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Bulletin 2010/35 - European Patent Office

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(C07D) II.1(1)<br />

(74) Schlich, George William, et al, Schlich & Co<br />

34 New Road, Littlehampton West Sussex<br />

BN17 5AT, GB<br />

C07D 487/04 → (51) C07D 491/04<br />

(51) C07D 491/04 (11) 1 469 809 B1<br />

C07D 487/04 A61K 31/519<br />

A61P <strong>35</strong>/00<br />

(25) En (26) En<br />

(21) 02801736.6 (22) 16.10.2002<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SK TR<br />

(43) 27.10.2004<br />

(86) US 2002/032963 16.10.2002<br />

(87) WO 2003/032911 2003/17 24.04.2003<br />

(30) 18.10.2001 US 982<strong>35</strong>1<br />

(54) • MEHRFACH WIRKENDE ANTIANGIOGENE<br />

UND ZYTOTOXISCHE VERBINDUNGEN<br />

UND VERFAHREN ZU IHRER VERWEN-<br />

DUNG<br />

• MULTIPLE ACTING ANTI-ANGIOGENIC<br />

AND CYTOTOXIC COMPOUNDS AND<br />

METHODS FOR USING THE SAME<br />

• COMPOSES ANTI-ANGIOGENIQUES ET<br />

CYTOTOXIQUES A EFFETS MULTIPLES ET<br />

LEURS PROCEDES D'UTILISATION<br />

(73) DUQUESNE UNIVERSITY OF THE HOLY<br />

GHOST, 505 Administration Building, Pittsburgh,<br />

PA 15282, US<br />

(72) GANGJEE, Aleem, Allison Park, PA 15101,<br />

US<br />

(74) Barton, Matthew Thomas, et al, Forrester &<br />

Boehmert Pettenkoferstrasse 20-22, 80336<br />

München, DE<br />

C07D 493/04 → (51) C07D 319/06<br />

(51) C07D 495/04 (11) 1 963 337 B1<br />

A61K 31/4365 A61P 25/00<br />

(25) En (26) En<br />

(21) 06831522.5 (22) 19.12.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 03.09.2008<br />

(86) HU 2006/000123 19.12.2006<br />

(87) WO 2007/072095 2007/26 28.06.2007<br />

(30) 20.12.2005 HU 0501171<br />

18.12.2006 HU 0600920<br />

(54) • THIENO[2,3-b]PYRIDIN DERIVATE<br />

• THIENO[2,3-b]PYRIDINE DERIVATIVES<br />

• COMPOSÉS DE THIENO[2,3-b]PYRIMI-<br />

DINE<br />

(73) Richter Gedeon Nyrt., Gyömröi út 19-21,<br />

1103 Budapest, HU<br />

(72) NÓGRÁDI, Katalin, H-1182 Budapest, HU<br />

WÁGNER, Gábor, H-1107 Budapest, HU<br />

KESERÜ, György, H-2089 Telki, HU<br />

BIELIK, Attila, H-2377 Örkény, HU<br />

GÁTI, Tamás, H-1114 Budapest, HU<br />

HÁDA, Viktor, H-1108 Budapest, HU<br />

KÓTI, János, H-4440 Tiszavasvári, HU<br />

GÁL, Krisztina, H-1193 Budapest, HU<br />

VASTAG, Mónika, H-1025 Budapest, HU<br />

BOBOK, Amrita, Ágnes, H-1025 Budapest,<br />

HU<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

(51) C07D 495/04 (11) 2 102 215 B1<br />

A61K 31/4365 A61P 3/04<br />

A61P 3/10<br />

(25) En (26) En<br />

(21) 07857234.4 (22) 28.11.2007<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 23.09.2009<br />

(86) EP 2007/062930 28.11.2007<br />

(87) WO 2008/068174 2008/24 12.06.2008<br />

(30) 08.12.2006 EP 06125715<br />

(54) • 4,5,6,7-TETRAHYDROTHIENO[2,3-C]PYRI-<br />

DINE ALS H3-MODULATOREN<br />

• 4,5,6,7-TETRAHYDRO-THIENO [2,3-C]<br />

PYRIDINES AS H3 MODULATORS<br />

• 4,5,6,7-TÉTRAHYDRO-THIÉNO [2,3-C]<br />

PYRIDINES EN TANT QUE MODULATEURS<br />

DE H3<br />

(73) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) CHEN, Li, Shanghai 201203, CN<br />

LAI, Wayne Wen, Shanghai 201203, CN<br />

NETTEKOVEN, Matthias, 79639 Grenzach-<br />

Wyhlen, DE<br />

ROCHE, Olivier, 68220 Folgensbourg, FR<br />

ZHENG, Deye, Shanghai 201204, CN<br />

(74) Klostermeyer-Rauber, Dörte, F. Hoffmann-La<br />

Roche AG Corporate Law <strong>Patent</strong>s (CLP)<br />

Grenzacherstrasse 124, 4070 Basel, CH<br />

C07D 495/04 → (51) A61K 31/519<br />

(51) C07D 498/04 (11) 2 004 657 B1<br />

C07D 513/04 A61K 31/5383<br />

A61K 31/542 A61P 9/00<br />

A61P 3/00<br />

(25) En (26) En<br />

(21) 07728050.1 (22) 12.04.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 24.12.2008<br />

