Bulletin 2011/31 - European Patent Office

(A61K) II.1(1)
(43) 02.11.2000
(86) FR 1999/000059 14.01.1999
(87) WO 1999/036066 1999/29 22.07.1999
(30) 16.01.1998 FR 9800453
(54) • PHARMAZEUTISCHE ZUSAMMENSET-
ZUNG, DIE EINEN SPEZIFISCHEN AMINO-
PEPTIDASE-A INHIBITOR ENTHÄLT,
INSBESONDERE EC33, ZUR SENKUNG
DES BLUTDRUCKS
• PHARMACEUTICAL COMPOSITION COM-
PRISING A SPECIFIC INHIBITOR OF AMI-
NOPEPTIDASE A, IN PARTICULAR EC33,
FOR DECREASING BLOOD PRESSURE
• COMPOSITION PHARMACEUTIQUE COM-
PRENANT UN INHIBITEUR SPÉCIFIQUE DE
L'AMINOPEPTIDASE A, EN PARTICULIER
L'EC33, POUR DIMINUER LA PRESSION
ARTÉRIELLE
(73) INSTITUT NATIONAL DE LA SANTE ET DE
LA RECHERCHE MEDICALE (INSERM), 101,
rue de Tolbiac, 75013 Paris, FR
CENTRE NATIONAL DE LA RECHERCHE
SCIENTIFIQUE (CNRS), 3, rue Michel-Ange,
75794 Paris Cedex 16, FR
(72) LLORENS-CORTES, Catherine, F-91440
Bures sur Yvette, FR
CORVOL, Pierre, F-75015 Paris, FR
FOURNIE-ZALUSKI, Marie-Claude, F-75011
Paris, FR
ROQUES, Bernard, Pierre, F-75014 Paris, FR
(74) Le Coupanec, Pascale A.M.P., et al, Cabinet
Lavoix 2, place d'Estienne d'Orves, 75441
Paris Cedex 09, FR
(51) A61K 31/185 (11) 2 004 168 B1
A61K 31/215 A61K 45/06
A61K 9/28 A61P 5/16
(25) En (26) En
(21) 07723634.7 (22) 27.03.2007
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IS IT LI LT LU LV MC MT NL PL PT
RO SE SI SK TR
(43) 24.12.2008
(86) EP 2007/002688 27.03.2007
(87) WO 2007/110226 2007/40 04.10.2007
(30) 28.03.2006 GB 0606212
(54) • STABILE ORALE PHARMAZEUTISCHE
ZUSAMMENSETZUNG MIT THYROIDHOR-
MONREZEPTORAGONISTEN
• STABLE ORAL PHARMACEUTICAL COM-
POSITION CONTAINING THYROID HOR-
MONE RECEPTOR AGONISTS
• COMPOSITION PHARMACEUTIQUE ORALE
STABLE CONTENANT DES AGONISTES
DES RÉCEPTEURS DES HORMONES
THYROÏDIENNES
(73) KARO BIO AB, Novum, 141 57 Huddinge, SE
Bristol-Myers Squibb Company, P.O. Box
4000, Princeton NJ 08543-4000, US
(72) GARG, Neeraj, S-141 57 Huddinge, SE
RAO, VENKATRAMANA M., Edison, NJ
08820, US
GANDHI, Rajesh, B., Plainsboro, NJ 08536,
US
WASHBURN, William N., Titusville, NJ
08560, US
KOEHLER, Konrad, 30161 Hannover, DE
MALM, Johan, S-142 66 Trängsund, SE
(74) Brady, Paul Andrew, et al, Abel & Imray 20
Red Lion Street, London WC1R 4PQ, GB
(51) A61K 31/192 (11) 1 976 502 B1
A61K 31/436 A61P 25/04
A61P 9/10
(25) En (26) En
(21) 06846858.6 (22) 29.12.2006
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IS IT LI LT LU LV MC NL PL PT RO
SE SI SK TR
Europäisches Patentblatt
European Patent Bulletin
Bulletin européen des brevets
(43) 08.10.2008
(86) US 2006/062715 29.12.2006
(87) WO 2007/079406 2007/28 12.07.2007
(30) 30.12.2005 US 755315 P
23.06.2006 US 426282
(54) • KLEINMOLEKULARE HEMMER VON PDZ-
WECHSELWIRKUNGEN
• SMALL MOLECULE INHIBITORS OF PDZ
INTERACTIONS
• PETITES MOLECULES INHIBITRICES DES
INTERACTIONS DU DOMAINE PDZ
(73) Arbor Vita Corporation, 6611 Dumbarton
Circle, Fremont, CA 94555, US
(72) BELMARES, Michael P., San Jose, CA
95129, US
LU, Peter S., Palo Alto, CA 94301, US
MENDOZA, Kenneth A., Oakland, CA 94610,
US
(74) Dehmel, Albrecht, Dehmel & Bettenhausen
