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Bulletin 2011/31 - European Patent Office

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(C07D) I.1(1)<br />

(25) En (26) En<br />

(21) 08875995.6 (22) 12.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) IN 2008/000767 12.11.2008<br />

(87) WO 2010/055526 2010/20 20.05.2010<br />

(54) • NEUES POLYMORPH VON EMTRICITABIN<br />

UND VERFAHREN ZU DESSEN HERSTEL-<br />

LUNG<br />

• A NOVEL POLYMORPH OF EMTRICITA-<br />

BINE AND A PROCESS FOR PREPARING<br />

OF THE SAME<br />

• NOUVEAU POLYMORPHE DE L'EMTRICI-<br />

TABINE ET PROCÉDÉ POUR SA PRÉPA-<br />

RATION<br />

(71) Lupin Ltd., 159, CST Road Kalina, Santacruz<br />

(East), Mumbai, Maharashtra 400 098, IN<br />

(72) SINGH, Girij, Pal, Pune 411 042 Maharashtra,<br />

IN<br />

SRIVASTAVA, Dhananjai, Pune 411 042<br />

Maharashtra, IN<br />

JADHAV, Harishchandra, Pune 411 042<br />

Maharashtra, IN<br />

PATHAK, Shailendra, Pune 411 042 Maharashtra,<br />

IN<br />

SAINI, Manmeet, Pune 411 042 Maharashtra,<br />

IN<br />

PATIL, Sudhakar, Pune 411 042 Maharashtra,<br />

IN<br />

(74) Srinivasan, Ravi Chandran, et al, J.A. Kemp<br />

& Co. 14 South Square Gray's Inn, London<br />

WC1R 5JJ, GB<br />

(51) C07D 413/00 (11) 2 350 066 A1*<br />

C07D 413/02<br />

(25) En (26) En<br />

(21) 09822445.4 (22) 15.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/060736 15.10.2009<br />

(87) WO 2010/048010 2010/17 29.04.2010<br />

(30) 21.10.2008 US 196849 P<br />

(54) • 2,5-DISUBSTIUIERTE PIPERIDINE ALS<br />

ANTAGONISTEN DES OREXINREZEPTORS<br />

• 2,5-DISUBSTITUTED PIPERIDINE OREXIN<br />

RECEPTOR ANTAGONISTS<br />

• PIPÉRIDINES 2,5-DISUBSTITUÉES<br />

COMME ANTAGONISTES DU RÉCEPTEUR<br />

DE L OREXINE<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907,<br />

US<br />

(72) BRESLIN, Michael, J., Rahway New Jersey<br />

07065-0907, US<br />

COLEMAN, Paul, J., Rahway New Jersey<br />

07065-0907, US<br />

COX, Christopher, D., Rahway New Jersey<br />

07065-0907, US<br />

SCHREIER, John, D., Rahway New Jersey<br />

07065-0907, US<br />

WHITMAN, David, B., Rahway New Jersey<br />

07065-0907, US<br />

(74) Buchan, Gavin MacNicol, et al, Merck & Co.,<br />

Inc. <strong>European</strong> <strong>Patent</strong> Department Hertford<br />

Road, Hoddesdon, Hertfordshire EN11 9BU,<br />

GB<br />

C07D 413/02 → (51) C07D 307/91<br />

C07D 413/02 → (51) C07D 413/00<br />

C07D 413/04 → (51) A61K <strong>31</strong>/4188<br />

C07D 413/04 → (51) C07D 409/04<br />

C07D 413/04 → (51) C07D 513/04<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

