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Bulletin 2011/31 - European Patent Office

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(C07D) II.1(1)<br />

C07D 409/06 C07D 409/12<br />

C07D 409/14 C07D 413/06<br />

C07D 417/06 C07D 417/14<br />

A61K <strong>31</strong>/4184 A61P 11/06<br />

(25) En (26) En<br />

(21) 08755478.8 (22) 15.05.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 17.02.2010<br />

(86) US 2008/063630 15.05.2008<br />

(87) WO 2008/147697 2008/49 04.12.2008<br />

(30) 22.05.2007 US 939452 P<br />

(54) • BENZIMIDAZOLONCHYMASEHEMMER<br />

• BENZIMIDAZOLONE CHYMASE INHIBI-<br />

TORS<br />

• INHIBITEURS DE BENZIMIDAZOLONE<br />

CHYMASE<br />

(73) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim, DE<br />

(84) AT BE BG CH CY CZ DK EE ES FI FR GB GR<br />

HR HU IE IS IT LI LT LU LV MC MT NL NO<br />

PL PT RO SE SI SK TR<br />

(73) Boehringer Ingelheim Pharma GmbH & Co.<br />

KG, Binger Strasse 173, 55216 Ingelheim,<br />

DE<br />

(84) DE<br />

(72) ABEYWARDANE, Asitha, Ridgefield, CT<br />

06877-0368, US<br />

COOK, Brian, Nicholas, Ridgefield, CT<br />

08677-0368, US<br />

DE LOMBAERT, Stephane, Ridgefield, CT<br />

06877-0368, US<br />

EMMANUEL, Michel, Jose, Ridgefield, CT<br />

06877-0368, US<br />

GUO, Xin, Ridgefield, CT 06877-0368, US<br />

KIM, Jin, Mi, Ridgefield, CT 06877-0368, US<br />

HAO, Ming-Hong, Ridgefield, CT 06877-<br />

0368, US<br />

LO, Ho, Yin, Ridgefield, CT 08677-0368, US<br />

MAN, Chuk, Chui, Ridgefield, CT 06877-<br />

0368, US<br />

MORWICK, Tina, Ridgefield, CT 06877-0368,<br />

US<br />

NEMOTO, Peter, Allen, Ridgefield, CT 06877-<br />

0368, US<br />

QIAN, Kevin, Chungeng, Ridgefield, CT<br />

06877-0368, US<br />

TAKAHASHI, Hidenori, Ridgefield, CT 06877-<br />

0368, US<br />

TAYLOR, Steven, John, Ridgefield, CT<br />

06877-0368, US<br />

(74) Hammann, Heinz, et al, Boehringer Ingelheim<br />

GmbH CD-<strong>Patent</strong>s Binger Straße 173, 55216<br />

Ingelheim am Rhein, DE<br />

(51) C07D 235/30 (11) 1 633 722 B1<br />

A61K <strong>31</strong>/4168<br />

(25) En (26) En<br />

(21) 04751430.2 (22) 06.05.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

(43) 15.03.2006<br />

(86) US 2004/014036 06.05.2004<br />

(87) WO 2004/100881 2004/48 25.11.2004<br />

(30) 09.05.2003 US 469619 P<br />

(54) • HERSTELLUNG UND VERWENDUNG VON<br />

ARYLALKYLSÄUREDERIVATEN ZUR<br />

BEHANDLUNG VON OBESITAS<br />

• PREPARATION AND USE OF ARYL ALKYL<br />

ACID DERIVATIVES FOR THE TREATMENT<br />

OF OBESITY<br />

• PREPARATION ET UTILISATION DE DERI-<br />

VES D'ARYL ALKYL ACIDE POUR LE<br />

TRAITEMENT DE L'OBESITE<br />

(73) Bayer HealthCare LLC, 555 White Plains<br />

Road, Tarrytown, NY 10591, US<br />

(72) SMITH, Roger, Madison, CT 06443, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

CAMPBELL, Ann-Marie, Monroe, CT 06468,<br />

US<br />

COISH, Philip, North Haven, CT 06473, US<br />

DAI, Miao, Briarwood, NY 11435, US<br />

JENKINS, Susan, Milford, CT 06460, US<br />

LOWE, Derek, Hamden, CT 06518, US<br />

O'CONNOR, Stephen, Guilford, CT 06437,<br />

US<br />

SU, Ning, Hamden, CT 06518, US<br />

WANG, Gan, Wallingord, CT 06492, US<br />

ZHANG, Mingbao, Stamford, CT 06905, US<br />

ZHU, Lei, Milford, CT 06460, US<br />

(74) Burkert, Frank, et al, Bayer HealthCare AG<br />

Law and <strong>Patent</strong>s, 51368 Leverkusen, DE<br />

C07D 239/32 → (51) C07D 473/16<br />

(51) C07D 239/48 (11) 2 070 914 B1<br />

A61P 19/00 A61K <strong>31</strong>/505<br />

(25) Fr (26) Fr<br />

(21) 0900<strong>31</strong>74.1 (22) 12.11.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 17.06.2009<br />