(86) EP 2007/05<strong>35</strong>83 12.04.2007<br />

(87) WO 2007/116097 2007/42 18.10.2007<br />

(30) 12.04.2006 CH 617062006<br />

(54) • KONDENSIERTE IMIDAZOLDERIVATE ALS<br />

ALDOSTERONSYNTHASEINHIBITOREN<br />

• CONDENSED IMIDAZOLE DERIVATIVES<br />

AS ALDOSTERONE SYNTHASE INHIBI-<br />

TORS<br />

• DÉRIVÉS D'IMIDAZOLE CONDENSÉS UTI-<br />

LISÉS EN TANT QU'INHIBITEURS DE<br />

L'ALDOSTÉRONE SYNTHASE<br />

(73) Novartis AG, Lichtstrasse <strong>35</strong>, 4056 Basel, CH<br />

(72) HEROLD, Peter, 4123 Allschwil, CH<br />

MAH, Robert, 4123 Allschwil, CH<br />

TSCHINKE, Vincenzo, 4123 Allschwil, CH<br />

STOJANOVIC, Aleksandar, 4123 Allschwil,<br />

CH<br />

MARTI, Christiane, 4123 Allschwil, CH<br />

STUTZ, Stefan, 4123 Allschwil, CH<br />

BENNACER, Bibia, 4123 Allschwil, CH<br />

(74) Carpmaels & Ransford, One Southampton<br />

Row, London WC1B 5HA, GB<br />

C07D 513/04 → (51) C07D 471/04<br />

C07D 513/04 → (51) C07D 498/04<br />

C07D 519/00 → (51) C07D 471/04<br />

(51) C07F 7/00 (11) 1 972 634 B1<br />

C09B 67/50 G03G 5/06<br />

(25) En (26) En<br />

(21) 08153160.0 (22) 20.03.2008<br />

(84) CH DE FR GB LI<br />

(43) 24.09.2008<br />

(30) 23.03.2007 JP 2007076598<br />

588<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

(54) • Titanylphthalocyanin umfassend ein spezifisches<br />

Polymorph und Herstellungsverfahren<br />

dafür sowie elektrofotografischer<br />

Fotorezeptor umfassend ladungserzeugendes<br />

Material daraus<br />

• Titanylphthalocyanine comprising specific<br />

polymorph and method for producing<br />

thereof, and electrophotographic photoreceptor<br />

comprising charge generating<br />

material thereof<br />

• Titanylphtalocyanine comprenant un polymorphe<br />

particulier et son procédé de<br />

fabrication, et photorécepteur électrophotographique<br />

comprenant son matériau de<br />

génération de charge<br />

(73) ORIENT CHEMICAL INDUSTRIES, LTD., 7-<br />

14, Shinmori 1-chome, Asahi-ku, Osaka-shi,<br />

Osaka, JP<br />

(72) Takaki, Kenji, Neyagawa-shi Osaka, JP<br />

Yamasaki, Yasuhiro, Neyagawa-shi Osaka,<br />

JP<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

(51) C07F 7/18 (11) 1 770 097 B1<br />

(25) En (26) En<br />

(21) 06255090.0 (22) 02.10.2006<br />

(84) DE FR IT<br />

(43) 04.04.2007<br />

(30) 30.09.2005 JP 2005285868<br />

(54) • Herstellung von sulfidkettentragenden<br />

Organosiliziumverbindungen<br />

• Preparation of sulfide chain-bearing organosilicon<br />

compounds<br />

• Préparation de composés organosiliciques<br />

portant un chaîne de sulfure<br />

(73) Shin-Etsu Chemical Co., Ltd., 6-1, Otemachi<br />

2-chome, Chiyoda-ku, Tokyo, JP<br />

(72) Yanagisawa, Hideyoshi, Shin-Etsu Chemical<br />

Co., Ltd, Matsuida-machi, Annaka-shi,<br />

Gunma-ken, JP<br />

(74) Stoner, Gerard Patrick, et al, Mewburn Ellis<br />

LLP 33 Gutter Lane, London EC2V 8AS, GB<br />

C07F 7/22 → (51) C07D 215/54<br />

C07F 9/02 → (51) C07B 63/00<br />

(51) C07F 9/6561 (11) 1 961 757 B1<br />

A61K 31/675 A61P 31/18<br />

(25) En (26) En<br />

(21) 08075531.7 (22) 16.09.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 27.08.2008<br />

(30) 17.09.2004 US 611061<br />

25.08.2005 US 711445<br />

26.08.2005 US 711565<br />

(54) • Phosphoindole als HIV-Inhibitoren<br />

• Phosphoindoles as HIV inhibitors<br />

• Phosphoindoles utilisés en tant qu'inhibiteurs<br />

du VIH<br />

(73) IDENIX Pharmaceuticals, Inc., One Kendall<br />

Square, Building 1400, Cambridge, MA<br />

02139, US<br />

(72) Storer, Richard, Folkestone, Kent, CT20 2JE,<br />

GB<br />

Dousson Cyril, F-34080 Montpellier, FR<br />

Alexandre, Francois-René, F-34090 Montpellier,<br />

FR<br />

Roland, Arlène, F-34590 Marsillargues, FR<br />

(74) Howard, Paul Nicholas, et al, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

(62) 05850774.0 / 1 799 696

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