Patentanwälte Herzogspitalstrasse 11, 80331
München, DE
A61K 31/198 → (51) A61K 9/08
A61K 31/198 → (51) C07K 16/30
(51) A61K 31/205 (11) 2 222 293 B1
A61P 9/00 A61P 9/10
(25) En (26) En
(21) 08857026.2 (22) 03.12.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA RS
(43) 01.09.2010
(86) EP 2008/066711 03.12.2008
(87) WO 2009/071585 2009/24 11.06.2009
(30) 04.12.2007 EP 07122272
04.12.2007 EP 07122273
(54) • MEDIZINISCHE VERWENDUNG VON 3-
(2,2,2-TRIMETHYLHYDRAZINIUM) PRO-
PIONATHYDROGENFUMARAT UND
DIHYDROGENPHOSPHAT
• MEDICAL USE OF 3-(2,2,2-TRIMETHYL-
HYDRAZINIUM) PROPIONATE HYDROGEN
FUMARATE AND DIHYDROGEN PHOS-
PHATE
• NOUVEL USAGE MÉDICAL DES SELS DE
3-(2,2,2-TRIMÉTHYLHYDRAZINIUM)
PROPIONATE
(73) Grindeks, a joint stock company, 53, Krustpils
Street, Riga 1057, LV
(72) STONANS, Ilmars, LV-1057 Riga, LV
TARARAK, Eduard, Moscow 121609, RU
ANDREYEVA, Elena, Moscow 121614, RU
A61K 31/215 → (51) A61K 31/185
(51) A61K 31/277 (11) 1 480 634 B1
A61P 13/08 A61P 5/26
A61K 31/32 A61K 31/165
(25) En (26) En
(21) 03737647.2 (22) 06.02.2003
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IT LI LU MC NL PT SE SI SK TR
(43) 01.12.2004
(86) US 2003/003447 06.02.2003
(87) WO 2003/065992 2003/33 14.08.2003
(30) 07.02.2002 US 354300 P
11.03.2002 US 362997 P
(54) • Selective Androgen-Rezeptor-Modulatoren
(SARMs) für die Behandlung der benignen
Prostatahyperplasie
• Selective androgen receptor modulators
(SARMs) for treating benign prostate
hyperplasia
• Modulateurs sélectifs de récepteur androgène
(SARMs) pour le traitement de
l'hypertrophie bénigne de la prostate.
727
Patente
Patents
Brevets (31/2011) 03.08.2011
(73) University of Tennessee Research Foundation,
211 Conference Center Building 600
Henley Street, Knoxville, TN 37996, US
(72) STEINER, Mitchell, S., Germantown, TN
38138, US
VEVERKA, Karen, A., Cordova, TN 38018, US
MILLER, Duane, D., Germantown, TN 38139,
US
DALTON, James, T., Upper Arlington, OH
43221, US
CHUNG, Kiwon, Collierville, TN 38017, US
GAO, Wenqing, Columbus, OH 43221, US
(74) Lord, Hilton David, Marks & Clerk LLP 90
Long Acre, London WC2E 9RA, GB
A61K 31/32 → (51) A61K 31/277
A61K 31/341 → (51) A61P 31/04
A61K 31/343 → (51) A61P 31/04
A61K 31/352 → (51) A61P 31/04
A61K 31/381 → (51) A61P 31/04
A61K 31/4025 → (51) A61P 31/04
A61K 31/404 → (51) C07D 209/08
A61K 31/404 → (51) C07D 209/88
A61K 31/415 → (51) C07D 235/18
A61K 31/4155 → (51) A61P 31/04
A61K 31/416 → (51) C07D 231/56
A61K 31/4166 → (51) C07D 401/12
A61K 31/4168 → (51) C07D 235/30
A61K 31/4184 → (51) A61P 31/04
A61K 31/4184 → (51) C07D 235/26
A61K 31/4192 → (51) A61P 31/04
A61K 31/42 → (51) C07D 261/20
A61K 31/421 → (51) C07D 263/48
A61K 31/422 → (51) A61P 31/04
A61K 31/423 → (51) A61P 31/04
A61K 31/424 → (51) A61K 31/5365
A61K 31/4245 → (51) A61P 31/04
A61K 31/427 → (51) A61P 31/04
A61K 31/428 → (51) A61P 31/04
A61K 31/429 → (51) A61P 31/04
A61K 31/435 → (51) C07D 401/12
A61K 31/435 → (51) C07D 471/04
A61K 31/4355 → (51) C07D 471/04
A61K 31/436 → (51) A61K 31/192
A61K 31/44 → (51) C07C 237/22
A61K 31/44 → (51) C07F 9/58
A61K 31/4439 → (51) C07D 235/18