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Bulletin 2010/35 - European Patent Office

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(C07D) I.1(1)<br />

HATEGAN, Georgeta, Naperville Illinois<br />

60565, US<br />

HAGEN, Timothy, Lisle Illinois 00006-0532,<br />

US<br />

(74) Graf von Stosch, Andreas, et al, Graf von<br />

Stosch <strong>Patent</strong>anwaltsgesellschaft mbH<br />

Prinzregentenstrasse 22, 80538 München,<br />

DE<br />

(51) C07D 207/16 (11) 2 222 639 A1*<br />

C07D 213/64 C07D 213/79<br />

C07D 231/12 C07D 239/42<br />

C07D 401/06 C07D 471/04<br />

C07D 473/18 C07D 473/40<br />

C07D 285/1<strong>35</strong> C07D 213/06<br />

C07D 213/74 C07D 213/75<br />

C07D 213/84 C07D 401/04<br />

(25) En (26) En<br />

(21) 08852110.9 (22) 20.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/084230 20.11.2008<br />

(87) WO 2009/067621 2009/22 28.05.2009<br />

(30) 21.11.2007 US 989551 P<br />

(54) • BIARYLE ALS PDE4-INHIBITOREN ZUR<br />

BEHANDLUNG VON LUNGEN- UND HERZ-<br />

KREISLAUF-ERKRANKUNGEN<br />

• BIARYL PDE4 INHIBITORS FOR TREATING<br />

PULMONARY AND CARDIOVASCULAR<br />

DISORDERS<br />

• INHIBITEURS DE BIARYLE PDE4 POUR LE<br />

TRAITEMENT DE TROUBLES PULMONAI-<br />

RES ET CARDIOVASCULAIRES<br />

(71) Decode Genetics EHF, Sturlugata 8, 101<br />

Reykjavik, IS<br />

(72) SINGH, Jasbir, Naperville Illinois 60564, US<br />

GURNEY, Mark, Grand Rapids Michigan<br />

49506, US<br />

BURGIN, Alex, Kingston Washington 98346,<br />

US<br />

KISELYOV, Alexander, San Diego California<br />

92130, US<br />

RAO, Munagala, Westmont Illinois 60559,<br />

US<br />

HAGEN, Timothy, Lisle Illinois 60532, US<br />

(74) Graf von Stosch, Andreas, et al, Graf von<br />

Stosch <strong>Patent</strong>anwaltsgesellschaft mbH<br />

Prinzregentenstrasse 22, 80538 München,<br />

DE<br />

C07D 209/04 → (51) A61K 31/00<br />

C07D 209/20 → (51) A61K 31/655<br />

C07D 211/58 → (51) C07D 207/12<br />

C07D 213/06 → (51) C07D 207/16<br />

(51) C07D 213/127 (11) 2 222 640 A1*<br />

(25) En (26) En<br />

(21) 08868720.7 (22) 16.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) IN 2008/000839 16.12.2008<br />

(87) WO 2009/0840<strong>35</strong> 2009/28 09.07.2009<br />

(30) 17.12.2007 IN CH30032007<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINES E-<br />

ISOMERS VON 1-(4-METHYLPHENYL)-1-<br />

(2-PYRIDYL)-3-PYRROLIDINO-PROP-1-<br />

EN UND SÄUREZUSATZSALZEN DARAUS<br />

• A PROCESS FOR PREPARATION OF E-<br />

ISOMER OF 1-(4-METHYLPHENYL)- 1-(2-<br />

PYRID YL)-3-PYRROLIDINO PROP-1-ENE<br />

AND ACID ADDITION SALTS THEREOF<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

• PROCÉDÉ DE PRÉPARATION DE L'ISO-<br />

MÈRE E DU 1-(4-MÉTHYLPHÉNYL)-1-(2-<br />

PYRIDYL)-3-PYRROLIDINO-PROP-1-ÈNE<br />

ET DE SES SELS D'ADDITION D'ACIDE<br />

(71) Hikal Limited, 32/1, Kalena Agrahara Banner<br />

Ghatta Road, Bangalore 560 076 KRN, IN<br />

(72) GUPTA, Raj ender Pershad, 560076 Bangalore,<br />

IN<br />

HIREMATH, Veerabhadra Swamy, 560076<br />

Bangalore, IN<br />

VASANNA, Raghavendra Arekal, 560076<br />

Bangalore, IN<br />

NEKKILAR, Vasantha Gowda, 560076 Bangalore,<br />

IN<br />

(74) Jones, Nicholas Andrew, et al, Withers &<br />

Rogers LLP Goldings House 2 Hays Lane,<br />

London SE1 2HW, GB<br />

C07D 213/30 → (51) C07C 311/08<br />

C07D 213/64 → (51) C07D 207/16<br />

C07D 213/643→ (51) C07C 311/08<br />

C07D 213/65 → (51) C07C 311/08<br />

C07D 213/74 → (51) C07D 207/16<br />

C07D 213/75 → (51) C07D 207/16<br />

C07D 213/79 → (51) C07D 207/16<br />

C07D 213/84 → (51) C07D 207/16<br />

C07D 215/04 → (51) C07C 233/73<br />

C07D 215/233→ (51) A61K 31/47<br />

C07D 215/48 → (51) C07C 233/73<br />

C07D 215/58 → (51) A61K 31/00<br />

C07D 217/06 → (51) C07D 413/04<br />

C07D 217/16 → (51) C07D 413/04<br />

C07D 217/22 → (51) C07D 413/04<br />

(51) C07D 217/26 (11) 2 222 641 A1*<br />

A61K 31/472 A61P 31/00<br />

A61P <strong>35</strong>/00<br />

(25) En (26) En<br />

(21) 08828485.6 (22) 27.08.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) PL 2008/050013 27.08.2008<br />

