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Bulletin 2010/35 - European Patent Office

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(C07C) II.1(1)<br />

(21) 03757879.6 (22) 22.09.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 27.07.2005<br />

(86) EP 2003/010501 22.09.2003<br />

(87) WO 2004/033416 2004/17 22.04.2004<br />

(30) 04.10.2002 DE 10246434<br />

(54) • CARBOXYALKOXY-SUBSTITUIERTE ACYL-<br />

CARBOXYPHENYL-HARNSTOFFDERIVATE,<br />

VERFAHREN ZU IHRE HERSTELLUNG UND<br />

IHRE VERWENDUNG ALS ARZNEIMITTEL<br />

• CARBOXYALKOXY-SUBSTITUTED ACYL-<br />

CARBOXYPHENYL-UREA DERIVATIVES,<br />

PRODUCTION METHOD AND USE<br />

THEREOF AS MEDICINE<br />

• DERIVES D'ACYL-CARBOXYPHENYL-<br />

UREE A SUBSTITUTION CARBOXYAL-<br />

COXY, LEUR PROCEDE DE PRODUCTION<br />

ET LEUR UTILISATION EN TANT QUE<br />

MEDICAMENT<br />

(73) Sanofi-Aventis Deutschland GmbH,<br />

Brüningstraße 50, 65929 Frankfurt am Main,<br />

DE<br />

(72) DEFOSSA, Elisabeth, 65510 Idstein, DE<br />

KADEREIT, Dieter, 63071 Offenbach, DE<br />

KLABUNDE, Thomas, 65926 Frankfurt am<br />

Main, DE<br />

BURGER, Hans-Joerg, Morristown, NJ<br />

07960, US<br />

HERLING, Andreas, 65520 Bad Camberg, DE<br />

WENDT, Karl-Ulrich, 65926 Frankfurt am<br />

Main, DE<br />

VON REODERN, Erich, 65795 Hattersheim,<br />

DE<br />

SCHOENAFINGER, Karl, 63755 Alzenau, DE<br />

ENHSEN, Alfons, 64572 Büttelborn, DE<br />

C07C 309/65 → (51) C07C 51/08<br />

C07C 317/40 → (51) C07C 323/42<br />

(51) C07C 323/42 (11) 1 006 107 B1<br />

C07C 317/40 C07D 213/70<br />

C07D 239/26 C07D 277/36<br />

C07D 277/76 C07D 285/12<br />

C07D 333/36 C07D 333/48<br />

C07D 3<strong>35</strong>/02 A01N 37/10<br />

A01N 43/10 A01N 43/18<br />

A01N 43/40 A01N 43/54<br />

A01N 47/02 A01N 47/12<br />

(25) En (26) En<br />

(21) 99123195.2 (22) 24.11.1999<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE<br />

(43) 07.06.2000<br />

(30) 30.11.1998 JP 34037998<br />

20.08.1999 JP 23432999<br />

(54) • Phthalamidderivate oder Salz davon, landund<br />

gartenbauwirtschaftliche Insektizide<br />

sowie Verfahren zu ihrer Verwendung<br />

• Phthalamide derivatives, or salt thereof<br />

agrohorticultural insecticide, and method<br />

for using the same<br />

• Dérivés de phtalamide ou leur sels, insecticides<br />

pour l'agriculture et l'horticulture et<br />

procédé pour leur mise en oeuvre<br />

(73) NIHON NOHYAKU CO., LTD., 1-2-5, Nihonbashi,<br />

Chuo-ku Tokyo100-0027, JP<br />

(72) Tohnishi, Masanori, Sakai-shi, JP<br />

Nakao, Hayami, Kawachinagano-shi, JP<br />

Kohno, Eiji, Habikino-shi, JP<br />

Nishida, Tateki, Tondabayashi-shi, JP<br />

Furuya, Takashi, Izumisano-shi, JP<br />

Shimizu, Toshiaki, Kawachinagano-shi, JP<br />

Seo, Akira, Hashimoto-shi, JP<br />

Sakata, Kazuyuki, Kawachinagano-shi, JP<br />

Fujioka, Shinsuke, Kawachinagano-shi,<br />

Osaka, JP<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

Kanno, Hideo, Ibaraki-shi, JP<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

C07D 205/04 → (51) C07D 207/14<br />

(51) C07D 207/14 (11) 1 430 027 B1<br />

C07D 211/56 C07D 405/12<br />

C07D 205/04 A61K 31/40<br />

A61K 31/445 A61K 31/4523<br />

A61P 1/04 A61P 3/04<br />

A61P 3/10 A61P 25/28<br />

A61P 37/08<br />

(25) En (26) En<br />

(21) 02764566.2 (22) 11.09.2002<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SK TR<br />

