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Bulletin 2011/31 - European Patent Office

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(C07D) I.1(2)<br />

(30) 22.09.2008 CN 200810070345<br />

(54) • NEUE KRISTALLINE FORMEN VON<br />

PEMETREXEDDISÄURE UND DEREN HER-<br />

STELLUNG<br />

• NEW CRYSTALLINE FORMS OF PEME-<br />

TREXED DIACID, AND PREPARATIONS<br />

THEREOF<br />

• TROIS NOUVELLES FORMES DE CRIS-<br />

TAUX DE DIACIDE DE PEMETREXED ET<br />

LEUR PROCÉDÉ DE PRÉPARATION<br />

(71) Chongqing Pharmaceutical Research Institute<br />

Co., Ltd., No. 565, Tushan Road Nan'an<br />

District, Chongqing 400061, CN<br />

(72) LUO, Jie, Chongqing 400061, CN<br />

LIN, Meng, Chongqing 400061, CN<br />

ZHU, Zhengyong, Chongqing 400061, CN<br />

LUO, Junlai, Chongqing 400061, CN<br />

YE, Wenrun, Chongqing 400061, CN<br />

QIN, Yongmei, Chongqing 400061, CN<br />

DENG, Jie, Chongqing 400061, CN<br />

(74) Epping - Hermann - Fischer, <strong>Patent</strong>anwaltsgesellschaft<br />

mbH Ridlerstrasse 55, 80339<br />

München, DE<br />

(51) C07D 487/04 (11) 2 351 756 A1<br />

A61K <strong>31</strong>/519 A61P 25/28<br />

A61P 25/18 A61P 25/26<br />

A61P 25/16 A61P 25/08<br />

A61P 9/10 A61P 3/04<br />

A61P 3/08 A61K 9/48<br />

A61K 9/08<br />

(25) Ru (26) En<br />

(21) 09819452.5 (22) 06.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) RU 2009/000518 06.10.2009<br />

(87) WO 2010/041983 2010/15 15.04.2010<br />

(30) 06.10.2008 RU 2008139495<br />

06.10.2008 RU 2008139496<br />

14.10.2008 RU 2008140599<br />

14.10.2008 RU 2008140601<br />

(54) • SUBSTITUIERTE 3-ARYLSULFONYL-<br />

PYRAZOLO[1,5-A]PYRIMIDINE, SEROTO-<br />

NIN-5-HT6-REZEPTORANTAGONISTEN<br />

SOWIE VERFAHREN ZU IHRER HERSTEL-<br />

LUNG UND VERWENDUNG<br />

• SUBSTITUTED 3-ARYLSULFONYL-PYRA-<br />

ZOLO[1,5-A]PYRIMIDINES, SEROTONIN<br />

5-HT6 RECEPTOR ANTAGONISTS AND<br />

METHODS FOR THE PRODUCTION AND<br />

USE THEREOF<br />

• 3-ARYLSULFONYL-PYRAZOLO[1,5-A]<br />

PYRIMIDINES SUBSTITUÉES, ANTAGO-<br />

NISTES DES RÉCEPTEURS 5-HT6 DE<br />

SÉROTONINE, PROCÉDÉS DE FABRICA-<br />

TION ET D'UTILISATION<br />

(71) Ivashchenko, Andrey Alexandrovich, Ul.<br />

Abramtsevskaya, 4-2-27, Moscow, 127576,<br />

RU<br />

Alla Chem, LLC., <strong>31</strong>8 N. Carson Street, Suite<br />

208, Carson City, NV 89701, US<br />

(72) IVASHCHENKO, Alexander Vasilievich, Encinitas<br />

CA 92024, US<br />

SAVCHUK Nikolay Filippovich, Rancho Santa<br />

Fe CA 92067, US<br />

LAVROVSKY Yan, San Diego 136 CA 92121,<br />

US<br />

MITKIN, Oleg Dmitrievich, Moskovskaya obl.<br />

141400, RU<br />

KADIEVA Madina Georgievna, Moscow<br />

region 141851, RU<br />

(74) Henrion, Oliver, et al, <strong>Patent</strong>anwälte Zellentin<br />

& Partner Rubensstrasse 30, 67061 Ludwigshafen,<br />

DE<br />

C07D 487/04 → (51) C07D 401/14<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(51) C07D 498/18 (11) 2 351 757 A1<br />

