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Bulletin 2010/35 - European Patent Office

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(C07D) I.1(2)<br />

C07D 409/14 → (51) C07D 333/22<br />

C07D 409/14 → (51) C07D 401/12<br />

C07D 413/04 → (51) C07D 417/04<br />

C07D 413/06 → (51) C07D 265/30<br />

C07D 413/12 → (51) C07D 401/12<br />

C07D 413/14 → (51) C07D 417/04<br />

(51) C07D 417/04 (11) 2 223 921 A1<br />

C07D 417/14 C07D 413/04<br />

C07D 413/14 C07D 403/04<br />

C07D 405/04 C07D 407/04<br />

C07D 409/04 A61K 31/41<br />

A61K 31/42 A61K 31/425<br />

(25) En (26) En<br />

(21) 10003376.0 (22) 24.01.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(30) 18.03.2005 CN 200510024468<br />

(54) • 2-Thiophen-2-yl-oxazol-, 2-Thiophen-2-ylthiazol-<br />

und 2-Thiophen-2-yl-1H-imidazol-<br />

Derivate als antivirale Wirkstoffe<br />

• 2-Thiophen-2-yl-oxazole, 2-Thiophen-2-ylthiazole<br />

and 2-Thiophen-2-yl-1H-imidazole<br />

derivatives as antiviral agents<br />

• Dérivés de 2-Thiophén-2-yl-oxazole, 2-<br />

Thiophén-2-yl-thiazole et 2-Thiophén-2-yl-<br />

1H-imidazole en tant que agents antivirales<br />

(71) Shanghai Institute of Materia Medica, Chinese<br />

Academy of Sciences, 555 Zu Chong<br />

Zhi Road Zhangjlang Hi-Tech Park Pudong<br />

New District, Shanghai <strong>2010</strong>23, CN<br />

(72) Nan, Fajun, Pudong New Shangai 201203,<br />

CN<br />

Zuo, Jianping, Pudong New Shangai<br />

201203, CN<br />

Wang, Wenlong, Pudong New Shangai<br />

201203, CN<br />

Wang, Guifeng, Pudong New Shangai<br />

201203, CN<br />

Chen, Haijun, Pudong New Shangai 201203,<br />

CN<br />

He, Peilan, Pudong New Shangai 201203,<br />

CN<br />

(74) Flaccus, Rolf-Dieter, Flaccus · Müller-Wolff<br />

<strong>Patent</strong>anwälte Bussardweg 10, 50389 Wesseling,<br />

DE<br />

(62) 06705545.9 / 1 889 843<br />

C07D 417/14 → (51) C07D 333/22<br />

C07D 417/14 → (51) C07D 417/04<br />

(51) C07D 473/00 (11) 2 223 922 A2<br />

C07D 473/16 C07D 473/24<br />

C07D 473/30 C07D 473/34<br />

C07D 473/38 C07D 473/40<br />

A61K 31/517 A61K 31/52<br />

A61P 19/10 A61P <strong>35</strong>/00<br />

(25) En (26) En<br />

(21) 10163434.3 (22) 24.04.2001<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

AL LT LV MK RO SI<br />

(27) 24.04.2001 EP 08006457<br />

(30) 25.04.2000 US 199655 P<br />

05.10.2000 US 238057 P<br />

(54) • Hemmer der menschlichen Phosphatidylinositol-3-kinase<br />

delta<br />

• Inhibitors of human phosphatidyl-inositol<br />

3-kinase delta<br />

• Inhibiteurs delta de phosphatidyl-inositol<br />

3-kinase humaine<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(71) ICOS Corporation, 22021 20th Avenue S.E.,<br />

Bothell WA 98201, US<br />

(72) Sadhu, Chancal, Bothell, WA 98012, US<br />

Dick, Ken, Bothell, VA 98021-8321, US<br />

Treiberg, Jennifer, Bothell, WA 98012, US<br />

Sowell, Gregory, Makilteo, WA 98275, US<br />

Kesicki, Edward A., Bothell, WA 98021, US<br />

Oliver, Amy, Bothell, WA 98012, US<br />

(74) Barton, Matthew Thomas, Forrester &<br />

Boehmert Pettenkoferstrasse 20-22, 80336<br />

München, DE<br />

(62) 08006457.9 / 1 939 203<br />

01928855.4 / 1 278 748<br />

C07D 473/16 → (51) C07D 473/00<br />

C07D 473/24 → (51) C07D 473/00<br />

C07D 473/30 → (51) C07D 473/00<br />

C07D 473/34 → (51) C07D 473/00<br />

C07D 473/38 → (51) C07D 473/00<br />

C07D 473/40 → (51) C07D 473/00<br />

(51) C07D 487/04 (11) 2 223 923 A1<br />

(25) En (26) En<br />

(21) 09382024.9 (22) 25.02.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(54) • Verfahren zur Herstellung eines chiralen<br />

