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Bulletin 2011/31 - European Patent Office

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(C07D) I.1(2)<br />

YOSHIKAWA, Naoki, Osaka-shi Osaka 553-<br />

0002, JP<br />

KUGIMIYA, Akira, Osaka-shi Osaka 553-<br />

0002, JP<br />

NAKAJIMA, Mado, Osaka-shi Osaka 553-<br />

0002, JP<br />

TANAKA, Nobuyuki, Osaka-shi Osaka 553-<br />

0002, JP<br />

(74) Webster, Jeremy Mark, et al, Mewburn Ellis<br />

LLP 33 Gutter Lane, London EC2V 8AS, GB<br />

C07D 239/26 → (51) C07D 213/30<br />

C07D 239/52 → (51) C07C 237/44<br />

(51) C07D 241/44 (11) 2 351 745 A1<br />

C07D 401/12 C07D 403/12<br />

C07D 407/12 C07D 409/12<br />

C07D 413/12 C07D 417/12<br />

C07D 471/04<br />

(25) En (26) En<br />

(21) 10184144.3 (22) 25.08.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK RS<br />

(30) 26.08.2005 US 711873 P<br />

26.08.2005 EP 05107838<br />

(54) • Pyrazinderivate und deren Verwendung als<br />

PI3K-Hemmer<br />

• Pyrazine derivatives and use as PI3K<br />

inhibitors<br />

• Dérivés de pyrazine et leurs utilisations en<br />

tant qu'inhibiteurs de PI3K<br />

(71) Merck Serono S.A., Centre Industriel, 1267<br />

Coinsins, CH<br />

(72) Gaillard, Pascale, 74160 Collonges s/s<br />

Salève, FR<br />

Quattropani, Anna, CH-1207 Geneva, CH<br />

Pomel, Vincent, 74570 Groisy, FR<br />

Rueckle, Thomas, 01220 Divonne-les-Bains,<br />

FR<br />

Klicic, Jasna, 88400 Biberach, DE<br />

Church, Dennis, CH-1291 Commugny, CH<br />

(62) 06793019.8 / 1 917 252<br />

C07D 249/04 → (51) C07D 307/46<br />

C07D 261/18 → (51) C07D 307/46<br />

C07D 263/34 → (51) C07D 307/46<br />

C07D 263/56 → (51) C07D 235/16<br />

C07D 275/02 → (51) C07D 307/46<br />

C07D 277/56 → (51) C07D 307/46<br />

C07D 277/64 → (51) C07D 235/16<br />

C07D 285/06 → (51) C07D 307/46<br />

(51) C07D 295/084 (11) 2 351 746 A1<br />

A61K <strong>31</strong>/495 A61P 25/24<br />

(25) Zh (26) En<br />

(21) 09818779.2 (22) 29.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) CN 2009/074<strong>31</strong>4 29.09.2009<br />

(87) WO 2010/040<strong>31</strong>5 2010/15 15.04.2010<br />

(30) 07.10.2008 CN 200810043821<br />

(54) • 1-BUTYL-2-HYDROXYARALKYL-PIPERA-<br />

ZIN-DERIVATE UND IHRE VERWENDUNG<br />

ALS ANTIDEPRESSIVA<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

• THE 1-BUTYL-2-HYDROXYARALKYL<br />

PIPERAZINE DERIVATIVES AND THE USES<br />

AS ANTI-DEPRESSION MEDICINE<br />

THEREOF<br />

• DÉRIVÉS DE 1-BUTYL-2-HYDROXYARAL-<br />

KYLPIPÉRAZINE ET LEURS UTILISATIONS<br />

COMME MÉDICAMENT ANTIDÉPRESSEUR<br />

(71) CSPC Zhongqi Pharmaceutical Technology<br />

(Shijiazhuang) Co., Ltd., No. 276 Zhongshan<br />

West Road Shijiazhuang, Hebei 050051, CN<br />

Shanghai Institute of Pharmaceutical Industry,<br />

No. 1320 Beijing West Road, Shanghai<br />

200040, CN<br />

(72) LI, Jianqi, Shanghai 200040, CN<br />

LV, Na, Shanghai 200040, CN<br />

JIN, Hua, Shanghai 200040, CN<br />

WENG, Zhijie, Shanghai 200040, CN<br />

ZHENG, Yongyong, Shanghai 200040, CN<br />

(74) Eisenführ, Günther, et al, Eisenführ, Speiser<br />

& Partner <strong>Patent</strong>anwälte Rechtsanwälte<br />

Postfach 10 60 78, 28060 Bremen, DE<br />

(51) C07D 307/46 (11) 2 351 747 A1<br />

C07D 249/04 C07D 333/38<br />

C07D 207/34 C07D 263/34<br />

C07D 277/56 C07D 2<strong>31</strong>/14<br />

C07D 233/90 C07D 261/18<br />

C07D 275/02 C07D 285/06<br />

A01N 43/08 A01N 43/10<br />

A01N 43/36 A01N 43/50<br />

A01N 43/56 A01N 43/707<br />

A01N 43/76 A01N 43/78<br />

A01N 43/80<br />

(25) En (26) En<br />

(21) 11163592.6 (22) 15.11.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK RS<br />

