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Bulletin 2010/35 - European Patent Office

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(A61K) I.1(1)<br />

(25) En (26) En<br />

(21) 08865547.7 (22) 26.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/073974 26.12.2008<br />

(87) WO 2009/082038 2009/27 02.07.2009<br />

(88) 27.08.2009<br />

(30) 26.12.2007 US 6133<br />

(54) • AMPA-REZEPTOR-ANTAGONISTEN UND<br />

ZONISAMID FÜR EPILEPSIE<br />

• AMPA RECEPTOR ANTAGONISTS AND<br />

ZONISAMIDE FOR EPILEPSY<br />

• ANTAGONISTES DES RÉCEPTEURS AMPA<br />

ET ZONISAMIDE POUR LE TRAITEMENT<br />

DE L'ÉPILEPSIE<br />

(71) Eisai R&D Management Co., Ltd., 6-10,<br />

Koishikawa 4-chome Bunkyo-ku, Tokyo 112-<br />

8088, JP<br />

(72) HANADA, Takahisa, Tsukuba-shi Ibaraki 300-<br />

26<strong>35</strong>, JP<br />

HIBI, Shigeki, New Jersey 07660-2104, US<br />

MIYAZAKI, Kazuki, Tsukuba-shi Ibaraki 300-<br />

26<strong>35</strong>, JP<br />

(74) Woods, Geoffrey Corlett, J.A. Kemp & Co. 14<br />

South Square Gray's Inn, London WC1R 5JJ,<br />

GB<br />

A61K 31/4245 → (51) C07D 413/04<br />

A61K 31/425 → (51) A01N 43/78<br />

A61K 31/425 → (51) C07D 513/04<br />

A61K 31/427 → (51) A61K 9/00<br />

A61K 31/427 → (51) A61K 31/00<br />

(51) A61K 31/429 (11) 2 222 297 A1*<br />

A61K 31/52 A61K 31/553<br />

A61K 31/198 A61K 45/06<br />

A23L 1/305 A61P <strong>35</strong>/00<br />

A61P 31/18 A61P 29/00<br />

A61P 25/28 A61P 19/02<br />

A61P 17/00 A61P 9/04<br />

A61P 3/10 A61P 1/14<br />

(25) En (26) En<br />

(21) 08855001.7 (22) 03.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/078667 03.10.2008<br />

(87) WO 2009/070378 2009/23 04.06.2009<br />

(30) 26.11.2007 US 990134 P<br />

18.03.2008 US 37371<br />

(54) • ZUSAMMENSETZUNGEN UND VERFAH-<br />

REN ZUR HEMMUNG DER AKTIVIERUNG<br />

VON DSRNA-ABHÄNGIGER PROTEINKI-<br />

NASE UND HEMMUNG DES TUMOR-<br />

WACHSTUMS<br />

• COMPOSITIONS AND METHODS FOR<br />

INHIBITING THE ACTIVATION OF DSRNA-<br />

DEPENDENT PROTEIN KINASE AND<br />

TUMOR GROWTH INHIBITION<br />

• COMPOSITIONS ET PROCÉDÉS POUR<br />

INHIBER L'ACTIVATION DE LA PROTÉINE<br />

KINASE DÉPENDANTE DE L'ARN À<br />

DOUBLE BRIN ET INHIBITION DE LA<br />

CROISSANCE DE TUMEUR<br />

(71) Nestec S.A., Avenue Nestlé 55, 1800 Vevey,<br />

CH<br />

(72) TISDALE, Michael, John, Claverdon Warwickshire<br />

CV<strong>35</strong> 8LW, GB<br />

ELEY, Helen, Laura, Rochester Kent<br />

ME37BB, GB<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

RUSSELL, Steve, Thomas, Wednesbury<br />

West Midlands WS10 7RR, GB<br />

MILLER, Kevin, Burke, Minneapolis Minnesota<br />

55404, US<br />

(74) Brearley, Helen Rebecca, Elkington and Fife<br />

LLP Prospect House 8 Pembroke Road,<br />

Sevenoaks Kent TN13 1XR, GB<br />

A61K 31/437 → (51) A61K 31/472<br />

A61K 31/437 → (51) C07D 471/04<br />

A61K 31/4375 → (51) C07D 455/02<br />

A61K 31/44 → (51) C07C 311/08<br />

A61K 31/44 → (51) C07D 401/06<br />

(51) A61K 31/4439 (11) 2 222 298 A1*<br />

A61P <strong>35</strong>/04<br />

(25) En (26) En<br />

(21) 08845565.4 (22) 29.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/081501 29.10.2008<br />

(87) WO 2009/058801 2009/19 07.05.2009<br />

(30) 02.11.2007 US 984978 P<br />

(54) • VERWENDUNG EINES CFMS-INHIBITORS<br />

ZUR BEHANDLUNG ODER PRÄVENTION<br />

VON KNOCHENKREBS UND DES KNO-<br />

CHENSCHWUNDS UND DER KNOCHEN-<br />

SCHMERZEN IM ZUSAMMENHANG MIT<br />

KNOCHENKREBS<br />

• USE OF CFMS INHIBITOR FOR TREATING<br />

OR PREVENTING BONE CANCER AND THE<br />

BONE LOSS AND BONE PAIN ASSOCIATED<br />

WITH BONE CANCER<br />

• UTILISATION D'INHIBITEUR CFMS POUR<br />

LE TRAITEMENT OU LA PRÉVENTION DU<br />

CANCER DES OS ET DE LA PERTE<br />

OSSEUSE ET DE LA DOULEUR OSSEUSE<br />

ASSOCIÉES AU CANCER DES OS<br />

(71) Janssen Pharmaceutica N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) MANTHEY, Carl L., Downingtown Pennsylvania<br />

