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Bulletin 2010/35 - European Patent Office

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(C07D) II.1(1)<br />

(86) JP 2006/304055 03.03.2006<br />

(87) WO 2006/093253 2006/36 08.09.2006<br />

(30) 03.03.2005 JP 2005058270<br />

(54) • NEUE CYCLISCHE VERBINDUNG MIT<br />

CHINOLYLALKYLTHIOGRUPPE<br />

• NOVEL CYCLIC COMPOUND HAVING<br />

QUINOLYLALKYLTHIO GROUP<br />

• NOUVEAU COMPOSE CYCLIQUE POSSE-<br />

DANT UN GROUPE QUINOLYALKYLTHIO<br />

(73) SANTEN PHARMACEUTICAL CO., LTD., 9-<br />

19, Shimoshinjo 3-chome, Higashiyodogawa-ku,<br />

Osaka-shi, Osaka 533-8651, JP<br />

(72) KAWASHIMA, Kenji, yama-cho, Ikoma-shi,<br />

Nara 6300101, JP<br />

HONDA, Takahiro, yama-cho, Ikoma-shi,<br />

Nara 6300101, JP<br />

TAJIMA, Hisashi, yama-cho, Ikoma-shi, Nara<br />

6300101, JP<br />

OKAMOTO, Kazuyoshi, yama-cho, Ikoma-shi,<br />

Nara 6300101, JP<br />

YAMAMOTO, Minoru, yama-cho, Ikoma-shi,<br />

Nara 6300101, JP<br />

(74) Müller-Boré & Partner <strong>Patent</strong>anwälte, Grafinger<br />

Straße 2, 81671 München, DE<br />

C07D 215/14 → (51) C07D 311/08<br />

C07D 215/18 → (51) C07D 311/08<br />

C07D 215/20 → (51) C07D 215/12<br />

(51) C07D 215/22 (11) 2 057 122 B1<br />

C07C 217/60 A61K 31/4<strong>35</strong><br />

A61K 31/137 A61P 9/00<br />

A61P 11/06 A61P 29/00<br />

A61P 27/06<br />

(25) En (26) En<br />

(21) 07819060.0 (22) 17.10.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 13.05.2009<br />

(86) EP 2007/008992 17.10.2007<br />

(87) WO 2008/046598 2008/17 24.04.2008<br />

(30) 20.10.2006 ES 200602676<br />

(54) • 4-( 2-AMINO-1-HYDROXYETHYL)- PHE-<br />

NOLDERIVATIVE ALS AGONISTEN DES 2-<br />

ADRENERGISCHEN REZEPTORS<br />

• DERIVATIVES OF 4-(2-AMINO-1-HYDRO-<br />

XYETHYL)PHENOL AS AGONISTS OF THE<br />

2 ADRENERGIC RECEPTOR<br />

• DÉRIVÉS DE 4-(2-AMINO-1-HYDROXYÉ-<br />

THYL)PHÉNOL EN TANT QU'AGONISTES<br />

DU RÉCEPTEUR ADRÉNERGIQUE 2<br />

(73) Almirall, S.A., Ronda del General Mitre 151,<br />

08022 Barcelona, ES<br />

(72) BACH TANA, Jordi, 08500 Vic, ES<br />

CRESPO CRESPO, Maria Isabel, 08036<br />

Barcelona, ES<br />

PUIG DURAN, Carlos, 08024 Barcelona, ES<br />

GUAL ROIG, Silvia, 08349 Cabrera de Mar,<br />

ES<br />

ORTEGA MUÑOZ, Alberto, Barcelona, ES<br />

(74) Srinivasan, Ravi Chandran, J.A. Kemp & Co.<br />

14 South Square Gray's Inn, London WC1R<br />

5JJ, GB<br />

C07D 215/22 → (51) C07D 311/08<br />

C07D 215/227→ (51) C07D 311/08<br />

(51) C07D 215/54 (11) 1 814 857 B1<br />

C07D 409/12 A61K 31/4<strong>35</strong><br />

A61P 25/00 C07F 7/22<br />

A61K 51/04 A61P 43/00<br />

(25) En (26) En<br />

(21) 05806497.3 (22) 09.11.2005<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 08.08.2007<br />

(86) HU 2005/000120 09.11.2005<br />

(87) WO 2006/051341 2006/20 18.05.2006<br />

(30) 15.11.2004 HU 0402371<br />

(54) • ISOTOPENMARKIERTE CHINOLINDERI-<br />

VATE ALS LIGANDEN DES ADENOSIN-A3-<br />

REZEPTORS<br />

• ISOTOPICALLY MARKED QUINOLINE<br />

DERIVATIVES AS ADENOSIN A3 RECEP-<br />

TOR LIGANDS<br />

• DÉRIVÉS DE QUINOLINE ISOTOPIQUE-<br />

MENT MARQUÉS ET EMPLOYÉS EN TANT<br />

QUE LIGANDS DU RÉCEPTEUR DE<br />

L'ADÉNOSINE A3<br />

(73) Sanofi-Aventis, 174, Avenue de France,<br />

75013 Paris, FR<br />

(72) TÍMÁRI, Géza, H-2220 Vecsés, HU<br />

BOER, Kinga, H-2013 Pomáz, HU<br />

TÓTH, Géza, H-6723 Szeged, HU<br />

TÖMBÖLY, Csaba, H-6723 Szeged, HU<br />

(74) Ori, Janos, et al, Chinoin Gyogyszer és<br />

Vegyészeti Termékek Gyara Zrt. To u. 1-5.,<br />

H-1045 Budapest, HU<br />

(51) C07D 231/44 (11) 1 286 969 B1<br />

(25) En (26) En<br />

(21) 01953994.9 (22) 07.06.2001<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 05.03.2003<br />