A61K <strong>31</strong>/436 A61P 35/00<br />

A61P 37/02<br />

(25) Zh (26) En<br />

(21) 09813972.8 (22) 17.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) CN 2009/001042 17.09.2009<br />

(87) WO 2010/0<strong>31</strong>251 2010/12 25.03.2010<br />

(30) 18.09.2008 CN 200810200073<br />

(54) • RAPAMYCIN-KOHLENSÄUREESTER-ANA-<br />

LOGA, PHARMAZEUTISCHE ZUSAMMEN-<br />

SETZUNGEN, ZUBEREITUNGEN UND IHRE<br />

VERWENDUNG<br />

• RAPAMYCIN CARBONIC ESTER ANALO-<br />

GUES, PHARMACEUTICAL COMPOSI-<br />

TIONS, PREPARATIONS AND USES<br />

THEREOF<br />

• PRODUIT SIMILAIRE À L ESTER DE<br />

CARBONATE DE SIROLIMUS, SON SEL ET<br />

SON COMPOSÉ MÉDICINAL PHARMA-<br />

CEUTIQUEMENT ACCEPTABLES, SON<br />

PROCÉDÉ DE PRÉPARATION ET SON<br />

UTILISATION<br />

(71) Shanghai Institute Materia Medica, Chinese<br />

Academy Of Sciences, 555 Zu Chong Zhi<br />

Road Zhang Jiang, Pudong, Shanghai<br />

201203, CN<br />

(72) NAN, Fajun, Shanghai 201203, CN<br />

DING, Jian, Shanghai 201203, CN<br />

ZUO, Jianping, Shanghai 201203, CN<br />

YU, Linqian, Shanghai 201203, CN<br />

MENG, Linghua, Shanghai 201203, CN<br />

ZHANG, Yangming, Shanghai 201203, CN<br />

YANG, Na, Shanghai 201203, CN<br />

GU, Min, Shanghai 201203, CN<br />

(74) Kador & Partner, Corneliusstrasse 15, 80469<br />

München, DE<br />

C07D 513/04 → (51) C07D 235/16<br />

(51) C07F 5/00 (11) 2 351 758 A1<br />

C07F 13/00 A61K 51/00<br />

A61P 35/04<br />

(25) Ru (26) En<br />

(21) 08877097.9 (22) 05.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) RU 2008/000748 05.12.2008<br />

(87) WO 2010/036140 2010/13 01.04.2010<br />

(30) 29.09.2008 RU 2008138587<br />

(54) • METALLKOMPLEXE, VERFAHREN ZU<br />

DEREN HERSTELLUNG UND DARAUF<br />

BASIERENDE RADIOPHARMAZEUTISCHE<br />

MITTEL<br />

• METAL COMPLEXES, A METHOD FOR<br />

PREPARING SAME, RADIOPHARMACEU-<br />

TICAL MEANS BASED THEREON<br />

• COMPLEXES MÉTALLIQUES, PROCÉDÉ<br />

DE PRODUCTION DE CES DERNIERS, ET<br />

AGENTS RADIO-PHARMACEUTIQUES LES<br />

UTILISANT<br />

(71) Zakrytoe Aktsionernoe Obschestvo "Farm-<br />

Sintez", Ul. Vavilova 15, Moscow 117<strong>31</strong>2, RU<br />

(72) MALYSHEVA, Anna Olegovna, Moscow<br />

125445, RU<br />

KLEMENTYEVA, Olga Evgenievna, Moscow<br />

123592, RU<br />

KODINA, Galina Evgenievna, Moscow<br />

123592, RU<br />

KORSUNSKY, Valentin Nikolaevich, Moscow<br />

127369, RU<br />

NAZARENKO, Mihail Evgenievich, Moscow<br />

11<strong>31</strong>91, RU<br />

MIHAYLOV, Oleg Rotislavovich, Moscow<br />

129642, RU<br />

411<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2011</strong>) 03.08.<strong>2011</strong><br />

