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Bulletin 2010/35 - European Patent Office

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(C07D) II.1(1)<br />

(73) BASF SE, 67056 Ludwigshafen, DE<br />

(72) EHLIS, Thomas, 79100 Freiburg, DE<br />

HÜGLIN, Dietmar, 79576 Weil am Rhein, DE<br />

BORSOS, Elek, CH-4127 Birsfelden, CH<br />

C07D 251/20 → (51) C07D 251/18<br />

C07D 261/10 → (51) C07D 213/71<br />

(51) C07D 261/12 (11) 2 022 788 B1<br />

A61K 31/42 A61P 19/02<br />

(25) Ja (26) En<br />

(21) 07744104.6 (22) 25.05.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

HR RS<br />

(43) 11.02.2009<br />

(86) JP 2007/060670 25.05.2007<br />

(87) WO 2007/138996 2007/49 06.12.2007<br />

(30) 26.05.2006 JP 2006146220<br />

(54) • NEUER KRISTALL VON 3-[5-[4-(CYCLO-<br />

PENTYLOXY)-2-HYDROXYBENZOYL]-2-<br />

[(3-HYDROXY-1,2-BENZISOXAZOL-6-YL)<br />

METHOXY]PHENYL]PROPIONSÄURE<br />

• NOVEL CRYSTAL OF 3-[5-[4-(CYCLOPEN-<br />

TYLOXY)-2- HYDROXYBENZOYL]-2-[(3-<br />

HYDROXY-1,2-BENZISOXAZOL-6-YL)<br />

METHOXY]PHENYL]PROPIONIC ACID<br />

• NOUVEAU CRISTAL D'ACIDE 3-[5-[4-<br />

(CYCLOPENTYLOXY)-2-HYDROXYBEN-<br />

ZOYL]-2-](3-HYDROXY-1,2-BENZISOXA-<br />

ZOL-6-YL)MÉTHOXY]PHÉNYL]PROPIO-<br />

NIQUE<br />

(73) TOYAMA CHEMICAL CO., LTD., 2-5, 3chome,<br />

Nishishinjuku, Shinjuku-ku, Tokyo<br />

160-0023, JP<br />

(72) YONEZAWA, Kenji, Toyama-shi, Toyama<br />

9308508, JP<br />

KOTSUBO, Hironori, Toyama-shi, Toyama<br />

9308508, JP<br />

BABA, Yasutaka, Toyama-shi, Toyama<br />

9308508, JP<br />

TADA, Yukie, Toyama-shi, Toyama 9308508,<br />

JP<br />

(74) Hartz, Nikolai, Wächtershäuser & Hartz<br />

<strong>Patent</strong>anwaltspartnerschaft Weinstrasse 8,<br />

80333 München, DE<br />

(51) C07D 277/34 (11) 1 594 854 B1<br />

C07D 277/46 A61K 31/4439<br />

A61P 29/00<br />

(25) En (26) En<br />

(21) 04709122.8 (22) 06.02.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

AL LT LV MK<br />

(43) 16.11.2005<br />

(86) US 2004/003879 06.02.2004<br />

(87) WO 2004/071440 2004/<strong>35</strong> 26.08.2004<br />

(30) 06.02.2003 US 445410 P<br />

(54) • ALS KINASEINHIBITOREN GEEIGNETE<br />

VERBINDUNGEN AUF THIAZOLYLBASIS<br />

• THIAZOLYL-BASED COMPOUNDS USEFUL<br />

AS KINASE INHIBITORS<br />

• COMPOSES A BASE DE THIAZOLYLE<br />

UTILISES COMME INHIBITEURS DE<br />

KINASES<br />

(73) Bristol-Myers Squibb Company, Route 206<br />

and Province Line Road, Princeton NJ<br />

08543-4000, US<br />

(72) HYNES, John, Washington Crossing, PA<br />

18977, US<br />

WU, Hong, New Hope PA 18938, US<br />

LEFTHERIS, Katerina, Skillman, NJ 08558,<br />

US<br />

LIU, Chunjian, Pennington, NJ 08534, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

DAS, Jagabandhu, Mercerville, NJ 08619, US<br />

MOQUIN, Robert, V., East Brunswick, NJ<br />

08816, US<br />

(74) Howard, Paul Nicholas, et al, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

C07D 277/36 → (51) C07C 323/42<br />

C07D 277/36 → (51) C07D 213/71<br />

C07D 277/46 → (51) C07D 277/34<br />

C07D 277/76 → (51) C07C 323/42<br />

(51) C07D 279/16 (11) 1 726 587 B1<br />

A61K 31/5415 A61P 29/00<br />

A61P 43/00 C07C 59/64<br />

C07C 69/734 C07C 205/56<br />

(25) Ja (26) En<br />

(21) 05720093.3 (22) 28.02.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) 29.11.2006<br />

