Bulletin 2010/35 - European Patent Office

(C07D) I.1(1)
• 3-HETEROCYCLIC SUBSTITUTED INDOLE
DERIVATIVES AND METHODS OF USE
THEREOF
• DÉRIVÉS D'INDOLE À SUBSTITUTION
HÉTÉROCYCLIQUE EN POSITION 3 ET
LEURS PROCÉDÉS D'UTILISATION
(71) Schering Corporation, 2000 Galloping Hill
Road, Kenilworth, NJ 07033-0530, US
(72) CHAN, Tin-Yau, Edison New Jersey 08817,
US
DUCA, Jose, S., Cranford New Jersey 07016,
US
HONG, Liwu, Edison New Jersey 08817, US
LESBURG, Charles, A., Short Hills New
Jersey 07078, US
MCKITTRICK, Brian, A., New Vernon New
Jersey 07976, US
PU, Haiyan, Livingston New Jersey 07039,
US
WANG, Li, Nanuet New York 10954, US
VACCARO, Henry, M., South Plainfield New
Jersey 07080, US
(74) van den Broek, Ludovicus A.G.M., et al, P.O.
Box 20, 5340 BH Oss, NL
C07D 401/04 → (51) C07D 207/16
(51) C07D 401/06 (11) 2 222 661 A2*
C07D 471/04 A61K 31/44
A61P 31/18
(25) En (26) En
(21) 08851089.6 (22) 14.11.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) US 2008/012774 14.11.2008
(87) WO 2009/067166 2009/22 28.05.2009
(88) 16.07.2009
(30) 20.11.2007 US 3769
(54) • NICHT-NUKLEOSIDISCHE REVERSE-
TRANSKRIPTASE-HEMMER
• NON-NUCLEOSIDE REVERSE TRAN-
SCRIPTASE INHIBITORS
• INHIBITEURS NON-NUCLÉOSIDIQUES DE
LA TRANSCRIPTASE INVERSE
(71) Merck Sharp & Dohme Corp., 126 East
Lincoln Avenue, Rahway, NJ 07065, US
(72) TUCKER, Thomas, J., Rahway New Jersey
07065-0907, US
TYNEBOR, Robert, Rahway New Jersey
07065-0907, US
SISKO, John, T., Rahway New Jersey 07065-
0907, US
ANTHONY, Neville, Rahway New Jersey
07065-0907, US
GOMEZ, Robert, Rahway New Jersey 07065-
0907, US
JOLLY, Samson, M., Rahway New Jersey
07065-0907, US
(74) Horgan, James Michael Frederic, Merck &
Co., Inc. European Patent Department Merck
Sharpe & Dohme Limited Hertford Road,
Hoddesdon Hertfordshire EN11 9BU, GB
C07D 401/06 → (51) C07D 207/16
(51) C07D 401/10 (11) 2 222 662 A2*
(25) En (26) En
(21) 08850245.5 (22) 13.11.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) US 2008/083321 13.11.2008
(87) WO 2009/064836 2009/21 22.05.2009
(88) 02.07.2009
(30) 15.11.2007 US 988231 P
Europäisches Patentblatt
European Patent Bulletin
Bulletin européen des brevets
(54) • INHIBITOREN DER KYNURENIN-AMINOT-
RANSFERASE
• KYNURENINE-AMINOTRANSFERASE INHI-
BITORS
• INHIBITEURS DE LA KYNURÉNINE-AMI-
NOTRANSFÉRASE
(71) University of Maryland, Baltimore, 520 West
Lombard Street, Baltimore MD 21201, US
Mitsubishi Tanabe Pharma Corporation, 2-
10, Dosho-machi 3-chome, Chuo-ku Osakashi
Osaka 541-8505, JP
(72) SCHWARCZ, Robert, Baltimore MD 21208,
US
KAJII, Yasushi, Osaka 541-8505, JP
ONO, Shin-ichiro, Osaka 541-8505, JP
(74) Kröncke, Rolf, et al, Gramm, Lins & Partner
Patent- und Rechtsanwaltssozietät GbR
Freundallee 13a, 30173 Hannover, DE
C07D 401/10 → (51) C07D 239/22
C07D 401/10 → (51) C07D 239/48
C07D 401/10 → (51) C07F 17/02
(51) C07D 401/12 (11) 2 222 663 A1*
(25) En (26) En
(21) 08870010.9 (22) 18.12.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) IN 2008/000842 18.12.2008
(87) WO 2009/087672 2009/29 16.07.2009
