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Bulletin 2010/35 - European Patent Office

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(C07D) I.1(1)<br />

(74) Hallybone, Huw George, et al, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

(51) C07D 239/48 (11) 2 222 648 A1*<br />

A61K 31/505 A61P 11/00<br />

A61P 17/00 A61P 27/14<br />

A61P 31/00 A61P <strong>35</strong>/00<br />

C07D 239/49 C07D 401/10<br />

C07D 401/12 C07D 403/10<br />

C07D 403/12 C07D 417/10<br />

(25) En (26) En<br />

(21) 08851708.1 (22) 21.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) SE 2008/051334 21.11.2008<br />

(87) WO 2009/067081 2009/22 28.05.2009<br />

(30) 22.11.2007 SE 0702577<br />

14.12.2007 US 13699 P<br />

(54) • PYRIMIDINDERIVATE ZUR BEHANDLUNG<br />

VON ASTHMA, COPD, ALLERGISCHER<br />

RHINITIS, ALLERGISCHER KONJUNKTIVI-<br />

TIS, ATOPISCHER DERMATITIS, KREBS,<br />

HEPATITIS B, HEPATITIS C, HIV, HPV,<br />

BAKTERIELLEN INFEKTIONEN UND DER-<br />

MATOSE<br />

• PYRIMIDINE DERIVATIVES FOR THE<br />

TREATMENT OF ASTHMA, COPD, ALLER-<br />

GIC RHINITIS, ALLERGIC CONJUNCTIVI-<br />

TIS, ATOPIC DERMATITIS, CANCER,<br />

HEPATITIS B, HEPATITIS C, HIV, HPV,<br />

BACTERIAL INFECTIONS AND DERMATO-<br />

SIS<br />

• DÉRIVÉS DE PYRIMIDINE POUR LE<br />

TRAITEMENT DE L'ASTHME, DE LA<br />

BRONCHO-PNEUMOPATHIE CHRONIQUE<br />

OBSTRUCTIVE (COPD), DE LA RHINITE<br />

ALLERGIQUE, DE LA CONJONCTIVITE<br />

ALLERGIQUE, DE LA DERMATITE ATO-<br />

PIQUE, DU CANCER, DE L'HÉPATITE B, DE<br />

L'HÉPATITE C, DU VIH, DU VPP, DES<br />

INFECTIONS BACTÉRIENNES ET DE LA<br />

DERMATOSE<br />

(71) AstraZeneca AB, 151 85 Södertälje, SE<br />

Dainippon Sumitomo Pharma Co., Ltd., 6-8,<br />

Dosho-machi 2-chome Chuo-ku Osaka-shi,<br />

Osaka 541-8524, JP<br />

(72) BENNETT, Nicholas, J., Loughborough, Leicestershire<br />

LE11 5RH, GB<br />

MCINALLY, Thomas, Loughborough, Leicestershire<br />

LE11 5RH, GB<br />

MOCHEL, Tobias, Loughborough, Leicestershire<br />

LE11 5RH, GB<br />

THOM, Stephen, Loughborough, Leicestershire<br />

LE11 5RH, GB<br />

TIDÉN, Anna-Karin, Loughborough Leicestershire<br />

LE11 5RH, GB<br />

C07D 239/49 → (51) C07D 239/48<br />

C07D 239/54 → (51) C07D 239/22<br />

(51) C07D 239/69 (11) 2 222 649 A2*<br />

A61P 9/12 A61P 11/00<br />

A61K 31/506<br />

(25) En (26) En<br />

(21) 08806793.9 (22) 24.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) GB 2008/050986 24.10.2008<br />

(87) WO 2009/053748 2009/18 30.04.2009<br />

(88) 18.06.2009<br />

(30) 24.10.2007 IN MU21082007<br />

(54) • NEUE KRISTALLINE FORMEN<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

• NOVEL CRYSTALLINE FORMS<br />

• NOUVELLES FORMES CRISTALLINES<br />

(71) Generics (UK) Limited, Albany Gate Darkes<br />

Lane, Potters Bar, Hertfordshire EN6 1AG,<br />

GB<br />

(72) GAITONDE, Abhay, Maharashtra 410208, IN<br />

MANOJKUMAR, Bindu, Maharashtra<br />

410208, IN<br />

MEKDE, Sandeep, Maharashtra 410208, IN<br />

BANSODE, Prakash, Maharashtra 410208, IN<br />

SHINDE, Dattatraya, Maharashtra 410208, IN<br />

PHADTARE, Sunanda, Maharashtra 410208,<br />

IN<br />

(74) Elend, Almut Susanne, et al, Venner Shipley<br />

LLP Byron House Cambridge Business Park<br />

Cowley Road, GB-Cambridge CB4 0WZ, GB<br />

(51) C07D 241/24 (11) 2 222 650 A1*<br />

C07D 403/06 C07D 405/12<br />

A61K 31/551 A61K 31/4965<br />

A61K 31/497 A61P 25/00<br />

(25) En (26) En<br />

(21) 08852038.2 (22) 17.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/083775 17.11.2008<br />