(43) 23.06.2004<br />

(86) DK 2002/000593 11.09.2002<br />

(87) WO 2003/024928 2003/13 27.03.2003<br />

(30) 14.09.2001 DK 200101344<br />

16.05.2002 DK 200200750<br />

(54) • NEUE AMINOAZETIDIN-, AMINOPYRROLI-<br />

DIN- UND AMINOPIPERIDINDERIVATIVE<br />

• NOVEL AMINOAZETIDINE, -PYRROLIDINE<br />

AND -PIPERIDINE DERIVATIVES<br />

• NOUVEAU DERIVES D'AMINOAZETIDINE,<br />

D'AMINOPYRROLIDINE ET D'AMINOPIPE-<br />

RIDINE<br />

(73) High Point Pharmaceuticals, LLC, 4170<br />

Mendenhall Oaks Parkway, High Point, NC<br />

27265, US<br />

(72) DÖRWALD, Florencio, Zaragoza, DK-2750<br />

Ballerup, DK<br />

HOHLWEG, Rolf, DK-3050 Humlebaek, DK<br />

(74) Russell, Lindsey, et al, Elkington and Fife<br />

LLP Thavies Inn House 3-4 Holborn Circus,<br />

London EC1N 2HA, GB<br />

C07D 207/14 → (51) C07D 401/12<br />

(51) C07D 209/14 (11) 1 921 063 B1<br />

B41M 5/26 C07F 17/02<br />

G02B 5/22 G11B 7/244<br />

C07F 15/06<br />

(25) Ja (26) En<br />

(21) 06781236.2 (22) 19.07.2006<br />

(84) DE FR GB<br />

(43) 14.05.2008<br />

(86) JP 2006/314229 19.07.2006<br />

(87) WO 2007/018015 2007/07 15.02.2007<br />

(30) 11.08.2005 JP 2005233329<br />

(54) • INDOLVERBINDUNG, OPTISCHER FILTER<br />

UND MATERIAL FÜR OPTISCHE AUF-<br />

ZEICHNUNG<br />

• INDOLE COMPOUND, OPTICAL FILTER<br />

AND OPTICAL RECORDING MATERIAL<br />

• COMPOSÉ INDOLIQUE, FILTRE OPTIQUE<br />

ET MATÉRIAU D ENREGISTREMENT<br />

OPTIQUE<br />

(73) Adeka Corporation, 2-<strong>35</strong>, Higashiogu 7chome<br />

Arakawa-ku, Tokyo 116-8554, JP<br />

(72) YANAGISAWA, Satoshi c/o ADEKA COR-<br />

PORATION, Tokyo 1168554, JP<br />

(74) Forstmeyer, Dietmar, et al, BOETERS &<br />

LIECK Oberanger 32, 80331 München, DE<br />

C07D 211/14 → (51) A61K 31/167<br />

C07D 211/16 → (51) A61K 31/167<br />

C07D 211/18 → (51) A61K 31/167<br />

C07D 211/22 → (51) A61K 31/167<br />

C07D 211/56 → (51) C07D 207/14<br />

582<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

C07D 213/70 → (51) C07C 323/42<br />

(51) C07D 213/71 (11) 1 979 322 B1<br />

C07D 233/84 C07D 241/18<br />

C07D 261/10 C07D 277/36<br />

C07D 295/18 C07D 295/22<br />

C07D 333/34 A61K 31/495<br />

A61P 1/00 A61P 25/00<br />

A61P 3/00<br />

(25) En (26) En<br />

(21) 07703820.6 (22) 12.01.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 15.10.2008<br />

(86) EP 2007/050279 12.01.2007<br />

(87) WO 2007/082840 2007/30 26.07.2007<br />

(30) 23.01.2006 EP 06100701<br />

(54) • CYCLOHEXYL-SULFONAMID-DERIVATE<br />

MIT H3-REZEPTORAKTIVITÄT<br />

• CYCLOHEXYL SULFONAMIDE DERIVA-<br />

TIVES HAVING H3 RECEPTOR ACTIVITY<br />

• DÉRIVÉS DE CYCLOHEXYLSULFONAMIDE<br />

PRÉSENTANT UNE ACTIVITÉ VIS-À-VIS<br />

DES RÉCEPTEURS H3<br />

(73) F.HOFFMANN-LA ROCHE AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) NETTEKOVEN, Matthias, 79639 Grenzach-<br />

Wyhlen, DE<br />

ROCHE, Olivier, F-68220 Folgensbourg, FR<br />

(74) Klostermeyer-Rauber, Dörte, et al, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(51) C07D 215/02 (11) 1 379 508 B1<br />

(25) En (26) En<br />

(21) 02802229.1 (22) 28.02.2002<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 14.01.2004<br />

(86) US 2002/005979 28.02.2002<br />

(87) WO 2002/067865 2002/36 06.09.2002<br />

(30) 28.02.2001 US 271985 P<br />

(54) • N-(ARYL)-2-ARYLETHENSULFONAMIDE<br />

UND IHRE THERAPEUTISCHEN ANWEN-<br />

DUNGEN<br />

• N-(ARYL)-2-ARYLETHENESULFONAMIDES<br />

AND THERAPEUTIC USES THEREOF<br />

• N-(ARYL)-2-ARYLETHENESULFONAMIDES<br />

ET LEUR USAGE THERAPEUTIQUE<br />

(73) Temple University - Of The Commonwealth<br />

System of Higher Education, Broad Street<br />

and Montgomery Avenue, Philadelphia, PA<br />

19122, US<br />

Onconova Therapeutics, Inc., 375 Pheasant<br />

Run, Newtown, PA 18940, US<br />

(72) REDDY, E., Premkumar, Villanova, PA<br />

19085, US<br />

REDDY, M., V., Ramana, Upper Darby, PA<br />

19082-5429, US<br />

BELL, Stanley, C., Narberth, PA 19072, US<br />

(74) Ouzman, Beverley Nicola Claire, et al,<br />

Murgitroyd & Company Scotland House 165-<br />

169 Scotland Street, Glasgow G5 8PL, GB<br />

(51) C07D 215/12 (11) 1 854 787 B1<br />

A61K 31/47 A61K 31/4709<br />

A61K 31/5377 A61P 9/00<br />

A61P 9/10 A61P 17/06<br />

A61P 19/02 A61P 27/02<br />

A61P 29/00 A61P <strong>35</strong>/00<br />

C07D 215/20 C07D 401/12<br />

C07D 401/14 C07D 409/12<br />

(25) Ja (26) En<br />

(21) 06715138.1 (22) 03.03.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 14.11.2007

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