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Bulletin 2010/35 - European Patent Office

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(C07D) II.1(1)<br />

C07D 417/06 → (51) A61K 31/167<br />

(51) C07D 451/04 (11) 1 874 766 B1<br />

A61K 31/40 A61P 1/00<br />

(25) En (26) En<br />

(21) 06740692.6 (22) 05.04.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

HR<br />

(43) 09.01.2008<br />

(86) US 2006/012978 05.04.2006<br />

(87) WO 2006/108127 2006/41 12.10.2006<br />

(30) 06.04.2005 US 668780 P<br />

(54) • KRISTALLINE FORM EINER CHINOLIN-<br />

CARBOXAMID-VERBINDUNG<br />

• CRYSTALLINE FORM OF A QUINOLINONE-<br />

CARBOXAMIDE COMPOUND<br />

• FORME CRISTALLINE D'UN COMPOSE<br />

QUINOLINONE-CARBOXAMIDE<br />

(73) Theravance, Inc., 901 Gateway Boulevard,<br />

South San Francisco, CA 94080, US<br />

(72) FATHEREE, Paul R., San Francisco, California<br />

94107, US<br />

TURNER, S. Derek, Reston, VA 20191, US<br />

GOLDBLUM, Adam, Berkeley, California<br />

94702, US<br />

CHAO, Robert, Santa Clara, California 95054,<br />

US<br />

GENOV, Daniel, San Francisco, California<br />

94109, US<br />

(74) Scott, Susan Margaret, et al, Abel & Imray 20<br />

Red Lion Street, London WC1R 4PQ, GB<br />

(51) C07D 471/04 (11) 1 560 488 B1<br />

C07D 513/04 C07D 519/00<br />

C07D 413/12 A61K 31/53<br />

A61K 31/44 A61K 31/47<br />

A61P 33/00<br />

(25) En (26) En<br />

(21) 03783156.7 (22) 04.11.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

LT LV<br />

(43) 10.08.2005<br />

(86) US 2003/0<strong>35</strong>206 04.11.2003<br />

(87) WO 2004/041210 2004/21 21.05.2004<br />

(30) 05.11.2002 US 423872 P<br />

(54) • ANTIBAKTERIELLE MITTEL<br />

• ANTIBACTERIAL AGENTS<br />

• AGENTS ANTIBACTERIENS<br />

(73) Glaxo Group Limited, Glaxo Wellcome House<br />

Berkeley Avenue Greenford, Middlesex UB6<br />

0NN, GB<br />

(72) AXTEN, Jeffrey, Michael, Collegeville, PA<br />

19426, US<br />

GALLAGHER, Timothy, Francis, Collegeville,<br />

PA 19426, US<br />

MILLER, William, Henry, Collegeville, PA<br />

19426, US<br />

SEEFELD, Mark, Anthony, Collegeville, PA<br />

19426, US<br />

(74) Valentine, Jill Barbara, et al, GlaxoSmithKline<br />

Corporate Intellectual Property (CN9.25.1)<br />

980 Great West Road, Brentford, Middlesex<br />

TW8 9GS, GB<br />

(51) C07D 471/04 (11) 1 709 047 B1<br />

A61K 31/4<strong>35</strong>5 A61P 31/14<br />

(25) En (26) En<br />

(21) 05705124.5 (22) 05.01.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) 11.10.2006<br />

(86) US 2005/000339 05.01.2005<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(87) WO 2005/067900 2005/30 28.07.2005<br />

(30) 06.01.2004 US 534839 P<br />

(54) • AZABENZOFURANSUBSTITUIERTE THIO-<br />

HARNSTOFFE ALS INHIBITOREN DER<br />

VIRUSREPLIKATION<br />

• AZABENZOFURAN SUBSTITUTED<br />

THIOUREAS AS INHIBITORS OF VIRAL<br />

REPLICATION<br />

• THIOUREES A SUBSTITUTION AZABEN-<br />

ZOFURANE UTILISEES EN TANT QU'INHI-<br />

BITEURS DE REPLICATION VIRALE<br />

(73) Achillion Pharmaceuticals, Inc., 300 George<br />

Street, New Haven, CT 06511, US<br />

(72) THURKAUF, Andrew, Ridgefield, CT 06877,<br />

US<br />

CHEN, Dawei, Middletown, CT 06457 Middlesex<br />

County, US<br />

PHADKE, Avinash, Branford, CT 06405, US<br />

LI, Shouming, Cheshire, CT 06410, US<br />

DESHPANDE, Milind, Madison, CT 06443,<br />

US<br />

(74) Smaggasgale, Gillian Helen, W.P. Thompson<br />

& Co 55 Drury Lane, London WC2B 5SQ, GB<br />

(51) C07D 471/04 (11) 2 102 205 B1<br />

A01N 43/90 A01P 13/00<br />

(25) En (26) En<br />

(21) 07848431.8 (22) 06.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 23.09.2009<br />