193<strong>35</strong>, US<br />

(74) Warner, James Alexander, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

A61K 31/444 → (51) A61K 31/423<br />

(51) A61K 31/445 (11) 2 222 299 A2*<br />

A61K 31/451 A61P 29/00<br />

(25) En (26) En<br />

(21) 08852672.8 (22) 27.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/081328 27.10.2008<br />

(87) WO 2009/067317 2009/22 28.05.2009<br />

(88) 06.08.2009<br />

(30) 19.11.2007 US 988913 P<br />

(54) • VERWENDUNG VON LEVOCABASTIN ZUR<br />

MODULIERUNG DER ERZEUGUNG VON<br />

PROINFLAMMATORISCHEN ZYTOKINEN<br />

• USE OF LEVOCABASTINE FOR MODULAT-<br />

ING GENERATION OF PRO-INFLAMMA-<br />

TORY CYTOKINES<br />

• COMPOSITIONS ET PROCÉDÉS DE<br />

MODULATION DE LA PRODUCTION DE<br />

CYTOKINES PRO-INFLAMMATOIRES<br />

(71) Bausch & Lomb Incorporated, One Bausch &<br />

Lomb Place, Rochester, NY 14604-2701, US<br />

(72) BUCOLO, Claudio, I-95125 Catania, IT<br />

36<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

WARD, Keith, Wayne, Ontario NY 14519, US<br />

ZHANG, Jinzhong, Pittsford NY 14534, US<br />

(74) Glas, Holger, Maiwald <strong>Patent</strong>anwalts GmbH<br />

Elisenhof Elisenstrasse 3, 803<strong>35</strong> München,<br />

DE<br />

(51) A61K 31/445 (11) 2 222 300 A1*<br />

A61P 7/02 A61P 9/10<br />

A61P 25/02<br />

(25) En (26) En<br />

(21) 08859016.1 (22) 13.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/086734 13.12.2008<br />

(87) WO 2009/076664 2009/25 18.06.2009<br />

(30) 13.12.2007 US 13377<br />

(54) • VERFAHREN UND ZUSAMMENSETZUNG<br />

ZUR BEHANDLUNG EINES ZUSTANDS,<br />

DER DURCH DEN SEROTONIN-REZEPTOR<br />

VERMITTELT WIRD<br />

• METHOD AND COMPOSITION FOR<br />

TREATING A SEROTONIN RECEPTOR-<br />

MEDIATED CONDITION<br />

• PROCÉDÉ ET COMPOSITION POUR TRAI-<br />

TER UNE AFFECTION VÉHICULÉE PAR<br />

RÉCEPTEUR DE LA SÉROTONINE<br />

(71) Vanda Pharmaceuticals Inc., 9605 Medical<br />

Center Drive, Suite 300, Rockville, NY 20850,<br />

US<br />

(72) POLYMEROPOULOS, Mihael, H., Potomac<br />

MD 20854, US<br />

BAROLDI, Paolo, MD 20854, US<br />

WOLFGANG, Curt, D., Germantown MD<br />

20874, US<br />

(74) Johnson, Graham Pierssene, Appleyard Lees<br />

15 Clare Road, Halifax HX1 2HY, GB<br />

(51) A61K 31/445 (11) 2 222 301 A1*<br />

A61P 13/08<br />

(25) En (26) En<br />

(21) 08859451.0 (22) 13.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/086733 13.12.2008<br />

(87) WO 2009/076663 2009/25 18.06.2009<br />

(30) 13.12.2007 US 13375<br />

(54) • VERFAHREN UND ZUSAMMENSETZUNG<br />

ZUR BEHANDLUNG EINER ERKRANKUNG,<br />

DIE DURCH DEN ALPHA-ADRENOZEPTOR<br />

VERMITTELT WIRD<br />

• METHOD AND COMPOSITION FOR<br />

TREATING AN ALPHA ADRENOCEPTOR-<br />

MEDIATED CONDITION<br />

• PROCÉDÉ ET COMPOSITION POUR TRAI-<br />

TER UNE AFFECTION VÉHICULÉE PAR<br />

ALPHA-ADRÉNOCEPTEUR<br />

(71) Vanda Pharmaceuticals Inc., 9605 Medical<br />

Center Drive, Suite 300, Rockville, NY 20850,<br />

US<br />

(72) POLYMEROPOULOS, Mihael, H., Potomac<br />

MD 20854, US<br />

BAROLDI, Paolo, Potomac MD 20854, US<br />

WOLFGANG, Curt, D., Germantown MD<br />

20874, US<br />

(74) Johnson, Graham Pierssene, Appleyard Lees<br />

15 Clare Road, Halifax HX1 2HY, GB<br />

A61K 31/4468 → (51) C07D 207/12<br />

A61K 31/451 → (51) A61K 31/445<br />

(51) A61K 31/46<br />

A61P 3/04<br />

(11) 2 222 302 A1*<br />

(25) En (26) En

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