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Bulletin 2010/35 - European Patent Office

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(C07D) II.1(1)<br />

TAKEMOTO, Masaki Mitsubishi Gas Chemical<br />

Co., Inc., Shinwari, Niigata-shi Niigata<br />

9503112, JP<br />

NAKANO, Rieko c/o Mitsubishi Gas Chemical<br />

Co., Inc, Shinwari, Niigata-shi Niigata<br />

9503112, JP<br />

(74) Harrison, Robert John, et al, 24IP Law Group<br />

Sonnenberg Fortmann <strong>Patent</strong>- & Rechtsanwälte<br />

Postfach 33 08 65, 80068 München,<br />

DE<br />

C07D 303/16 → (51) C07D 301/12<br />

(51) C07D 305/12 (11) 1 751 126 B1<br />

A61K 31/3<strong>35</strong> A61P 3/00<br />

(25) De (26) De<br />

(21) 05716736.3 (22) 18.02.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) 14.02.2007<br />

(86) EP 2005/050719 18.02.2005<br />

(87) WO 2005/080366 2005/<strong>35</strong> 01.09.2005<br />

(30) 23.02.2004 DE 102004009076<br />

(54) • ALKYLCARBAMAT-SUBSTITUIERTE<br />

BUTYROLACTONE ALS LIPASE-INHIBITO-<br />

REN<br />

• ALKYL CARBAMATE-SUBSTITUTED<br />

BUTYROLACTONES SERVING AS LIPASE<br />

INHIBITORS<br />

• BUTYROLACTONES SUBSTITUEES PAR<br />

CARBAMATE D'ALKYLE, UTILISEES<br />

COMME INHIBITEURS DE LIPASE<br />

(73) Abbott Products GmbH, Hans-Böckler-Allee<br />

20, 30173 Hannover, DE<br />

(72) WALDECK, Harald, 30916 Isernhagen, DE<br />

ANTEL, Jochen, 31848 Bad Münder, DE<br />

EYTING, Sabine, 48159 Münster, DE<br />

WURL, Michael, 30826 Garbsen, DE<br />

GREGORY, Peter-Colin, 30559 Hannover, DE<br />

WOLFF, Maike, 30171 Hannover, DE<br />

(74) Gosmann, Martin, et al, Abbott Products<br />

GmbH IP Department (PH-ZP), Hans-Böckler-Allee<br />

20 30173 Hannover, DE<br />

C07D 307/20 → (51) C07D 319/06<br />

C07D 309/12 → (51) C07D 319/06<br />

(51) C07D 309/30 (11) 1 555 261 B1<br />

A61K 8/36 A61Q 13/00<br />

C11B 9/00 A23L 1/226<br />

A23L 2/00<br />

(25) Ja (26) En<br />

(21) 03753957.4 (22) 26.09.2003<br />

(84) CH DE ES FR GB LI<br />

(43) 20.07.2005<br />

(86) JP 2003/012341 26.09.2003<br />

(87) WO 2004/029033 2004/15 08.04.2004<br />

(30) 27.09.2002 JP 2002282675<br />

23.10.2002 JP 2002308952<br />

16.09.2003 JP 2003323125<br />

(54) • VALEROLACTONVERBINDUNGEN UND<br />

PARF MZUSAMMENSETZUNG<br />

• VALEROLACTONE COMPOUNDS AND<br />

PERFUME COMPOSITION<br />

• COMPOSES DE VALEROLACTONE ET<br />

COMPOSITION DE PARFUM<br />

(73) KAO CORPORATION, 14-10, Nihonbashi<br />

Kayaba-cho 1-chome, Chuo-ku, Tokyo 103-<br />

8210, JP<br />

(72) Tanaka, Sakuya, Wakayama-shi, Wakayama<br />

640-8580, JP<br />

Fukuda, Kazuyuki, Sumida-ku, Tokyo 131-<br />

8501, JP<br />

Asada, Takahiro, Wakayama-shi, Wakayama<br />

640-8580, JP<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

(51) C07D 311/08 (11) 2 019 825 B1<br />

A61K 31/<strong>35</strong>2 A61K 31/47<br />

A61P 31/18 C07D 215/22<br />

C07D 215/14 C07D 215/18<br />

C07D 311/12 C07D 311/14<br />

C07D 401/04 C07D 401/12<br />

C07D 405/04 C07D 409/04<br />

C07D 413/12 C07D 215/227<br />

(25) En (26) En<br />

(21) 07784947.9 (22) 14.05.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

BA HR RS<br />

(43) 04.02.2009<br />

(86) CA 2007/000845 14.05.2007<br />

(87) WO 2007/131<strong>35</strong>0 2007/47 22.11.2007<br />

(30) 16.05.2006 US 747311 P<br />

(54) • HEMMER DER NEUBILDUNG MENSCH-<br />

LICHER IMMUNDEFEKT-VIREN<br />

• INHIBITORS OF HUMAN IMMUNODEFI-<br />

CIENCY VIRUS REPLICATION<br />

• INHIBITEURS DE LA RÉPLICATION DU<br />

VIRUS DE L'IMMUNODÉFICIENCE<br />

HUMAINE<br />

(73) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim, DE<br />

(84) AT BE BG CH CY CZ DK EE ES FI FR GB GR<br />

HU IE IS IT LI LT LU LV MC MT NL PL PT RO<br />

SE SI SK TR<br />