(86) JP 2005/003821 28.02.2005<br />

(87) WO 2005/082872 2005/36 09.09.2005<br />

(30) 02.03.2004 JP 2004057808<br />

(54) • BENZOTHIAZIN-3-ONE VERBINDUNG UND<br />

ZWISCHENPRODUKT DAFÜR<br />

• BENZOTHIAZIN-3-ONE COMPOUND AND<br />

INTERMEDIATE THEREFOR<br />

• COMPOSE DE BENZOTHIAZINE-3-ONE ET<br />

PRODUIT INTERMEDIAIRE POUR CELUI-<br />

CI<br />

(73) Dainippon Sumitomo Pharma Co., Ltd., 6-8,<br />

Dosho-machi 2-chome Chuo-ku Osaka-shi,<br />

Osaka 541-8524, JP<br />

(72) SAMIZO, Fumio, 33-94, Enoki-cho, Suita-shi,<br />

Osaka, JP<br />

HORIUCHI, Yoshihiro c/o Dainippon Sumitomo<br />

Pharma Co., Ltd., Osaka-shi, Osaka, JP<br />

FUKUDA, Nobuhisa c/o Dainippon Sumitomo<br />

Pharma Co., Ltd., Osaka-shi, Osaka, JP<br />

TSUBOI, Katsunori, 33-94, Enoki-cho Suitashi,<br />

Osaka, JP<br />

MAKITA, Atsushi c/o Dainippon Sumitomo<br />

Pharma Co., Ltd., Osaka-shi, Osaka, JP<br />

(74) Duckworth, Timothy John, et al, J.A. Kemp &<br />

Co. 14 South Square Gray's Inn, London<br />

WC1R 5JJ, GB<br />

C07D 285/12 → (51) C07C 323/42<br />

(51) C07D 295/03 (11) 1 701 945 B1<br />

C07D 295/145 C07D 403/12<br />

G01N 33/58<br />

(25) En (26) En<br />

(21) 05705033.8 (22) 05.01.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) 20.09.2006<br />

(86) US 2005/000223 05.01.2005<br />

(87) WO 2005/068446 2005/30 28.07.2005<br />

(30) 05.01.2004 US 751<strong>35</strong>4<br />

05.01.2004 US 751388<br />

05.01.2004 US 751387<br />

05.01.2004 US 751<strong>35</strong>3<br />

12.04.2004 US 822639<br />

24.05.2004 US 852730<br />

(54) • MARKIERUNGSREAGENTIEN, MARKIERTE<br />

ANALYTEN, EINSCHLIESSLICH MI-<br />

SCHUNGEN DAVON, UND DAVON ABGE-<br />

LEITETE FRAGMENTIONEN UND<br />

VERFAHREN ZU DEREN ANALYSE<br />

584<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

• LABELING REAGENTS, LABELED ANA-<br />

LYTES, INCLUDING MIXTURES THEREOF,<br />

AND FRAGMENT IONS DERIVED THERE-<br />

FROM AND METHODS FOR THE ANALYSIS<br />

THEREOF<br />

• REACTIFS DE MARQUAGE, ANALYTES<br />

MARQUES, Y COMPRIS MELANGE DE<br />

CEUX-CI ET IONS-FRAGMENTS DERIVES<br />

DE CEUX-CI ET PROCEDES POUR LEUR<br />

ANALYSE<br />

(73) Life Technologies Corporation, 5791 Van<br />

Allen Way, Carlsbad, CA 92008, US<br />

(72) DEY, Subhakar, Billerica, MA 01862, US<br />

PAPPIN, Darryl, J.C., Boxborough, MA<br />

01719, US<br />

PURKAYASTHA, Subhasish, Acton, MA<br />

01720, US<br />

PILLAI, Sasi, Littleton, MA 01460, US<br />

COULL, James, M., Westford, MA 01886, US<br />

(74) Schnappauf, Georg, et al, Dr. Volker Vossius<br />

<strong>Patent</strong>- und Rechtsanwaltskanzlei Geibelstrasse<br />

6, 81679 München, DE<br />

(51) C07D 295/10 (11) 1 388 538 B1<br />

G03F 7/031 C09K 19/54<br />

G02F 1/1333<br />

(25) En (26) En<br />

(21) 03014990.0 (22) 02.07.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 11.02.2004<br />

(30) 09.07.2002 EP 02015208<br />

(54) • Polymerizationsinitiator<br />

• Polymerisation Initiator<br />

• Initiateur de polymérisation<br />

(73) Merck <strong>Patent</strong> GmbH, Frankfurter Strasse<br />

250, 64293 Darmstadt, DE<br />

(72) Eastwood, Amanda, St Denys Southampton<br />

HANTS SO17 2NU, GB<br />

Parri, Owain Llyr, Poole, Dorset BH15 2LN,<br />

GB<br />

Slaney, Kim, Christchurch, Dorset BH23<br />

1QX, GB<br />

C07D 295/1<strong>35</strong>→ (51) A61K 31/167<br />

C07D 295/145→ (51) C07D 295/03<br />

C07D 295/18 → (51) C07D 213/71<br />

C07D 295/22 → (51) C07D 213/71<br />

C07D 301/10 → (51) B01J 23/68<br />

(51) C07D 301/12 (11) 1 914 228 B1<br />

C07D 303/16<br />

(25) Ja (26) En<br />

(21) 06767689.0 (22) 30.06.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 23.04.2008<br />

(86) JP 2006/313081 30.06.2006<br />

(87) WO 2007/004549 2007/02 11.01.2007<br />

(30) 01.07.2005 JP 2005194149<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON 2-<br />

HYDROXYISOBUTTERSÄURE-GLYCIDY-<br />

LESTER<br />

• PROCESS FOR PRODUCING GLYCIDYL 2-<br />

HYDROXYISOBUTYRATE<br />

• PROCEDE DE FABRICATION DE 2-<br />

HYDROXYISOBUTYRATE DE GLYCIDYLE<br />

(73) MITSUBISHI GAS CHEMICAL COMPANY,<br />

INC., 5-2, Marunouchi 2-chome, Chiyoda-ku,<br />

Tokyo 100-8324, JP<br />

(72) SHIMA, Yoshikazu Mitsubishi Gas Chemical<br />

Co., Inc., Shinwari, Niigata-shi Niigata<br />

9503112, JP

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