<br />

GOULAOUIC, Hélène, F-75012 Paris, FR<br />

(74) Le Coupanec, Pascale A.M.P., et al, Nony &<br />

Associés 3, rue de Penthièvre, 75008 Paris,<br />

FR<br />

(51) C07D 471/04 (11) 1 893 612 B1<br />

A61K <strong>31</strong>/435 C07C 49/517<br />

A61P 35/00<br />

(25) En (26) En<br />

(21) 06773861.7 (22) 21.06.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

RS<br />

(43) 05.03.2008<br />

(86) US 2006/024524 21.06.2006<br />

(87) WO 2007/002433 2007/01 04.01.2007<br />

(30) 22.06.2005 US 692960 P<br />

28.10.2005 US 7<strong>31</strong>528 P<br />

(54) • PYRROLO[2,3-B]PYRIDINDERIVATE ALS<br />

PROTEINKINASEINHIBITOREN<br />

• PYRROLO [2, 3-B]PYRIDINE DERIVA-<br />

TIVES AS PROTEIN KINASE INHIBITORS<br />

• DERIVES DE PYRROLO [2, 3-B]PYRIDINE<br />

UTILISES COMME INHIBITEURS DE PRO-<br />

TEINES KINASES<br />

(73) PLEXXIKON, INC., 91 Bolivar Drive, Suite A,<br />

Berkeley, CA 94710, US<br />

(72) IBRAHIM, Prabha, N., Mountain View, CA<br />

94040, US<br />

ARTIS, Dean, R., Kensington, CA 94707, US<br />

BREMER, Ryan, Oakland, CA 94610, US<br />

HABETS, Gaston, Pleasant Hill, CA 94523,<br />

US<br />

MAMO, Shumeye, Oakland, CA 94619, US<br />

NESPI, Marika, Berkeley, CA 94707, US<br />

ZHANG, Chao, Moraga, CA 94556, US<br />

ZHANG, Jiazhong, Foster City, CA 94404, US<br />

ZHU, Yong-Liang, Fremont, CA 94539, US<br />

ZUCKERMAN, Rebecca, Alameda, CA 94501,<br />

US<br />

WEST, Brian, San Francisco, CA 94110, US<br />

SUZUKI, Yoshihisa, San Pablo, CA 94806,<br />

US<br />

TSAI, James, Vallejo, CA 94591, US<br />

HIRTH, Klaus-Peter, San Francisco, CA<br />

94114, US<br />

BOLLAG, Gideon, Orinda, CA 94563, US<br />

SPEVAK, Wayne, Berkeley, CA 94708, US<br />

CHO, Hanna, Oakland, CA 94610, US<br />

GILLETTE, Samuel, J., Oakland, CA 94610,<br />

US<br />

WU, Guoxian, Palo Alto, CA 94306, US<br />

ZHU, Hongyao, Berkeley, CA 94710, US<br />

779<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

SHI, Shenghua, San Diego, California 92130,<br />

US<br />

(74) Zimmermann & Partner, Postfach 330 920,<br />

80069 München, DE<br />

(51) C07D 471/04 (11) 2 125 807 B1<br />

A61K <strong>31</strong>/4355<br />

(25) En (26) En<br />

(21) 07855374.0 (22) 14.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 02.12.2009<br />

(86) BE 2007/000127 14.12.2007<br />

(87) WO 2008/070937 2008/25 19.06.2008<br />

(30) 14.12.2006 GB 0624983<br />

(54) • ALS PESTIVIRUS-INHIBITOREN GEEIG-<br />

NETE IMIDAZO[1,2-A]PYRROLO[3,2-C]<br />

PYRIDINVERBINDUNGEN<br />

• IMIDAZO[1,2-A]PYRROLO[3,2-C]PYRI-<br />

DINE COMPOUNDS USEFUL AS PESTI-<br />

VIRUS INHIBITORS<br />

• IMIDAZO[1,2-A]PYRROLO[3,2-C]PYRIDI-<br />

NES EN TANT QU'INHIBITEURS DE PES-<br />

TIVIRUS<br />

(73) Katholieke Universiteit Leuven, K.U. Leuven<br />

R&D Minderbroedersstraat 8A - bus 5105,<br />

3000 Leuven, BE<br />

Université D'Auvergne Clermont 1, Dept. de<br />

valorisation et transfert de techologies<br />

Pierre-Charles Romond -5eme étage CBRV<br />

Faculté de Médicine et de Pharmacie 28<br />

place H. Dunant, 63001 Clermont-Ferrand,<br />

FR<br />

Université Francois Rabelais de Tours, 3, rue<br />

des Tanneurs, 37041 Tours Cedex 1, FR<br />

(72) NEYTS, Johan, 3010 Kessel-Lo, BE<br />

PAESHUYSE, Jan, 3010 Kessel-Lo, BE<br />

CHAVIGNON, Olivier, 63001 Clermont-Ferrand,<br />

FR<br />

CHEZAL, Jean-Michel, 63001 Clermont-Ferrand,<br />

FR<br />

GAUMET, Vincent, 63001 Clermont-Ferrand,<br />

FR<br />

GUEIFFIER, Alain, 37200 Tours, FR<br />

TEULADE, Jean-Claude, 63001 Clermont-<br />

Ferrand, FR<br />

(74) Bird, William Edward, et al, Bird Goën & Co<br />

Klein Dalenstraat 42A, 3020 Winksele, BE<br />

(51) C07D 471/08 (11) 2 194 056 B1<br />

A61K <strong>31</strong>/551 A61P 25/00<br />

(25) En (26) En<br />

(21) 10154049.0 (22) 29.05.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 09.06.2010<br />

(30) 30.05.2006 DK 2006007<strong>31</strong><br />

30.05.2006 US 809024 P<br />

(54) • Neue 1,4-diaza-bicyclo[3.2.2]nonyl-oxadiazolyl-Derivate<br />

und deren medizinische<br />

Verwendung<br />

• Novel 1,4-diaza-bicyclo[3.2.2]nonyl oxadiazolyl<br />

derivatives and their medical use<br />

• Nouveaux dérivés 1,4-diaza-bicyclo[3.2.2]<br />

nonyl-oxadiazolyle et leur utilisation médicale<br />

(73) NeuroSearch A/S, Pederstrupvej 93, 2750<br />

Ballerup, DK<br />

(72) Peters, Dan, 2750 Ballerup, DK<br />

Olsen, Gunnar, M., 2765 Smørum, DK<br />

Nielsen, Elsebet, Østergaard, 2750 Ballerup,<br />

DK<br />

Timmermann, Daniel, B., 2750 Ballerup, DK<br />

Loechel, Steven, Charles, 2000 Frederiksberg,<br />

DK<br />

Mikkelsen, Jens, Damsgaard, 2750 Ballerup,<br />

DK

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