(86) EP 2001/007398 07.06.2001<br />

(87) WO 2001/094315 2001/50 13.12.2001<br />

(30) 09.06.2000 US 210803 P<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

PESTIZIDEN VERBINDUNGEN<br />

• PROCESS FOR THE PREPARATION OF<br />

PESTICIDAL COMPOUNDS<br />

• PROCEDE DE PREPARATION DE COMPO-<br />

SES PESTICIDES<br />

(73) Merial Limited, 3239 Satellite Blvd, Duluth,<br />

GA 30096-4640, US<br />

(72) ROUSSEAU, Jean-François, F-93160 Noisy<br />

Le Comte, FR<br />

(74) Clyde-Watson, Zöe, et al, D Young & Co LLP<br />

120 Holborn, London EC1N 2DY, GB<br />

C07D 233/84 → (51) C07D 213/71<br />

C07D 239/26 → (51) C07C 323/42<br />

(51) C07D 239/36 (11) 1 845 092 B1<br />

A61K 31/505 A61K 31/513<br />

A61P 3/06 A61P 3/10<br />

A61P 19/10 A61P 25/28<br />

C07D 405/06<br />

(25) Zh (26) En<br />

(21) 05824250.4 (22) 23.12.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 17.10.2007<br />

(86) CN 2005/002293 23.12.2005<br />

(87) WO 2006/066512 2006/26 29.06.2006<br />

(30) 23.12.2004 CN 200410101710<br />

(54) • PYRIMIDINONVERBINDUNGEN, IHRE<br />

HERSTELLUNG UND IHRE VERWENDUNG<br />

• PYRIMIDINONE COMPOUNDS, THEIR<br />

PREPARATION AND USE THEREOF<br />

• DÉRIVÉS DE PYRIMIDINONE, LEUR SYN-<br />

THÈSE ET LEURS APPLICATIONS<br />

(73) Yao, Hui, Room 2-201, 19th Bldg. 88<br />

Yuanmingyuan West Rd, Haidian District<br />

Beijing 100091, CN<br />

Zhejiang Hisun Pharmaceutical Co. Ltd., 46<br />

Waisha Road, Jiaojiang District Taizhou City<br />

Zhejiang Province 318000, CN<br />

583<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

(72) YAO, Hui, Beijing 100091, CN<br />

(74) Collin, Jérôme, et al, Cabinet Régimbeau 20,<br />

rue de Chazelles, 75847 Paris Cedex 17, FR<br />

C07D 239/47 → (51) C07D 401/14<br />

(51) C07D 241/04 (11) 2 038 260 B1<br />

(25) En (26) En<br />

(21) 07730171.1 (22) 14.06.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 25.03.2009<br />

(86) EP 2007/055914 14.06.2007<br />

(87) WO 2007/144409 2007/51 21.12.2007<br />

(30) 16.06.2006 EP 06115607<br />

(54) • STEREOSELEKTIVE SYNTHESE VON (S)-1-<br />

METHYL-3-PHENYLPIPERAZIN<br />

• STEREOSELECTIVE SYNTHESIS OF (S)-1-<br />

METHYL-3-PHENYLPIPERAZINE<br />

• SYNTHÈSE STÉRÉOSÉLECTIVE DE (S)-1-<br />

MÉTHYL-3-PHÉNYLPIPÉRAZINE<br />

(73) N.V. Organon, Kloosterstraat 6, 5349 AB<br />

Oss, NL<br />

(72) VAN VLIET, Michiel, Christian, Alexander,<br />

2611 VC Delft, NL<br />

KEMPERMAN, Gerardus Johannes, 5340 BH<br />

Oss, NL<br />

SCHREUDER GOEDHEIJT, Marcel, 5340 BH<br />

Oss, NL<br />

(74) Broekkamp, Chris L. E., et al, P.O. Box 20,<br />

5340 BH Oss, NL<br />

C07D 241/18 → (51) C07D 213/71<br />

(51) C07D 249/06 (11) 2 139 871 B1<br />

C08K 5/3472<br />

(25) En (26) En<br />

(21) 08747077.9 (22) 29.04.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 06.01.<strong>2010</strong><br />

(86) US 2008/061844 29.04.2008<br />

(87) WO 2008/134674 2008/45 06.11.2008<br />

(30) 30.04.2007 US 914923 P<br />

(54) • UV-ABSORBER FÜR BRILLENGLASMATE-<br />

RIAL<br />

• UV-ABSORBERS FOR OPHTHALMIC LENS<br />

MATERIALS<br />

• ABSORBEURS D'ULTRAVIOLETS POUR<br />

DES MATÉRIAUX DE LENTILLE OPHTAL-<br />

MIQUE<br />

(73) Alcon, Inc., P.O. Box 62 Bösch 69, 6331<br />

Hünenberg, CH<br />

(72) SCHLUETER, Douglas, C., Azle, Texas<br />

76020, US<br />

(74) Keller, Günter, Lederer & Keller <strong>Patent</strong>anwälte<br />

Prinzregentenstrasse 16, 80538<br />

München, DE<br />

C07D 249/08 → (51) A61K 31/4196<br />

(51) C07D 251/18 (11) 1 585 493 B1<br />

C07D 251/20<br />

(25) En (26) En<br />

(21) 04701597.9 (22) 13.01.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 19.10.2005<br />

(86) EP 2004/000164 13.01.2004<br />

(87) WO 2004/064797 2004/32 05.08.2004<br />

(30) 20.01.2003 EP 03405018<br />

(54) • TRIAZINDERIVATE ALS UV-ABSORBER<br />

• TRIAZINE DERIVATIVES AS UV ABSOR-<br />

BERS<br />

• DERIVES DE LA TRIAZINE UTILISES<br />

COMME ABSORBANTS U.V.

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