(87) WO 2009/028972 2009/10 05.03.2009<br />

(30) 28.08.2007 PL 38321107<br />

(54) • NEUER DD-PEPTIDASE-HEMMER UND<br />

SEINE VERWENDUNG ALS ANTIBIOTIKUM<br />

ODER KREBSMITTEL<br />

• A NEW INHIBITOR OF DD-PEPTIDASE AND<br />

ITS USE AS ANTIBIOTIC OR ANTICANCER<br />

DRUG<br />

• NOUVEL INHIBITEUR DE DD-PEPTIDASE<br />

ET SON UTILISATION EN TANT QU'ANTI-<br />

BIOTIQUE OU MÉDICAMENT ANTICANCÉ-<br />

REUX<br />

(71) Panstwowy Zaklad Higieny, Ul. Chocimska<br />

24, 00-791 Warszawa, PL<br />

Instytut Chemii Organicznej Pan, ul. Kasprzaka<br />

44/52, 01-244 Warszawa, PL<br />

(72) SOLECKA, JOLANTA, PL-04-758 Warszawa,<br />

PL<br />

KOZERSKI, LECH, PL-02-744 Warszawa, PL<br />

84<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

(74) Witek, Rafal, WTS <strong>Patent</strong> Attorneys, ul.<br />

Rudolfa Weigla 12, 53-114 Wroclaw, PL<br />

(51) C07D 221/22 (11) 2 222 642 A1*<br />

C07D 489/02<br />

(25) En (26) En<br />

(21) 08861695.8 (22) 17.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/013776 17.12.2008<br />

(87) WO 2009/078987 2009/26 25.06.2009<br />

(30) 17.12.2007 US 14094<br />

(54) • VERFAHREN UND VERBINDUNGEN ZUR<br />

HERSTELLUNG VON (+) OPIATEN<br />

• PROCESS AND COMPOUNDS FOR THE<br />

PRODUCTION OF (+) OPIATES<br />

• PROCÉDÉ ET COMPOSÉS DE PRODUC-<br />

TION D'OPIACÉS (+)<br />

(71) Mallinckrodt Inc., 675 McDonnell Boulevard,<br />

Hazelwood, MO 63042, US<br />

(72) WANG, Peter, X., Clarkson Valley Missouri<br />

63005, US<br />

JIANG, Tao, St. Louis Missouri 63146, US<br />

CANTRELL, Gary, L., Troy Illinois 62294, US<br />

BERBERICH, David, W., St. Peters Missouri<br />

63376, US<br />

TRAWICK, Bobby, N., Florissant Missouri<br />

63034, US<br />

OSIEK, Todd, Ballwin Missouri 63011, US<br />

LIAO, Subo, Ballwin Missouri 63021, US<br />

MOSER, Frank, W., Arnold Missouri 63010,<br />

US<br />

MCCLURG, Joseph, P., Manchester Missouri<br />

63011-3946, US<br />

(74) Beckmann, Claus, Kraus & Weisert <strong>Patent</strong>und<br />

Rechtsanwälte Thomas-Wimmer-Ring<br />

15, 80539 München, DE<br />

(51) C07D 221/28 (11) 2 222 643 A1*<br />

C07D 489/02 A61K 31/485<br />

(25) En (26) En<br />

(21) 08862724.5 (22) 17.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/013777 17.12.2008<br />

(87) WO 2009/078988 2009/26 25.06.2009<br />

(30) 17.12.2007 US 14099<br />

(54) • SINOMENINDERIVATE UND VERFAHREN<br />

FÜR IHRE SYNTHESE<br />

• SINOMENINE DERIVATIVES AND PRO-<br />

CESSES FOR THEIR SYNTHESIS<br />

• DÉRIVÉS DE SINOMÉNINE ET PROCÉDÉS<br />

DE SYNTHÈSE<br />

(71) Mallinckrodt Inc., 675 McDonnell Boulevard,<br />

Hazelwood, MO 63042, US<br />

(72) WANG, Peter, X., Clarkson Valley Missouri<br />

63005, US<br />

JIANG, Tao, St. Louis Missouri 63146, US<br />

CANTRELL, Gary, L., Troy Illinois 62294, US<br />

BERBERICH, David, W., St. Peters Missouri<br />

63376, US<br />

TRAWICK, Bobby, N., Florissant Missouri<br />

63034, US<br />

LIAO, Subo, Ballwin Missouri 63021, US<br />

BRANDT, John, St. Charles Missouri 63301,<br />

US<br />

(74) Beckmann, Claus, Kraus & Weisert <strong>Patent</strong>und<br />

Rechtsanwälte Thomas-Wimmer-Ring<br />

15, 80539 München, DE<br />

C07D 223/16 → (51) C07D 413/04<br />

C07D 231/12 → (51) C07D 207/16

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