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Bulletin 2010/35 - European Patent Office

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(C07C) I.1(2)<br />

Tennant, Brent, Alain, Kingsport, TN 37660-<br />

5075, US<br />

(74) Wibbelmann, Jobst, Wuesthoff & Wuesthoff<br />

<strong>Patent</strong>- und Rechtsanwälte Schweigerstrasse<br />

2, 81541 München, DE<br />

(62) 02737303.4 / 1 392 634<br />

C07C 53/00 → (51) C12P 7/52<br />

C07C 63/26 → (51) C07C 51/265<br />

C07C 67/31 → (51) C07C 2<strong>35</strong>/06<br />

C07C 67/313 → (51) C07C 2<strong>35</strong>/06<br />

C07C 68/00 → (51) C07C 41/54<br />

C07C 69/675 → (51) C07C 2<strong>35</strong>/06<br />

(51) C07C 2<strong>35</strong>/06 (11) 2 223 909 A1<br />

C07C 67/31 C07C 67/313<br />

C07C 69/675 C07D 239/42<br />

C07F 9/5<strong>35</strong><br />

(25) En (26) En<br />

(21) 10164317.9 (22) 27.08.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(30) 28.08.2007 EP 07016872<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

PENTANDISÄUREDERIVATE<br />

• Process for preparing pentanoic diacid<br />

derivatives<br />

• PROCÉDÉ DE FABRICATION DE DÉRIVÉS<br />

DE DIACIDE PENTANOÏQUE<br />

(71) Ratiopharm GmbH, Graf-Arco-Strasse 3,<br />

89079 Ulm, DE<br />

(72) Börner, Armin, 18059 Rostock, DE<br />

König, Gerd, 08056 Zwickau, DE<br />

Andrushko, Vasyl, 76137 Karlsruhe, DE<br />

Andrushko, Natalia, 76137 Karlsruhe, DE<br />

(74) Teipel, Stephan, et al, Lederer & Keller<br />

<strong>Patent</strong>anwälte Prinzregentenstrasse 16,<br />

80538 München, DE<br />

(62) 08801731.4 / 2 181 089<br />

(51) C07C 251/66 (11) 2 223 910 A1<br />

C07C 255/64 C07C 323/47<br />

C07C 323/63 C07C 391/02<br />

C07D 215/18 C07D 307/91<br />

C07D 327/08 C07D 333/76<br />

C07D 345/00 C07F 9/50<br />

C08F 2/50 C08L 101/00<br />

(25) Ja (26) En<br />

(21) 07860061.6 (22) 25.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(86) JP 2007/074832 25.12.2007<br />

(87) WO 2009/081483 2009/27 02.07.2009<br />

(54) • OXIMESTER UND PHOTOPOLYMERISA-<br />

TIONSINITIATOREN, DIE DIESE ENTHAL-<br />

TEN<br />

• OXIME ESTERS AND PHOTOPOLYMERI-<br />

ZATION INITIATORS CONTAINING THE<br />

SAME<br />

• ESTERS D'OXIME ET INITIATEURS DE<br />

PHOTOPOLYMÉRISATION LES CONTE-<br />

NANT<br />

(71) Adeka Corporation, 2-<strong>35</strong>, Higashiogu 7chome<br />

Arakawa-ku, Tokyo 116-8554, JP<br />

(72) SAWAMOTO, Daisuke, Tokyo 116-8554, JP<br />

TOMINAGA, Nobuhide, Tokyo 116-8554, JP<br />

(74) Forstmeyer, Dietmar, et al, BOETERS &<br />

LIECK Oberanger 32, 80331 München, DE<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

C07C 255/64 → (51) C07C 251/66<br />

C07C 317/28 → (51) A61K 31/40<strong>35</strong><br />

C07C 323/47 → (51) C07C 251/66<br />

C07C 323/63 → (51) C07C 251/66<br />

C07C 391/02 → (51) C07C 251/66<br />

(51) C07D 201/04 (11) 2 223 911 A1<br />

C07D 225/02 C07B 61/00<br />

(25) Ja (26) En<br />

(21) 08853278.3 (22) 19.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/071044 19.11.2008<br />

(87) WO 2009/069522 2009/23 04.06.2009<br />

(30) 29.11.2007 JP 2007308746<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

LAUROLACTAM<br />

• METHOD FOR PRODUCTION OF LAURO-<br />

LACTAM<br />

• PROCÉDÉ DE FABRICATION DE LAURO-<br />

LACTAME<br />

(71) Ube Industries, Ltd., 1978-96, Oaza Kogushi,<br />

Ube-shi Yamaguchi 755-8633, JP<br />

(72) KUGIMOTO, Junichi, Ube-shi Yamaguchi<br />

755-8633, JP<br />

KAWAI, Joji, Ube-shi Yamaguchi 755-8633,<br />

JP<br />

SHIMOMURA, Hideo, Ube-shi Yamaguchi<br />

755-8633, JP<br />

YASUMATSU, Ryouta, Ube-shi Yamaguchi<br />

755-8633, JP<br />

II, Nobuhiro, Ube-shi Yamaguchi 755-8633,<br />

JP<br />

(74) Cabinet Plasseraud, 52, rue de la Victoire,<br />

75440 Paris Cedex 09, FR<br />

C07D 209/08 → (51) C07D 401/12<br />

C07D 209/48 → (51) A61K 31/40<strong>35</strong><br />

C07D 209/86 → (51) H01L 51/50<br />

(51) C07D 213/61 (11) 2 223 912 A1<br />

(25) Ja (26) En<br />

(21) 08863865.5 (22) 19.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/073221 19.12.2008<br />

