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Bulletin 2011/31 - European Patent Office

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(C07D) II.1(1)<br />

C07D 401/04 → (51) C07D 295/125<br />

C07D 401/06 → (51) C07D 2<strong>31</strong>/56<br />

C07D 401/06 → (51) C07D 235/26<br />

C07D 401/06 → (51) C07D 295/125<br />

(51) C07D 401/12 (11) 1 794 146 B1<br />

C07D 403/12 A61K <strong>31</strong>/519<br />

A61K <strong>31</strong>/4166 A61P 25/06<br />

(25) En (26) En<br />

(21) 05796599.8 (22) 09.09.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 13.06.2007<br />

(86) US 2005/032288 09.09.2005<br />

(87) WO 2006/0<strong>31</strong>676 2006/12 23.03.2006<br />

(30) 13.09.2004 US 609294 P<br />

(54) • TRICYCLISCHE ANILID-SPIROHYDAN-<br />

TOIN-CGRP-REZEPTORANTAGONISTEN<br />

• TRICYCLIC ANILIDE SPIROHYDANTOIN<br />

CGRP RECEPTOR ANTAGONISTS<br />

• ANTAGONISTE DES RECEPTEURS CGRP<br />

SPIROHYDANTOIN ANILIDE TRICYCLIQUE<br />

(73) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) BELL, Ian, M., Rahway, New Jersey 07065-<br />

0907, US<br />

GALLICCHIO, Steven, N., Rahway, New<br />

Jersey 07065-0907, US<br />

ZARTMAN, C. Blair, Rahway, New Jersey<br />

07065-0907, US<br />

THEBERGE, Cory, R., Rahway, New Jersey<br />

07065-0907, US<br />

ZHANG, Xufang, Rahway, New Jersey<br />

07065-0907, US<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

(51) C07D 401/12 (11) 1 948 638 B1<br />

A61K <strong>31</strong>/4709 A61P 29/00<br />

(25) En (26) En<br />

(21) 06789659.7 (22) 10.08.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 30.07.2008<br />

(86) US 2006/0<strong>31</strong>151 10.08.2006<br />

(87) WO 2007/021803 2007/08 22.02.2007<br />

(30) 12.08.2005 US 707653 P<br />

(54) • VERBINDUNGEN ZUR BEHANDLUNG<br />

ENTZÜNDLICHER ERKRANKUNGEN<br />

• COMPOUNDS FOR THE TREATMENT OF<br />

INFLAMMATORY DISORDERS<br />

• COMPOSES POUR TRAITER DES MALA-<br />

DIES INFLAMMATOIRES<br />

(73) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033-0530, US<br />

(72) ZHU, Zhaoning, Plainsboro, New Jersey<br />

08536, US<br />

MAZZOLA, Robert, D., Stewartsville, NJ<br />

08886, US<br />

YU, Wensheng, Edison, New Jersey 08820,<br />

US<br />

KOZLOWSKI, Joseph, A., Princeton, New<br />

Jersey 08540, US<br />

(74) Jaap, David Robert, et al, MSD Hertford<br />

Road, Hoddesdon, Herts EN11 9BU, GB<br />

(51) C07D 401/12 (11) 2 125 782 B1<br />

C07D 401/14 C07D 405/14<br />

C07D 417/14 A61K <strong>31</strong>/435<br />

A61P 29/00 A61P <strong>31</strong>/18<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(25) En (26) En<br />

(21) 08709083.3 (22) 18.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(43) 02.12.2009<br />

(86) EP 2008/051951 18.02.2008<br />

(87) WO 2008/101905 2008/35 28.08.2008<br />

(30) 19.02.2007 EP 07102622<br />

(54) • ARYLCARBONSÄURECYCLOHEXYLAMID-<br />

DERIVATE<br />

• ARYL CARBOXYLIC ACID CYCLOHEXYL<br />

AMIDE DERIVATIVES<br />

• DÉRIVÉS CYCLOHEXYL AMIDE D'ACIDE<br />

CARBOXYLIQUE ARYLE<br />

(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) HERSPERGER, René, CH-4142 Münchenstein,<br />

CH<br />

JANSER, Philipp, CH-4053 Basel, CH<br />

MILTZ, Wolfgang, CH-4054 Basel, CH<br />

(74) von Sprecher, Georg, et al, Novartis Pharma<br />

AG <strong>Patent</strong> Department, 4002 Basel, CH<br />

C07D 401/12 → (51) C07D 221/16<br />

C07D 401/12 → (51) C07D 235/18<br />

(51) C07D 401/14 (11) 1 853 587 B1<br />

C07D 413/14 C07D 417/14<br />

A61K <strong>31</strong>/497 A61P <strong>31</strong>/00<br />

A61P 29/00<br />

(25) En (26) En<br />

(21) 06735003.3 (22) 14.02.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 14.11.2007<br />

