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Bulletin 2011/31 - European Patent Office

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(C07D) I.1(1)<br />

(51) C07D 487/14 (11) 2 350 087 A1*<br />

A61K <strong>31</strong>/4162 A61P 35/00<br />

(25) En (26) En<br />

(21) 097639<strong>31</strong>.4 (22) 26.11.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2009/065930 26.11.2009<br />

(87) WO 2010/060968 2010/22 03.06.2010<br />

(30) 27.11.2008 EP 08305856<br />

(54) • REGIOSELEKTIVE REDUKTION KONDEN-<br />

SIERTER PYRROLOCARBAZOL-5,7-DIO-<br />

NEN<br />

• REGIOSELECTIVE REDUCTION OF FUSED<br />

PYRROLOCARBAZOLES-5,7-DIONES<br />

• RÉDUCTION RÉGIOSÉLECTIVE DE PYR-<br />

ROLOCARBAZOLE-5,7-DIONES CONDEN-<br />

SÉES<br />

(71) Cephalon France, 20 Rue Charles Martigny,<br />

94704 Maisons-Alfort Cedex, FR<br />

(72) PRAT-LACONDEMINE, Laurence, F-77340<br />

Pontault Combault, FR<br />

(74) Balmefrezol, Ludovic Francis Pierre, et al,<br />

Cabinet Lavoix 62, rue de Bonnel, FR-69448<br />

Lyon Cedex 03, FR<br />

C07D 487/14 → (51) C07D 487/12<br />

(51) C07D 491/048 (11) 2 350 088 A1*<br />

A61K <strong>31</strong>/40 A61P 25/00<br />

A61P 25/06 A61P 25/16<br />

A61P 25/18 A61P 25/22<br />

A61P 25/24 A61P 25/28<br />

(25) En (26) En<br />

(21) 09781255.6 (22) 29.07.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2009/059829 29.07.2009<br />

(87) WO 2010/012789 2010/05 04.02.2010<br />

(30) 30.07.2008 EP 08161485<br />

(54) • 1,6-DIHYDRO-2H-3-OXA-6-AZA-AS-INDA-<br />

CENVERBINDUNGEN<br />

• 1,6-DIHYDRO-2H-3-OXA-6-AZA-AS-INDA-<br />

CENE COMPOUNDS<br />

• COMPOSÉS DE LA 1,6-DIHYDRO-2H-3-<br />

OXA-6-AZA-AS-INDACENE<br />

(71) Ferrer Internacional, S.A., Gran Via Carles III<br />

94, 08028 Barcelona, ES<br />

(72) FALCÓ, José L., E-08004 Barcelona, ES<br />

PALOMER, Albert, E-08014 Barcelona, ES<br />

GUGLIETTA, Antonio, E-08750 Molins de<br />

Rei, ES<br />

(74) Reitstötter - Kinzebach, <strong>Patent</strong>anwälte<br />

Sternwartstrasse 4, 81679 München, DE<br />

(51) C07D 491/048 (11) 2 350 089 A1*<br />

A61K <strong>31</strong>/496 A61P 19/00<br />

(25) En (26) En<br />

(21) 09783392.5 (22) 24.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) EP 2009/062407 24.09.2009<br />

(87) WO 2010/034789 2010/13 01.04.2010<br />

(30) 24.09.2008 GB 0817425<br />

(54) • PROTEASE-INHIBITOREN<br />

• PROTEASE INHIBITORS<br />

• INHIBITEURS DE PROTÉASES<br />

(71) Medivir AB, P.O. Box 1086, 141 22 Huddinge,<br />

SE<br />

(72) IVANOV, Vladimir, S-141 22 Huddinge, SE<br />

SAMUELSSON, Bertil, S-141 22 Huddinge,<br />

SE<br />

JOHANSSON, Per-Ola, S-141 22 Huddinge,<br />

SE<br />

KAHNBERG, Pia, S-141 22 Huddinge, SE<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

WÄHLING, Horst, S-141 22 Huddinge, SE<br />

(74) Goodall, Scott, Sagittarius IP Taylor House<br />

39 High Street, Marlow Buckinghamshire<br />

SL7 1AF, GB<br />

C07D 491/10 → (51) C07D 235/02<br />

C07D 491/10 → (51) C07D 491/20<br />

C07D 491/107→ (51) C07D 417/04<br />

C07D 491/107→ (51) C07D 491/20<br />

C07D 491/113→ (51) C07D 471/04<br />

(51) C07D 491/20 (11) 2 350 090 A2*<br />

C07D 495/20 C07D 498/20<br />

C07D 491/10 C07D 513/20<br />

A61K <strong>31</strong>/407 A61P 25/00<br />

(25) En (26) En<br />

(21) 09740589.8 (22) 13.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/060537 13.10.2009<br />