(73) Boehringer Ingelheim Pharma GmbH & Co.<br />

KG, Binger Strasse 173, 55216 Ingelheim,<br />

DE<br />

(84) DE<br />

(72) TSANTRIZOS, Youla, S., Laval, Quebec H7S<br />

2G5, CA<br />

BOES, Michael, 80796 Munich, DE<br />

BROCHU, Christian, Laval, Québec H7S 2G5,<br />

CA<br />

FENWICK, Craig, Laval, Québec H7S 2G5, CA<br />

MALENFANT, Eric, Laval, Québec H7S 2G5,<br />

CA<br />

MASON, Stephen, Laval, Québec H7S 2G5,<br />

CA<br />

PESANT, Marc, Laval, Québec H7S 2G5, CA<br />

(74) Hammann, Heinz, Boehringer Ingelheim<br />

GmbH CD-<strong>Patent</strong>s Binger Straße 173, 55216<br />

Ingelheim am Rhein, DE<br />

C07D 311/12 → (51) C07D 311/08<br />

C07D 311/14 → (51) C07D 311/08<br />

C07D 317/24 → (51) C07D 319/06<br />

(51) C07D 319/06 (11) 1 637 528 B1<br />

C07D 317/24 C07D 309/12<br />

C07D 307/20 C07D 493/04<br />

A61K 31/<strong>35</strong> A61P 31/12<br />

(25) En (26) En<br />

(21) 05028389.4 (22) 18.04.1996<br />

(84) AT BE CH DE DK ES FI FR GB GR IE IT LI LU<br />

MC NL PT SE<br />

AL LT LV SI<br />

(43) 22.03.2006<br />

(30) 19.04.1995 US 424810<br />

(54) • Sulfonamide, die einen sauerstoffhaltigen<br />

Heterozyklus enthalten als Inhibitoren von<br />

Aspartyl-Protease<br />

• Oxygenated-heterocycle containing sulfonamide<br />

inhibitors of aspartyl protease<br />

• Sufamides contenant des hétérocycles<br />

oxygénés et agissant comme inhibiteurs de<br />

l'aspartyle protéase<br />

585<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

(73) VERTEX PHARMACEUTICALS INCORPO-<br />

RATED, 130 Waverly Street, Cambridge, MA<br />

02139-4242, US<br />

(72) Tung, Roger D., San Diego, CA 92130, US<br />

Bhisetti, Govinda Rao, Lexington MA 02421,<br />

US<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

(62) 0111<strong>35</strong>75.3 / 1 136 479<br />

96913811.4 / 0 833 826<br />

C07D 333/16 → (51) C12P 17/16<br />

C07D 333/20 → (51) C12P 17/16<br />

C07D 333/34 → (51) C07D 213/71<br />

C07D 333/36 → (51) C07C 323/42<br />

C07D 333/36 → (51) C07D 409/12<br />

C07D 333/48 → (51) C07C 323/42<br />

C07D 3<strong>35</strong>/02 → (51) C07C 323/42<br />

(51) C07D 401/04 (11) 1 607 394 B1<br />

(25) Zh (26) En<br />

(21) 04717008.9 (22) 04.03.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

(43) 21.12.2005<br />

(86) CN 2004/000167 04.03.2004<br />

(87) WO 2004/085422 2004/41 07.10.2004<br />

(30) 27.03.2003 CN 03120994<br />

(54) • WASSERLÖSLICHE THALIDOMINDERI-<br />

VATE<br />

• WATER-SOLUBLE THALIDOMINE DERI-<br />

VATIVES<br />

• DERIVES DE THALIDOMIDE HYDROSO-<br />

LUBLE<br />

(73) Tian Jin Hemay Bio-Tech Co., Ltd., Xiao<br />

Yuan Xin Cun 31-101 Teda, Tianjin 300457,<br />

CN<br />

(72) ZHANG, Hesheng, Tianjin, 300457, CN<br />

(74) Stuttard, Garry Philip, Urquhart-Dykes &<br />

Lord LLP Tower North Central Merrion Way,<br />

Leeds LS2 8PA, GB<br />

C07D 401/04 → (51) C07D 311/08<br />

C07D 401/04 → (51) C07D 401/14<br />

C07D 401/06 → (51) A61K 31/167<br />

C07D 401/06 → (51) A61K 31/496<br />

(51) C07D 401/12 (11) 1 856 096 B1<br />

C07D 207/14 A61K 31/4725<br />

A61K 31/40<br />

(25) En (26) En<br />

(21) 067177<strong>35</strong>.2 (22) 09.01.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 21.11.2007<br />

(86) US 2006/000571 09.01.2006<br />

(87) WO 2006/076246 2006/29 20.07.2006<br />

(30) 10.01.2005 US 642751 P<br />

(54) • ALS ANTIKOAGULANZIEN VERWENDBARE<br />

PHENYLGLYCINAMID-DERIVATE<br />

• PHENYLGLYCINAMIDE DERIVATIVES<br />

USEFUL AS ANTICOAGULANTS<br />

• DERIVES DE PHENYLGLYCINAMIDE UTI-<br />

LISES COMME ANTICOAGULANTS<br />

(73) Bristol-Myers Squibb Company, Route 206<br />

and Province Line Road, Princeton NJ<br />

08543-4000, US

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