(86) US 2006/005128 14.02.2006<br />

(87) WO 2006/088840 2006/34 24.08.2006<br />

(30) 16.02.2005 US 653332 P<br />

(54) • NEUE HETEROZYKLISCHE SUBSTITU-<br />

IERTE PYRIDIN- ODER PHENYLVERBIN-<br />

DUNGEN MIT CXCR3-<br />

ANTAGONISTISCHER AKTIVITÄT<br />

• NOVEL HETEROCYCLIC SUBSTITUTED<br />

PYRIDINE OR PHENYL COMPOUNDS<br />

WITH CXCR3 ANTAGONIST ACTIVITY<br />

• NOUVEAUX COMPOSES PYRIDINE OU<br />

PHENYLE SUBSTITUES HETEROCYCLI-<br />

QUES A ACTIVITE ANTAGONISTE CXCR3<br />

(73) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033-0530, US<br />

Pharmacopeia, LLC, 10275 Science Center<br />

Drive, San Diego, CA 92121, US<br />

(72) ANILKUMAR, Gopinadhan, N., Edison, New<br />

Jersey 08820, US<br />

ZENG, Qingbei, Edison, New Jersey 08820,<br />

US<br />

ROSENBLUM, Stuart, B., West Orange, New<br />

Jersey 07052, US<br />

KOZLOWSKI, Joseph, A., Princeton, New<br />

Jersey 08540, US<br />

MCGUINNESS, Brian, F., Plainsboro, New<br />

Jersey 08536, US<br />

HOBBS, Douglas, W., Chesterfield, MO<br />

63005-4541, US<br />

(74) Horgan, James Michael Frederic, et al, Merck<br />

Sharp & Dohme Ltd. <strong>European</strong> <strong>Patent</strong><br />

Department Hertford Road, Hoddesdon<br />

Hertfordshire EN11 9BU, GB<br />

C07D 401/14 → (51) C07D 235/26<br />

C07D 401/14 → (51) C07D 401/12<br />

778<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

C07D 403/06 → (51) C07D 2<strong>31</strong>/56<br />

C07D 403/06 → (51) C07D 235/26<br />

C07D 403/06 → (51) C07D 295/125<br />

C07D 403/12 → (51) C07D 401/12<br />

C07D 403/14 → (51) C07D 235/26<br />

C07D 405/12 → (51) C07D 221/16<br />

C07D 405/12 → (51) C07D 235/26<br />

C07D 405/14 → (51) C07D 235/26<br />

C07D 405/14 → (51) C07D 401/12<br />

C07D 407/14 → (51) C07D 295/125<br />

C07D 409/06 → (51) C07D 235/26<br />

C07D 409/12 → (51) C07D 221/16<br />

C07D 409/12 → (51) C07D 235/18<br />

C07D 409/12 → (51) C07D 235/26<br />

(51) C07D 409/14 (11) 1 720 866 B1<br />

(25) De (26) De<br />

(21) 04804455.6 (22) <strong>31</strong>.12.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

HR LV<br />

(43) 15.11.2006<br />

(86) EP 2004/014870 <strong>31</strong>.12.2004<br />

(87) WO 2005/068456 2005/30 28.07.2005<br />

(30) 15.01.2004 DE 102004002044<br />

(54) • HERSTELLVERFAHREN<br />

• PRODUCTION METHOD<br />

• PROCEDE DE PREPARATION<br />

(73) Bayer Schering Pharma Aktiengesellschaft,<br />

Müllerstrasse 178, 13353 Berlin, DE<br />

(72) BERWE, Mathias, 45549 Sprockhövel, DE<br />

THOMAS, Christian, 42111 Wuppertal, DE<br />

REHSE, Joachim, 42799 Leichlingen, DE<br />

GROTJOHANN, Dirk, 51377 Leverkusen, DE<br />

C07D 409/14 → (51) C07D 235/26<br />

C07D 413/04 → (51) C07D 263/48<br />

C07D 413/06 → (51) C07D 235/26<br />

C07D 413/12 → (51) C07D 221/16<br />

C07D 413/12 → (51) C07D 239/557<br />

C07D 413/12 → (51) C07D 263/48<br />

C07D 413/12 → (51) C07J 1/00<br />

C07D 413/14 → (51) C07D 221/16<br />

C07D 413/14 → (51) C07D 401/14<br />

(51) C07D 417/04 (11) 2 155 738 B1<br />

(25) En (26) En<br />

(21) 08759910.6 (22) 22.05.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 24.02.2010<br />

(86) EP 2008/056309 22.05.2008<br />

(87) WO 2008/145596 2008/49 04.12.2008<br />

(30) 01.06.2007 EP 07109458<br />

(54) • PIPERIDIN-AMIDDERIVATE

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