(87) WO 2009/067405 2009/22 28.05.2009<br />

(30) 20.11.2007 US 989236 P<br />

(54) • SUBSTITUIERTE PYRAZINYLAMIDVER-<br />

BINDUNGEN ALS MODULATOREN DES<br />

HISTAMIN-H3-REZEPTORS<br />

• SUBSTITUTED PYRAZINYL AMIDE COM-<br />

POUNDS AS MODULATORS OF THE HIS-<br />

TAMINE H3 RECEPTOR<br />

• COMPOSÉS PYRAZINYLAMIDE SUBSTI-<br />

TUÉS COMME MODULATEURS DU<br />

RÉCEPTEUR H3 DE L'HISTAMINE<br />

(71) Janssen Pharmaceutica, N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) ALLISON, Brett, D., Del Mar California<br />

92014, US<br />

GRICE, Cheryl, A., Carlsbad California 92009,<br />

US<br />

LETAVIC, Michael, A., San Diego California<br />

92130, US<br />

(74) Warner, James Alexander, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

C07D 249/18 → (51) A61K 47/48<br />

(51) C07D 251/62 (11) 2 222 651 A2*<br />

(25) En (26) En<br />

(21) 08865550.1 (22) 27.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/010073 27.11.2008<br />

(87) WO 2009/080176 2009/27 02.07.2009<br />

(88) 20.08.2009<br />

(30) 20.12.2007 EP 07024777<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

MELAMIN<br />

• PROCESS FOR THE PREPARATION OF<br />

MELAMINE<br />

• PROCÉDÉ DE PRÉPARATION DE MÉLA-<br />

MINE<br />

(71) DSM IP Assets B.V., Het Overloon 1, 6411<br />

TE Heerlen, NL<br />

(72) TJIOE, Tjay, Tjien, NL-61<strong>35</strong> JA Sittard, NL<br />

(74) Polypatent, Braunsberger Feld 29, 51429<br />

Bergisch Gladbach, DE<br />

(51) C07D 251/68 (11) 2 222 652 A2*<br />

C08K 5/00<br />

86<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

(25) En (26) En<br />

(21) 08859404.9 (22) 09.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/067070 09.12.2008<br />

(87) WO 2009/074548 2009/25 18.06.2009<br />

(88) 01.10.2009<br />

(30) 12.12.2007 EP 07123044<br />

(54) • STABILE SPEICHERLÖSUNGEN FÜR<br />

OPTISCHE AUFHELLER<br />

• STORAGE STABLE SOLUTIONS OF OPTI-<br />

CAL BRIGHTENERS<br />

• SOLUTIONS STABLES AU STOCKAGE<br />

D'AZURANTS OPTIQUES<br />

(71) Clariant Finance (BVI) Limited, Citco Building<br />

Wickhams Cay P.O. Box 662, Road Town,<br />

Tortola, VG<br />

(72) FARRAR, John Martin, Rawdon Leeds LS19<br />

6RQ, GB<br />

JACKSON, Andrew Clive, CH-4142 Münchenstein<br />

BL, CH<br />

MAHON, Margaret, West Yorkshire BD10<br />

9DH, GB<br />

OBERHOLZER, Martin, CH-4108 Witterswil,<br />

CH<br />

(74) Mikulecky, Klaus, et al, Clariant Produkte<br />

(Deutschland) GmbH Group Intellectual<br />

Property Am Unisys-Park 1, 65843 Sulzbach,<br />

DE<br />

C07D 257/04 → (51) A61K 31/655<br />

(51) C07D 261/04 (11) 2 222 653 A1*<br />

A61K 31/42 A61P 5/30<br />

A61P 5/32<br />

(25) En (26) En<br />

(21) 08852127.3 (22) 21.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) FI 2008/050675 21.11.2008<br />

(87) WO 2009/066009 2009/22 28.05.2009<br />

(30) 23.11.2007 FI 20070897<br />

(54) • NEUE 4,5-DIHYDROISOXAZOLE MIT ÖST-<br />

ROGENER WIRKUNG<br />

• NOVEL 4,5-DIHYDROISOXAZOLES WITH<br />

ESTROGENIC ACTIVITY<br />

• NOUVEAUX 4,5-DIHYDROISOXAZOLES<br />

AVEC UNE ACTIVITÉ STROGÉNIQUE<br />

(71) Pulkkinen, Juha, Mäkikatu 3 A 21, 70110<br />

Kuopio, FI<br />

Honkakoski, Paavo, Luistelijantie 7 C 17,<br />

70200 Kuopio, FI<br />

Peräkylä, Mikael, Tuomikuja 1 D 20, 70420<br />

Kuopio, FI<br />

Berczi, Istvan, Box 143A, RR 2, Lorette,<br />

Manitoba R0A 0Y0, CA<br />

Laatikainen, Reino, Kuntokuja 6 A 6, 70200<br />

Kuopio, FI<br />

(72) PULKKINEN, Juha, FI-70100 Kuopio, FI<br />

HONKAKOSKI, Paavo, FI-70200 Kuopio, FI<br />

PERÄKYLÄ, Mikael, FI-70420 Kuopio, FI<br />

BERCZI, Istvan, Manitoba R0A 0Y0, CA<br />

LAATIKAINEN, Reino, FI-70200 Kuopio, FI<br />

(74) Matilainen, Mirja Helena, et al, Oy Jalo Ant-<br />

Wuorinen AB, Iso Roobertinkatu 4-6 A,<br />

00120 Helsinki, FI<br />

(51) C07D 263/18 (11) 2 222 654 A1*<br />

C07D 263/52 C07D 317/34<br />

C07D 317/72 A23L 1/27<br />

A23L 1/305<br />

(25) De (26) De<br />

(21) 08865833.1 (22) 01.12.2008

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