Beta-Aminosäurederivats und Zwischenprodukte<br />

davon<br />

• Process for the preparation of a chiral beta<br />

aminoacid derivative and intermediates<br />

thereof<br />

• Procédé pour la préparation d'un dérivé<br />

d'acide aminé chiral bêta et intermédiaires<br />

correspondants<br />

(71) Esteve Química, S.A., Av. Mare de Déu de<br />

Montserrat 12, 08024 Barcelona, ES<br />

(72) Bartra Sanmarti, Martí, 08024, Barcelona, ES<br />

Rustullet Oliver, Albert, 08024, Barcelona, ES<br />

Fernandez Hernandez, Sara, 08024, Barcelona,<br />

ES<br />

Monsalvatje Llagostera, Montserrat, 08024,<br />

Barcelona, ES<br />

(74) ZBM <strong>Patent</strong>s, Zea, Barlocci & Markvardsen<br />

Plaza Catalunya, 1, 08002 Barcelona, ES<br />

C07D 491/04 → (51) C07D 231/54<br />

C07D 493/04 → (51) A01N 43/90<br />

(51) C07F 5/06 (11) 2 223 924 A1<br />

(25) Ja (26) En<br />

(21) 09825957.5 (22) 07.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) JP 2009/058616 07.05.2009<br />

(87) WO <strong>2010</strong>/055704 <strong>2010</strong>/20 20.05.<strong>2010</strong><br />

(30) 12.11.2008 JP 2008289952<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

ALUMINIUM-DIALKYLMONOHALID<br />

• PROCESS FOR PRODUCTION OF ALUMI-<br />

NUM DIALKYL MONOHALIDE<br />

• PROCÉDÉ POUR LA PRODUCTION DE<br />

MONOHALOGÉNURE DE DIALKYLALUMI-<br />

NIUM<br />

(71) Nippon Aluminium Alkyls, Ltd., 2-2, Uchisaiwaicho<br />

2-chome Chiyoda-ku, Tokyo 100-<br />

0011, JP<br />

256<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

(72) TAKAHASHI, Hideya, Takaishi-shi Osaka<br />

592-8501, JP<br />

NISHIDA, Tadao, Takaishi-shi Osaka 592-<br />

8501, JP<br />

KOGA, Seijiro, Takaishi-shi Osaka 592-8501,<br />

JP<br />

OKUTANI, Masanori, Takaishi-shi Osaka 592-<br />

8501, JP<br />

(74) Cabinet Plasseraud, 52, rue de la Victoire,<br />

75440 Paris Cedex 09, FR<br />

(51) C07F 9/09 (11) 2 223 925 A1<br />

A61K 31/437 A61P <strong>35</strong>/00<br />

(25) En (26) En<br />

(21) 10165143.8 (22) 08.10.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(30) 09.10.2006 US 539857<br />

18.04.2007 US 912625 P<br />

10.10.2006 PCT/US2006/039667<br />

(54) • Kinase-Inhibitoren<br />

• Kinase inhibitors<br />

• Inhibiteurs de kinase<br />

(71) Takeda Pharmaceutical Company Limited, 1-<br />

1, Doshomachi 4-chome Chuo-ku, Osaka<br />

541-0045, JP<br />

(72) Brown, Jason W., San Diego, CA 92107, US<br />

Dong, Qing, San Diego, CA 92130, US<br />

Paraselli, Bheema R., San Diego, CA 92130,<br />

US<br />

Stafford, Jeffrey Alan, San Diego, CA 92130,<br />

US<br />

Wallace, Michael B., San Diego, CA 92117,<br />

US<br />

(74) Duncan, Garreth Andrew, D Young & Co LLP<br />

120 Holborn, London EC1N 2DY, GB<br />

(62) 07868389.3 / 2 081 930<br />

C07F 9/50 → (51) C07C 251/66<br />

C07F 9/5<strong>35</strong> → (51) C07C 2<strong>35</strong>/06<br />

C07F 9/6512 → (51) C07F 9/6561<br />

(51) C07F 9/6558 (11) 2 223 926 A1<br />

A61K 31/661 A61P 31/10<br />

(25) Ja (26) En<br />

(21) 08868067.3 (22) 26.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/073697 26.12.2008<br />

(87) WO 2009/084621 2009/28 09.07.2009<br />

(30) 27.12.2007 JP 2007336977<br />

27.12.2007 US 17053<br />

(54) • HETEROZYKLUS- UND PHOSPHONOXY-<br />

METHYL-SUBSTITUIERTES PYRIDINDER-<br />

IVAT UND ANTIMYKOTIKUM DAMIT<br />

• PYRIDINE DERIVATIVE SUBSTITUTED<br />

WITH HETEROCYCLE AND PHOSPHO-<br />

NOXYMETHYL GROUP AND ANTIFUNGAL<br />

AGENT CONTAINING THE SAME<br />

• DÉRIVÉ DE PYRIDINE SUBSTITUÉ PAR UN<br />

HÉTÉROCYCLE ET UN GROUPE PHOS-<br />

PHONOXYMÉTHYLE ET AGENT ANTIFON-<br />

GIQUE LE CONTENANT<br />

(71) Eisai R&D Management Co., Ltd., 6-10,<br />

Koishikawa 4-chome Bunkyo-ku, Tokyo 112-<br />

8088, JP<br />

(72) MATSUKURA, Masayuki, Tsukuba-shi Ibaraki<br />

300-26<strong>35</strong>, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE

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