(87) WO 2010/045251 2010/16 22.04.2010<br />

(88) 18.11.2010<br />

(30) 17.10.2008 US 106464 P<br />

(54) • SPIRO-OXINDOLVERBINDUNGEN UND<br />

IHRE VERWENDUNG ALS THERAPEUTI-<br />

SCHE MITTEL<br />

• SPIRO-OXINDOLE COMPOUNDS AND<br />

THEIR USE AS THERAPEUTIC AGENTS<br />

• COMPOSÉS SPIRO-OXINDOLE ET LEUR<br />

UTILISATION COMME AGENTS THÉRA-<br />

PEUTIQUES<br />

(71) Xenon Pharmaceuticals Inc., 3650 Gilmore<br />

Way, Burnaby, BC V5G 4W8, CA<br />

(72) CHAFEEV, Mikhail, Burnaby British Columbia<br />

V5H 4V9, CA<br />

CHOWDHURY, Sultan, Surrey British<br />

Columbia V3S 7S3, CA<br />

FRASER, Lauren, Surrey British Columbia<br />

V4N 0Z2, CA<br />

FU, Jianmin, Coquitlam British Columbia V3E<br />

3B6, CA<br />

LANGILLE, Jonathan, Quaker Hill Connecticut<br />

06375-1205, US<br />

LIU, Shifeng, Coquitlam British Columbia<br />

V3E 3E1, CA<br />

SUN, Jianyu, California 94403, US<br />

SUN, Shaoyi, Coquitlam British Columbia<br />

V3K 1G3, CA<br />

SVIRIDOV, Serguei, Burnaby British Columbia<br />

V5H 4N8, CA<br />

WOOD, Mark, Port Moody British Columbia<br />

V3H 5K4, CA<br />

ZENOVA, Alla, Vancouver British Columbia<br />

V6J 2B1, CA<br />

JIA, Qi, Burnaby British Columbia V5J 5M6,<br />

CA<br />

CADIEUX, Jean-Jacques, Burnaby British<br />

Columbia V5B 1P6, CA<br />

GAUTHIER, Simon, J., Vancouver British<br />

Columbia V6Z 2Y7, CA<br />

DOUGLAS, Amy Frances, Vancouver British<br />

Columbia V6R 2H6, CA<br />

HSIEH, Tom, Toronto Ontario M5S 2E8, CA<br />

CHAKKA, Nagasree, Waltham Massachusetts<br />

02452, US<br />

CIKOJEVIC, Zoran, Port Coquitlam British<br />

Columbia V3B 7J8, CA<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

(51) C07D 491/20 (11) 2 350 091 A1*<br />

C07D 491/107 A61K <strong>31</strong>/407<br />

A61P 25/00 A61P 29/00<br />

189<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

(25) En (26) En<br />

(21) 09741118.5 (22) 13.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/060455 13.10.2009<br />

(87) WO 2010/045197 2010/16 22.04.2010<br />

(30) 17.10.2008 US 106410 P<br />

(54) • SPIRO-OXINDOLVERBINDUNGEN UND<br />

IHRE VERWENDUNG ALS THERAPEUTI-<br />

SCHE MITTEL<br />

• SPIRO-OXINDOLE COMPOUNDS AND<br />

THEIR USE AS THERAPEUTIC AGENTS<br />

• COMPOSÉS SPIRO-OXINDOLE ET LEUR<br />

UTILISATION COMME AGENTS THÉRA-<br />

PEUTIQUES<br />

(71) Xenon Pharmaceuticals Inc., 3650 Gilmore<br />

Way, Burnaby, BC V5G 4W8, CA<br />

(72) CHAFEEV, Mikhail, Burnaby, British Columbia<br />

V5H 4V9, CA<br />

CHOWDHURY, Sultan, Surrey, British<br />

Columbia V3S 7S3, CA<br />

FRASER, Lauren, Surrey, British Columbia<br />

V4N 0Z2, CA<br />

FU, Jianmin, Coquitlam, British Columbia<br />

V3E 3B6, CA<br />

LANGILLE, Jonathan, Quaker Hill, Connecticut<br />

06375-1205, US<br />

LIU, Shifeng, Coquitlam, British Columbia<br />

V3E 3E1, CA<br />

SUN, Jianyu, San Mateo, California 94403,<br />

US<br />

SUN, Shaoyi, Coquitlam, British Columbia<br />

V3K 1G3, CA<br />

SVIRIDOV, Serguei, Burnaby, British<br />

Columbia V5H 4N8, CA<br />

WOOD, Mark, Port Moody, British Columbia<br />

V3H 5K4, CA<br />

ZENOVA, Alla, Vancouver, British Columbia<br />

V6J 2B1, CA<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

C07D 493/04 → (51) C07D 307/12<br />

C07D 493/10 → (51) C07D 307/12<br />

(51) C07D 495/04 (11) 2 350 092 A1*<br />

A61K <strong>31</strong>/519 A61P 25/30<br />

(25) En (26) En<br />

(21) 09736343.6 (22) 29.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) US 2009/058705 29.09.2009<br />

(87) WO 2010/045006 2010/16 22.04.2010<br />

(30) 13.10.2008 US 104781 P<br />

05.06.2009 US 479158<br />

(54) • METHYLENAMINE VON THIENO[2,3-D]<br />

PYRIMIDIN UND DEREN VERWENDUNG<br />

ALS ANTAGONISTEN DES ADENOSIN-<br />

A2A-REZEPTORS<br />

• METHYLENE AMINES OF THIENO Ý2,3-<br />

D¨PYRIMIDINE AND THEIR USE AS ADE-<br />

NOSINE A2A RECEPTOR ANTAGONISTS<br />

• AMINES MÉTHYLÉNIQUES DE THIÉNO<br />

Ý2,3-D¨PYRIMIDINE ET LEUR UTILISA-<br />

TION COMME ANTAGONISTES DES<br />

RÉCEPTEURS DE L ADÉNOSINE A2A<br />

(71) Janssen Pharmaceutica, N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) BARBAY, J., Kent, Flourtown, PA 190<strong>31</strong>, US<br />

CHAKRAVARTY, Devraj, Hillsborough, NJ<br />

08844, US<br />

SHOOK, Brian, Christopher, Gilbertsville, PA<br />

19525, US<br />

WANG, Aihua, Jamison, PA 18929, US

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