(30) 18.12.2007 IN MU24892007
(54) • VERFAHREN ZUR HERSTELLUNG VON
STABILEM AMORPHEM R-LANSOPRAZOL
• A PROCESS FOR PREPARATION OF
STABLE AMORPHOUS R-LANSOPRAZOLE
• PROCÉDÉ DE PRÉPARATION DE R-LAN-
SOPRAZOLE AMORPHE STABLE
(71) Watson Pharma Private Limited, 201/301,
Corporate Enclave HDO-Corporate Bldg, B
Wing B.D. Sawant Marg, Chakala Off Wester
Express Highway Andheri (East), Mumbai
400 099, IN
(72) NAIK, Samir, Thane 400 604 Maharashtra, IN
BODKE, Arjun, Ulhasnagar 3, IN
MAHAJAN, Kishor, Maharashtra, IN
BHANU, Manjunath, Narayan, Pune 211 021
Maharashtra, IN
(74) Shaw, Matthew Nigel, Forrester & Boehmert
Pettenkoferstrasse 20-22, 80336 München,
DE
C07D 401/12 → (51) C07D 239/48
(51) C07D 401/14 (11) 2 222 664 A1*
C07D 407/14 C07D 409/14
A61K 31/495 A61P 25/00
(25) En (26) En
(21) 08852442.6 (22) 17.11.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) US 2008/083764 17.11.2008
(87) WO 2009/067401 2009/22 28.05.2009
(30) 20.11.2007 US 989246 P
(54) • CYCLOALKYLOXY- UND HETEROCYC-
LOALKYLOXYPYRIDINVERBINDUNGEN
ALS MODULATOREN DES HISTAMIN-H3-
REZEPTORS
• CYCLOALKYLOXY-AND HET ROCY-
CLOALKY- LOXYPYRIDINE COMPOUNDS
AS MODULATORS OF THE HISTAMINE H3
RECEPTOR
88
Anmeldungen
Applications
Demandes (35/2010) 01.09.2010
• COMPOSÉS CYCLOALKYLOXY-PYRIDINE
ET HÉTÉROCYCLOALKYLOXY-PYRIDINE
COMME MODULATEURS DU RÉCEPTEUR
H3 DE L'HISTAMINE
(71) Janssen Pharmaceutica, N.V., Turnhoutseweg
30, 2340 Beerse, BE
(72) LETAVIC, Michael A., San Diego California
92130, US
STOCKING, Emily M., Encinitas California
92024, US
(74) Warner, James Alexander, Carpmaels &
Ransford One Southampton Row, London
WC1B 5HA, GB
C07D 403/04 → (51) C07D 401/04
(51) C07D 403/06 (11) 2 222 665 A1*
C07D 409/14 A61K 31/41
A61P 15/00
(25) En (26) En
(21) 08849494.3 (22) 06.11.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) IB 2008/054634 06.11.2008
(87) WO 2009/063365 2009/21 22.05.2009
(30) 15.11.2007 US 988184 P
(54) • AZETIDINE ALS EP-2-ANTAGONISTEN
• AZETIDINES AS EP2 ANTAGONISTS
• AZÉTIDINES COMME ANTAGOSNISTES DE
L' EP2
(71) Pfizer Limited, Ramsgate Road, Sandwich,
Kent CT13 9NJ, GB
(72) SKERRATT, Sarah Elizabeth, Sandwich Kent
CT13 9NJ, GB
DACK, Kevin Neil, Sandwich Kent CT13 9NJ,
GB
(74) Cosway, Sarah Michelle, Pfizer Limited
European Patent Department Ramsgate
Road, Sandwich, Kent CT13 9NJ, GB
C07D 403/06 → (51) C07D 241/24
C07D 403/10 → (51) C07D 239/22
C07D 403/10 → (51) C07D 239/48
C07D 403/12 → (51) C07D 239/48
C07D 403/14 → (51) C07D 239/48
C07D 403/14 → (51) C07D 401/04
C07D 405/06 → (51) C07D 455/02
C07D 405/10 → (51) C07D 309/28
(51) C07D 405/12 (11) 2 222 666 A1*
A61P 9/12 A61P 13/08
A61K 31/517
(25) En (26) En
(21) 08775904.9 (22) 10.07.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
AL BA MK RS
(86) GB 2008/002362 10.07.2008
(87) WO 2009/081087 2009/27 02.07.2009
(30) 24.12.2007 IN MU25372007
(54) • KRISTALLINES POLYMORPH VON DOXA-
ZOSIN-MESYLAT (FORM IV) UND VER-
FAHREN ZU DEREN HERSTELLUNG
• CRYSTALLINE POLYMORPH OF DOXAZO-
SIN MESYLATE (FORM IV) AND PROCESS
FOR PREPARATION THEREOF