PERMINOV, Sergei Vladimirovich, Moscow<br />

109444, RU<br />

UVAROV, Nikolai Aleksandrovich, Moscow<br />

127410, RU<br />

FEDOROV, Vladimir Egorovich, Moscow<br />

125028, RU<br />

(74) Held, Stephan, et al, Meissner, Bolte &<br />

Partner GbR Widenmayerstraße 48, D-80538<br />

München, DE<br />

(51) C07F 7/10 (11) 2 351 759 A1<br />

C09K 11/06 H01L 51/50<br />

(25) Ja (26) En<br />

(21) 09824553.3 (22) 28.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2009/005689 28.10.2009<br />

(87) WO 2010/052852 2010/19 14.05.2010<br />

(30) 10.11.2008 JP 2008287919<br />

(54) • AROMATISCHES AMINDERIVAT UND<br />

ORGANISCHES ELEKTROLUMINESZENZ-<br />

ELEMENT DAMIT<br />

• AROMATIC AMINE DERIVATIVE, AND<br />

ORGANIC ELECTROLUMINESCENT ELE-<br />

MENT COMPRISING SAME<br />

• DÉRIVÉ D AMINE AROMATIQUE ET ÉLÉ-<br />

MENT ÉLECTROLUMINESCENT LE COM-<br />

PRENANT<br />

(71) Idemitsu Kosan Co., Ltd., 1-1 Marunouchi 3chome,<br />

Chiyoda-ku Tokyo 100-8321, JP<br />

(72) MIZUKI, Yumiko, Sodegaura-shi Chiba 299-<br />

0293, JP<br />

ITO, Mitsunori, Sodegaura-shi Chiba 299-<br />

0293, JP<br />

FUNAHASHI, Masakazu, Sodegaura-shi<br />

Chiba 299-0293, JP<br />

(74) Gille Hrabal Struck Neidlein Prop Roos,<br />

<strong>Patent</strong>anwälte Brucknerstrasse 20, 40593<br />

Düsseldorf, DE<br />

(51) C07F 7/10 (11) 2 351 760 A1<br />

C09K 11/06 H01L 51/50<br />

H05B 33/12<br />

(25) Ja (26) En<br />

(21) 09824632.5 (22) 09.11.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2009/005953 09.11.2009<br />

(87) WO 2010/052932 2010/19 14.05.2010<br />

(30) 07.11.2008 JP 2008286479<br />

(54) • VERBINDUNG MIT TRIPHENYLSILYL-<br />

GRUPPE UND TRIARYLAMINSTRUKTUR<br />

SOWIE ORGANISCHES ELEKTROLUMI-<br />

NESZENZELEMENT<br />

• COMPOUND HAVING TRIPHENYLSILYL<br />

GROUP AND TRIARYLAMINE STRUCTURE<br />

AND ORGANIC ELECTROLUMINESCENT<br />

ELEMENT<br />

• COMPOSÉ AYANT UN GROUPE TRIPHÉ-<br />

NYLSILYLE ET UNE STRUCTURE DE<br />

TRIARYLAMINE ET ÉLÉMENT ÉLECTRO-<br />

LUMINESCENT ORGANIQUE<br />

(71) Hodogaya Chemical Co., Ltd., 2-4-1, Shiba<br />

koen Minato-ku, Tokyo 105-0011, JP<br />

Shinshu University, 3-1-1, Asahi, Matsumoto-shi,<br />

Nagano 390-8621, JP<br />

(72) YOKOYAMA, Norimasa, Tsukuba-shi Ibaraki<br />

305-0841, JP<br />

HAYASHI, Shuichi, Tsukuba-shi Ibaraki 305-<br />

0841, JP<br />

TANIGUCHI, Yoshio, Ueda-shi Nagano 386-<br />

8567, JP<br />

ICHIKAWA, Musubu, Ueda-shi Nagano 386-<br />

8567, JP<br />

MATSUKI, Shinichi, Ueda-shi Nagano 386-<br />

8567, JP

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