(30) 01.02.2006 EP 06356008<br />

(54) • Dérivés de N-cycloalkyl-benzylamide utiles<br />

comme fongicides<br />

• Fungicide n-cycloalkyl-benzyl-amide derivatives<br />

• N-cycloalkyl-Benzylamid-Verbindungen als<br />

Fungizide<br />

(71) Bayer CropScience AG, Alfred-Nobel-Straße<br />

50, 40789 Monheim, DE<br />

(72) Carbonne, Stéphane, 69480 Lucenay, FR<br />

Coqueron, Pierre-Yves, 69003 Lyon, FR<br />

Desbordes, Philippe, 69006 Lyon, FR<br />

Dunkel, Ralf, 42799 Leichlingen-Krähwinkel,<br />

DE<br />

Gary, Stéphanie, 69410 Champagne-Au-<br />

Mont-d'Or, FR<br />

Grosjean-Cournoyer, Marie-Claire, 69250<br />

Curis Au Mont d'Or, FR<br />

Tuch, Arounarith, 69009 Lyon, FR<br />

Mansfield, Darren, 51515 Kürten, DE<br />

Villier, Alain, 69660 Collonges Au Mont d'<br />

Or, FR<br />

Vors, Jean-Pierre, 69110 Sainte Foy-Les-<br />

Lyon, FR<br />

(74) Guitton, Carole, <strong>Patent</strong>s & Licensing Dpt. 14<br />

Impasse Pierre Baizet, 69009 Lyon, FR<br />

(62) 06807817.9 / 1 981 866<br />

C07D 307/79 → (51) C07D 209/14<br />

C07D <strong>31</strong>1/66 → (51) C07C 51/43<br />

C07D 333/38 → (51) C07D 307/46<br />

C07D 333/52 → (51) C07D 209/14<br />

(51) C07D 401/04 (11) 2 351 748 A1<br />

A61K <strong>31</strong>/4725 A61P 1/04<br />

409<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

A61P 1/16 A61P 3/00<br />

A61P 9/00 A61P 9/12<br />

A61P 11/00 A61P 11/06<br />

A61P 13/10 A61P 17/00<br />

A61P 19/02 A61P 19/10<br />

A61P 25/00 A61P 25/14<br />

A61P 25/16 A61P 25/18<br />

A61P 25/24 A61P 25/28<br />

A61P 27/14<br />

(25) Ja (26) En<br />

(21) 09819245.3 (22) 08.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2009/067546 08.10.2009<br />

(87) WO 2010/041711 2010/15 15.04.2010<br />

(30) 09.10.2008 JP 2008262340<br />

(54) • ISOCHINOLINDERIVAT UND DIESES ALS<br />

WIRKSTOFF ENTHALTENDER PDE-HEM-<br />

MER<br />

• ISOQUINOLINE DERIVATIVE, AND PDE<br />

INHIBITOR COMPRISING SAME AS<br />

ACTIVE INGREDIENT<br />

• DÉRIVÉ D'ISOQUINOLÉINE ET INHIBITEUR<br />

DE LA PDE LE COMPORTANT EN TANT QU<br />

INGRÉDIENT ACTIF<br />

(71) Kyorin Pharmaceutical Co., Ltd., 5, Kanda<br />

Surugadai 2-chome Chiyoda-ku, Tokyo 101-<br />

8<strong>31</strong>1, JP<br />

(72) KOHNO Yasushi, Shimotsuga-gun Tochigi<br />

329-0114, JP<br />

TAKITA Satoshi, Shimotsuga-gun Tochigi<br />

329-0114, JP<br />

KOJIMA Akihiko, Shimotsuga-gun Tochigi<br />

329-0114, JP<br />

(74) Weinberger, Rudolf, et al, Vossius & Partner<br />

Siebertstrasse 4, 81675 München, DE<br />

C07D 401/06 → (51) C07D 209/14<br />

(51) C07D 401/12 (11) 2 351 749 A1<br />

A61K <strong>31</strong>/496 A61P 7/12<br />

A61P 13/00 A61P 13/08<br />

A61P 13/10 A61P 25/20<br />

C07D 405/12 C07D 409/12<br />

C07D 417/12<br />

(25) Ja (26) En<br />

(21) 09824819.8 (22) 05.11.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) JP 2009/068902 05.11.2009<br />

(87) WO 2010/05<strong>31</strong>20 2010/19 14.05.2010<br />

(30) 06.11.2008 JP 2008285466<br />

(54) • CARBAMATVERBINDUNG ODER SALZ<br />

DAVON<br />

• CARBAMATE COMPOUND OR SALT<br />

THEREOF<br />

• COMPOSÉ DE CARBAMATE OU SON SEL<br />

(71) Astellas Pharma Inc., 3-11, Nihonbashi-<br />

Honcho 2-chome Chuo-ku, Tokyo 103-8411,<br />

JP<br />

(72) ISHII, Takahiro, Tokyo 103-8411, JP<br />

SUGANE, Takashi, Tokyo 103-8411, JP<br />

MUNAKATA, Ryosuke, Tokyo 103-8411, JP<br />

AOKI, Satoshi, Tokyo 103-8411, JP<br />

HIGAKI, Masahide, Tokyo 103-8411, JP<br />

SOMEYA, Akiyoshi, Tokyo 103-8411, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München, DE<br />

C07D 401/12 → (51) C07D 241/44<br />

(51) C07D 401/14 (11) 2 351 750 A1<br />

C09K 11/06 H05B 33/14<br />

H05B 33/22

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