(87) WO 2009/081872 2009/27 02.07.2009<br />

(30) 21.12.2007 JP 2007330516<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINES 6-<br />

HALOGENO-3-ARYLPYRIDIN-DERIVATS<br />

• METHOD FOR PRODUCING 6-HALOGENO-<br />

3-ARYLPYRIDINE DERIVATIVE<br />

• PROCÉDÉ DE FABRICATION D'UN DÉRIVÉ<br />

DE 6-HALOGÉNO-3-ARYLPYRIDINE<br />

(71) Kuraray Co., Ltd., 1621, Sakazu Kurashikishi,<br />

Okayama 710-8622, JP<br />

(72) KASHIKI, Nobusuke, Tainai-shi Niigata 959-<br />

2653, JP<br />

MORI, Toshiki, Tsukuba-shi Ibaraki 305-<br />

0841, JP<br />

UJITA, Katsuji, Tainai-shi Niigata 959-2653,<br />

JP<br />

(74) Copsey, Timothy Graham, et al, Kilburn &<br />

Strode LLP 20 Red Lion Street, GB-London<br />

WC1R 4PJ, GB<br />

C07D 215/18 → (51) C07C 251/66<br />

254<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

C07D 225/02 → (51) C07D 201/04<br />

(51) C07D 231/54 (11) 2 223 913 A1<br />

C07D 405/12 C07D 491/04<br />

A61K 31/4155 A61K 31/416<br />

A61K 9/107<br />

(25) En (26) En<br />

(21) 10154393.2 (22) 23.02.<strong>2010</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(30) 25.02.2009 IT MI20090262<br />

(54) • Tricyclische Pyrazolderivate und deren<br />

Mikroemulsionen als CB1- und/oder CB2-<br />

Inhibitoren<br />

• Tricyclic pyrazole derivatives and microemulsions<br />

thereof as CB1- and/or CB2inhibitors<br />

• Dérivés de pyrazole tricycliques et leurs<br />

microémulsions comme inhibiteurs de CB1<br />

et/ou CB2<br />

(71) Neuroscienze Pharmaness S.C. A R.L., Loc.<br />

Piscinamanna Edificio 5, 09010 Pula (CA), IT<br />

(72) Lazzari, Paolo, 09010, PULA (CAGLIARI), IT<br />

Loriga, Giovanni, 07100, SASSARI, IT<br />

Manca, Ilaria, 07100, SASSARI, IT<br />

Pinna, Gerard Aime, 07100, SASSARI, IT<br />

(74) Sama, Daniele, Sama <strong>Patent</strong>s, Via G.B.<br />

Morgagni, 2, 20129 Milano, IT<br />

(51) C07D 231/54 (11) 2 223 914 A1<br />

C07D 491/04 A61K 31/4184<br />

A61K 31/4188 A61K 31/4155<br />

A61K 31/416 A61P 3/00<br />

A61P 25/00 A61P <strong>35</strong>/00<br />

(25) En (26) En<br />

(21) 10154463.3 (22) 24.02.<strong>2010</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(30) 25.02.2009 IT MI20090263<br />

(54) • Tricyclische kondensierte Pyrazolderivate<br />

als CB1-Inhibitoren<br />

• Tricyclic condensed pyrazole derivatives as<br />

CB1 inhibitors<br />

• Dérivés de pyrazole tricycliques condensés<br />

comme inhibiteurs de CB1<br />

(71) Neuroscienze Pharmaness S.C. A R.L., Loc.<br />

Piscinamanna Edificio 5, 09010 Pula (CA), IT<br />

(72) Lazzari, Paolo, 09010, Pula (CAGLIARI), IT<br />

Loriga, Giovanni, 07100, SASSARI, IT<br />

Manca, Ilaria, 07100, SASSARI, IT<br />

Pinna, Gerard Aime, 07100, SASSARI, IT<br />

(74) Sama, Daniele, Sama <strong>Patent</strong>s, Via G.B.<br />

Morgagni, 2, 20129 Milano, IT<br />

(51) C07D 233/58 (11) 2 223 915 A1<br />

(25) En (26) En<br />

(21) 09002653.5 (22) 25.02.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(54) • Ionische, flüssige Lösemittel<br />

• Ionic liquid solvents<br />

• Solvants liquides ioniques<br />

(71) Dublin City University, Collins Avenue Glasnevin,<br />

Dublin D9, IE<br />

(72) Gathergood, Nicholas, Ashbourne, County<br />

Meath, IE<br />

Morrissey, Saibh, Artane, Dublin 9, IE<br />

Pegot, Bruce, 94340 Joinville-le-pont, FR<br />

Beadham, Ian, Santry, Dublin 9, IE<br />

Gurbisz, Monika, Glasnevin, Dublin 9, IE<br />

Ghavre, Mukund, D., Santry, Dublin 9, IE

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