C07D 413/06 → (51) A61K <strong>31</strong>/4025<br />

C07D 413/06 → (51) C07D 211/76<br />

C07D 413/06 → (51) C07D 217/26<br />

C07D 413/12 → (51) A61P 3/10<br />

C07D 413/12 → (51) C07C 39/42<br />

C07D 413/12 → (51) C07D 207/08<br />

C07D 413/12 → (51) C07D 211/76<br />

C07D 413/12 → (51) C07D 211/96<br />

C07D 413/12 → (51) C07D 239/34<br />

C07D 413/12 → (51) C07D 239/91<br />

C07D 413/12 → (51) C07D 263/56<br />

C07D 413/12 → (51) C07D 401/12<br />

C07D 413/14 → (51) A61K <strong>31</strong>/4025<br />

C07D 413/14 → (51) A61K <strong>31</strong>/4188<br />

C07D 413/14 → (51) C07D 211/76<br />

C07D 413/14 → (51) C07D 401/12<br />

C07D 413/14 → (51) C07D 401/14<br />

C07D 413/14 → (51) C07D 407/06<br />

C07D 413/14 → (51) C07D 409/04<br />

C07D 417/00 → (51) C07D 213/40<br />

C07D 417/02 → (51) C07D 307/91<br />

(51) C07D 417/04 (11) 2 350 067 A2*<br />

C07D 417/14 C07D 471/10<br />

C07D 487/04 C07D 487/08<br />

C07D 285/135 C07D 271/113<br />

C07D 491/107 A61K <strong>31</strong>/4355<br />

A61K <strong>31</strong>/437 A61K <strong>31</strong>/4439<br />

A61K <strong>31</strong>/444 A61P 3/10<br />

(25) En (26) En<br />

(21) 09740590.6 (22) 14.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2009/060610 14.10.2009<br />

(87) WO 2010/045303 2010/16 22.04.2010<br />

(88) 05.08.2010<br />

(30) 16.10.2008 US 105965 P<br />

(54) • PYRROLIDIN-, PIPERIDIN- UND PIPERA-<br />

ZINDERIVATE UND VERFAHREN ZU<br />

DEREN ANWENDUNG<br />

• PYRROLIDINE, PIPERIDINE AND PIPERA-<br />

ZINE DERIVATIVES AND METHODS OF<br />

USE THEREOF<br />

• DÉRIVÉS DE PYRROLIDINE, DE PIPÉRI-<br />

DINE ET DE PIPÉRAZINE ET LEURS<br />

MÉTHODES D'UTILISATION<br />

(71) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033-0530, US<br />

(72) PALANI, Anandan, Bridgewater New Jersey<br />

08807, US<br />

BERLIN, Michael, Y., Flemington New Jersey<br />

08822, US<br />

ASLANIAN, Robert, G., Rockaway New<br />

Jersey 07866, US<br />

VACCARO, Henry, M., South Plainfield New<br />

Jersey 07080, US<br />

185<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

CHAN, Tin-Yau, Edison New Jersey 08817,<br />

US<br />

XIAO, Dong, Warren New Jersey 07059, US<br />

DEGRADO, Sylvia, Scotch Plains New Jersey<br />

07076, US<br />

RAO, Ashwin, U., Avenel New Jersey 07001,<br />

US<br />

CHEN, Xiao, Edison New Jersey 08820, US<br />

LEE, Yoon, Joo, Scotch Plains New Jersey<br />

07076, US<br />

SOFOLARIDES, Michael, J., Hoboken New<br />

Jersey 07030, US<br />

SHAO, Ning, Clark New Jersey 07066, US<br />

HUANG, Ying, R., Berkeley Heights New<br />

Jersey 07922, US<br />

LIU, Zhidan, Edison New Jersey 08820, US<br />

WANG, Li Yuan, Warren New Jersey 07059,<br />

US<br />

PU, Haiyan, Livingston New Jersey 07039,<br />

US<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

C07D 417/04 → (51) C07D 207/08<br />

C07D 417/04 → (51) C07D 211/96<br />

C07D 417/04 → (51) C07D 213/40<br />

C07D 417/04 → (51) C07D 409/04<br />

C07D 417/04 → (51) C07D 513/04<br />

C07D 417/06 → (51) C07D 217/26<br />

C07D 417/10 → (51) C07D 213/40<br />

C07D 417/10 → (51) C07D 213/64<br />

C07D 417/12 → (51) C07D 211/76<br />

C07D 417/12 → (51) C07D 211/96<br />

C07D 417/14 → (51) A61K <strong>31</strong>/4025<br />

C07D 417/14 → (51) C07D 207/08<br />

C07D 417/14 → (51) C07D 211/96<br />

C07D 417/14 → (51) C07D 213/40<br />

C07D 417/14 → (51) C07D 213/81<br />

C07D 417/14 → (51) C07D 401/14<br />

C07D 417/14 → (51) C07D 403/04<br />

C07D 417/14 → (51) C07D 403/14<br />

C07D 417/14 → (51) C07D 409/04<br />

C07D 417/14 → (51) C07D 417/04<br />

(51) C07D 451/02 (11) 2 350 068 A2*<br />

C07D 519/00 A61K <strong>31</strong>/46<br />

A61P 3/00<br />

(25) En (26) En<br />

(21) 09740684.7 (22) 22.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2009/063913 22.10.2009<br />

(87) WO 2010/046445 2010/17 29.04.2010<br />

(88) 01.07.2010<br />

(30) 23.10.2008 EP 08167440

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