(86) GB 2007/004662 06.12.2007<br />

(87) WO 2008/071918 2008/25 19.06.2008<br />

(30) 12.12.2006 GB 0624760<br />

(54) • ALS HERBIZIDE VERBINDUNGEN GEEIG-<br />

NETE PYRIDOPYRAZINDERIVATE<br />

• PYRIDO-PYRAZINE DERIVATIVES USEFUL<br />

AS HERBICIDAL COMPOUNDS<br />

• DÉRIVÉS DE PYRIDO-PYRAZINE UTILES<br />

EN TANT QUE COMPOSÉS HERBICIDES<br />

(73) Syngenta Limited, <strong>European</strong> Regional Centre<br />

Priestley Road Surrey Research Park, Guildford<br />

Surrey GU2 7YH, GB<br />

(72) CARTER, Neil Brian, Berkshire RG42 6EY, GB<br />

CORDINGLEY, Matthew Robert, Berkshire<br />

RG42 6EY, GB<br />

CROWLEY, Patrick Jelf, Berkshire RG42 6EY,<br />

GB<br />

TURNBULL, Michael Drysdale, Berkshire<br />

RG42 6EY, GB<br />

(74) Ward, Steven Paul, et al, Syngenta Limited,<br />

Intellectual Property Department, Jealott's<br />

Hill International Research Centre, P.O. Box<br />

<strong>35</strong>38, Bracknell , Berkshire RG42 6YA, GB<br />

C07D 471/04 → (51) A61K 31/167<br />

(51) C07D 471/14 (11) 1 558 614 B1<br />

A61K 31/4375 A61P 29/00<br />

A61P 11/00<br />

(25) En (26) En<br />

(21) 03809672.3 (22) 28.10.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

LT LV<br />

(43) 03.08.2005<br />

(86) CA 2003/001658 28.10.2003<br />

(87) WO 2004/039807 2004/20 13.05.2004<br />

(30) 30.10.2002 US 422443 P<br />

26.06.2003 US 482626 P<br />

(54) • PYRIDOPYRROLIZIN- UND PYRIDOINDO-<br />

LIZINDERIVATE<br />

• PYRIDOPYRROLIZINE AND PYRIDOINDO-<br />

LIZINE DERIVATIVES<br />

587<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

• PYRIDOPYRROLIZINE ET DERIVES DE<br />

PYRIDOINDOLIZINE<br />

(73) Merck Frosst Canada Ltd., 16711 Trans-<br />

Canada Highway, Kirkland, Québec H9H 3L1,<br />

CA<br />

(72) LEBLANC, Yves, Kirkland, Québec H9H 3L1,<br />

CA<br />

DUFRESNE, Claude, Kirkland, Québec H9H<br />

3L1, CA<br />

ROY, Patrick, Kirkland, Québec H9H 3L1, CA<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

(51) C07D 487/04 (11) 1 812 439 B1<br />

A61K 31/53 A61P 25/16<br />

A61P 29/00 A61P <strong>35</strong>/00<br />

A61P 25/18 A61P 25/24<br />

A61P 25/28<br />

(25) En (26) En<br />

(21) 05810<strong>35</strong>3.2 (22) 14.10.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 01.08.2007<br />

(86) US 2005/037059 14.10.2005<br />

(87) WO 2006/044687 2006/17 27.04.2006<br />

(30) 15.10.2004 US 619302<br />

11.05.2005 US 679690<br />

(54) • KINASEINHIBITOREN<br />

• KINASE INHIBITORS<br />

• INHIBITEURS DE KINASE<br />

(73) Takeda Pharmaceutical Company Limited, 1-<br />

1 Doshomachi 4-chome Chuo-ku, Osaka-shi,<br />

Osaka 541-0045, JP<br />

(72) DONG, Qing, San Diego, CA 92130, US<br />

HOSFIELD, David, Solana Beach, CA 92075,<br />

US<br />

PARASELLI, Bheema R., San Diego, CA<br />

92130, US<br />

SCORAH, Nicholas, San Diego, CA 92130,<br />

US<br />

STAFFORD, Jeffrey A., San Diego, CA 92130,<br />

US<br />

WALLACE, Michael, San Diego, CA 92117,<br />

US<br />

ZHANG, Zhiyuan, San Diego, CA 92130, US<br />

(74) Duncan, Garreth Andrew, et al, D Young &<br />

Co LLP 120 Holborn, London EC1N 2DY, GB<br />

(51) C07D 487/04 (11) 1 883 639 B1<br />

(25) En (26) En<br />

(21) 06743955.4 (22) 19.05.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 06.02.2008<br />

(86) GB 2006/001877 19.05.2006<br />

(87) WO 2006/123175 2006/47 23.11.2006<br />

(30) 20.05.2005 GB 0510345<br />

(54) • HERSTELLUNG VON FAMCICLOVIR UND<br />

ANDEREN PURINDERIVATEN<br />

• PREPARATION OF FAMCICLOVIR AND<br />

OTHER PURINE DERIVATIVES<br />

• SYNTHÈSE DU FAMCICLOVIR ET D'AUTRE<br />

DÉRIVÉS DE PURINE<br />

(73) Arrow International Limited, 57 St Christopher<br />

Street, Valetta, VLT 08, MT<br />

Chongqing Shenghuaxi Pharmaceutical Co.,<br />

Ltd., Renjiawan, Dashiba, Nan-an Chongqing,<br />

CN<br />

(72) HE, Liang, Renjiawan, Dashiba Nan-an,<br />

Chongqing, CN<br />

JIANG, Weiping, Renjiawan, Dashiba Nan-an,<br />

Chongqing, CN

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