(30) 19.11.2002 FR 0214429<br />

(54) • Neue antagonistische Derivate des Vitronektinrezeptors,<br />

ihr Herstellungsverfahren,<br />

ihre Anwendung als Arzneimittel und die<br />

pharmazeutischen Zusammensetzungen,<br />

die sie enthalten<br />

• New antagonist derivatives of the vitronectin<br />

receptor, method for their preparation,<br />

their application as medicine and<br />

pharmaceutical compositions containing<br />

them<br />

• Nouveaux dérivés antagonistes du récepteur<br />

de la vitronectine, leur procédé de<br />

préparation, leur application comme médicaments<br />

et les compositions pharmaceutiques<br />

les renfermant<br />

(73) Galapagos SAS, 102, Avenue Gaston Roussel,<br />

93230 Romainville, FR<br />

(72) Ruxer, Jean -Marie, 92130 Issy les Moulineaux,<br />

FR<br />

Lefrancois, Jean-Michel, 93340 Le Raincy,<br />

FR<br />

Heckmann, Bertrand, 91440 Bures sur<br />

Yvette, FR<br />

(74) Lord, Hilton David, Marks & Clerk LLP 90<br />

Long Acre, London WC2E 9RA, GB<br />

(62) 03799611.3 / 1 565 467<br />

(51) C07D 239/48 (11) 2 132 185 B1<br />

A61K <strong>31</strong>/506 A61P 25/00<br />

(25) En (26) En<br />

(21) 08737283.5 (22) 10.04.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(43) 16.12.2009<br />

(86) HU 2008/000032 10.04.2008<br />

(87) WO 2008/125891 2008/43 23.10.2008<br />

(30) 11.04.2007 HU 0700269<br />

(54) • PYRIMIDINYL-PIPERAZINE ALS DOPAMIN<br />

D3/D2-REZEPTORLIGANDEN<br />

• PYRIMIDINYL-PIPERAZINES USEFUL AS<br />

DOPAMINE D3/D2 RECEPTOR LIGANDS<br />

• PYRIMIDINYL-PIPÉRAZINES UTILES EN<br />

TANT QUE LIGANDS DES RÉCEPTEURS<br />

D3/D2 DE LA DOPAMINE<br />

(73) Richter Gedeon Nyrt., Gyömröi út 19-21,<br />

1103 Budapest, HU<br />

(72) BARTÁNÉ SZALAI, Gizella, H-1162 Budapest,<br />

HU<br />

ÁGAINÉ CSONGOR, Éva, H-10<strong>31</strong> Budapest,<br />

HU<br />

DOMÁNY, György, H-7695 Óbánya, HU<br />

776<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

GYERTYÁN, István, H-1161 Budapest, HU<br />

KISS, Béla, H-1182 Budapest, HU<br />

LASZY, Judit, H-2094 Nagykovácsi, HU<br />

SÁGHY, Katalin, H-1082 Budapest, HU<br />

SCHMIDT, Éva, H-2089 Telki, HU<br />

FARKAS, Sándor, H-1103 Budapest, HU<br />

KOMLÓDI, Zsolt, H-1203 Budapest, HU<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München, DE<br />

C07D 239/48 → (51) C07D 473/16<br />

C07D 239/52 → (51) C07D 473/16<br />

(51) C07D 239/557 (11) 1 819 683 B1<br />

C07D 413/12 A61K <strong>31</strong>/513<br />

A61P <strong>31</strong>/18<br />

(25) En (26) En<br />

(21) 05852866.2 (22) 02.12.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 22.08.2007<br />

(86) US 2005/043781 02.12.2005<br />

(87) WO 2006/060730 2006/23 08.06.2006<br />

(30) 03.12.2004 US 63<strong>31</strong>32 P<br />

(54) • KALIUMSALZ EINES HIV-INTEGRASE-<br />

INHIBITORS<br />

• POTASSIUM SALT OF AN HIV INTEGRASE<br />

INHIBITOR<br />

• SELS DE POTASSIUM D'UN INHIBITEUR<br />

D'INTEGRASE HIV<br />

(73) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

ISTITUTO DI RICERCHE DI BIOLOGIA<br />

MOLECOLARE P. ANGELETTI S.P.A., Via<br />

Pontina Km. 30.600, 00040 Pomezia, IT<br />

MERCK SHARP & DOHME LTD., Hertford<br />

Road, Hoddesdon, Hertfordshire EN11 9BU,<br />

GB<br />

(72) PYE, Philip, Rahway, New Jersey 07065-<br />

0907, US<br />

ANGELAUD, Remy, Rahway, New Jersey<br />

07065-0907, US<br />

MANCHENO, Danny, Rahway, New Jersey<br />

07065-0907, US<br />

(74) Man, Jocelyn, et al, Merck & Co., Inc.<br />

<strong>European</strong> <strong>Patent</strong> Department Hertford Road<br />

Hoddesdon, Hertfordshire EN11 9BU, GB<br />

C07D 241/04 → (51) A61K <strong>31</strong>/495<br />

C07D 249/08 → (51) C07C <strong>31</strong>1/51<br />

(51) C07D 261/20 (11) 1 425 272 B1<br />

A61K <strong>31</strong>/42 A61P 25/18<br />

(25) En (26) En<br />

(21) 02767454.8 (22) 30.08.2002<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SK TR<br />

(43) 09.06.2004<br />

(86) EP 2002/009700 30.08.2002<br />

(87) WO 2003/020707 2003/11 13.03.2003<br />

(30) <strong>31</strong>.08.2001 US <strong>31</strong>6390 P<br />

(54) • OPTISCHE ISOMERE EINES ILOPERIDON-<br />

METABOLITEN<br />

• OPTICAL ISOMERS OF AN ILOPERIDONE<br />

METABOLITE<br />

• ISOMERES OPTIQUES D'UN METABOLITE<br />

D'ILOPERIDONE<br />

(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(84) BE BG CH CY CZ DE DK EE ES FI FR GB GR<br />

IE IT LI LU MC NL PT SE SK TR<br />

(73) Novartis Pharma GmbH, Brunner Strasse 59,<br />

1230 Wien, AT<br />

(84) AT

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