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Bulletin 2010/35 - European Patent Office

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(C07C) I.1(1)<br />

(30) 19.12.2007 GB 0724783<br />

02.10.2008 GB 0818068<br />

(54) • VERBINDUNGEN ZUR VERSTÄRKUNG DER<br />

AMPA-REZEPTORWIRKUNG UND IHRE<br />

VERWENDUNG IN DER MEDIZIN<br />

• COMPOUNDS WHICH POTENTIATE THE<br />

AMPA RECEPTOR AND USES THEREOF IN<br />

MEDICINE<br />

• COMPOSÉS POTENTIATEURS DU RÉCEP-<br />

TEUR AMPA ET LEURS UTILISATIONS<br />

DANS LE DOMAINE MÉDICAL<br />

(71) Glaxo Group Limited, Glaxo Wellcome House<br />

Berkeley Avenue, Greenford, Middlesex UB6<br />

0NN, GB<br />

(72) BERTHELEME, Nicolas, Harlow Essex CM19<br />

5AW, GB<br />

CHAN, Wai, Ngor, Harlow Essex CM19 5AW,<br />

GB<br />

SCOTT, Jaqueline, Sandra, Harlow Essex<br />

CM19 5AW, GB<br />

WARD, Simon, E., Harlow Essex CM19 5AW,<br />

GB<br />

(74) Sewell, Richard Charles, et al, GlaxoSmithKline<br />

(CN925.1), 980 Great West Road,<br />

Brentford, Middlesex TW8 9GS, GB<br />

(51) C07C 313/04 (11) 2 222 633 A1*<br />

(25) Fr (26) Fr<br />

(21) 08854361.6 (22) 25.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/066162 25.11.2008<br />

(87) WO 2009/068534 2009/23 04.06.2009<br />

(30) 27.11.2007 FR 0708282<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINES<br />

TRIFLUORMETHANSULPHINSÄURESAL-<br />

ZES<br />

• METHOD FOR PREPARING A TRIFLUOR-<br />

OMETHANESULPHINIC ACID SALT.<br />

• PROCEDE DE PREPARATION D'UN SEL DE<br />

L'ACIDE TRIFLUOROMETHANESULFINI-<br />

QUES.<br />

(71) Rhodia Opérations, 40 Rue de La Haie Coq,<br />

93306 Aubervilliers, FR<br />

(72) SCHANEN, Vincent, F-69006 Lyon, FR<br />

BUISINE, Olivier, F-69230 Saint Genis Laval,<br />

FR<br />

METZ, Bernard, F-69540 Irigny, FR<br />

BESSON, Bernard, F-01700 Les Echets, FR<br />

(74) Dutruc-Rosset, Marie-Claude, et al, Rhodia<br />

Services Direction Propriété Industrielle 40,<br />

rue de la Haie-Coq, 93306 Aubervilliers<br />

Cedex, FR<br />

(51) C07C 313/04 (11) 2 222 634 A1*<br />

(25) Fr (26) Fr<br />

(21) 08855128.8 (22) 25.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/066161 25.11.2008<br />

(87) WO 2009/068533 2009/23 04.06.2009<br />

(30) 27.11.2007 FR 0708281<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

TRIFLUORMETHANSULFINSÄURE<br />

• METHOD FOR PREPARING TRIFLUORO-<br />

METHANESULPHINIC ACID<br />

• PROCEDE DE PREPARATION DE L'ACIDE<br />

TRIFLUOROMETHANESULFINIQUE.<br />

(71) Rhodia Opérations, 40 Rue de La Haie Coq,<br />

93306 Aubervilliers, FR<br />

(72) SCHANEN, Vincent, F-69006 Lyon, FR<br />

BUISINE, Olivier, F-69230 Saint Genis Laval,<br />

FR<br />

METZ, Bernard, F-69540 Irigny, FR<br />

BESSON, Bernard, F-01700 Les Echets, FR<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(74) Dutruc-Rosset, Marie-Claude, et al, Rhodia<br />

Services Direction Propriété Industrielle 40,<br />

rue de la Haie-Coq, 93306 Aubervilliers<br />

Cedex, FR<br />

(51) C07C 401/00 (11) 2 222 6<strong>35</strong> A2*<br />

(25) En (26) En<br />

(21) 08851<strong>35</strong>1.0 (22) 20.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/084142 20.11.2008<br />

(87) WO 2009/067578 2009/22 28.05.2009<br />

(88) 26.11.2009<br />

(30) 20.11.2007 US 989167 P<br />

08.09.2008 US 205998<br />

(54) • NEUE VITAMIN-D-REZEPTORAKTIVATO-<br />

REN UND HERSTELLUNGSVERFAHREN<br />

• NEW VITAMIN D RECEPTOR ACTIVATORS<br />

AND METHODS OF MAKING<br />

• NOUVEAUX ACTIVATEURS DU RÉCEP-<br />

TEUR DE LA VITAMINE D ET PROCÉDÉS<br />

DE FABRICATION<br />

(71) Abbott Laboratories, 100 Abbott Park Road,<br />

Abbott Park, Illinois 60064, US<br />

(72) VON GELDERN, Thomas W., Richmond<br />

Illinois 60071, US<br />

BARKALOW, Jufang, H., Deerfield Illinois<br />

60015, US<br />

BARNES, David M., Bristol Wisconsin 53104,<br />

US<br />

HAIGHT, Anthony R., Wadsworth Illinois<br />

60083, US<br />

HENGEVELD, John E., Kenosha Wisconsin<br />

53142, US<br />

LI, Xiaofeng, Gurnee Illinois 60031, US<br />

MCLAUGHLIN, Maureen A., Kenosha Wisconsin<br />

53142, US<br />

NOONAN, William T., Mason Ohio 45040, US<br />

PEI, Zhonghua, Burlingame California 94010,<br />

US<br />

WU-WONG, Jinshyun Ruth, Libertyville Illinois<br />

60048, US<br />

(74) Modiano, Micaela Nadia, et al, Modiano &<br />

Partners Thierschstrasse 11, 80538<br />

München, DE<br />

(51) C07D 207/08 (11) 2 222 636 A2*<br />

C07D 207/09 C07D 498/04<br />

A61K 31/402 A61P 5/26<br />

(25) En (26) En<br />

(21) 08865188.0 (22) 12.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/013657 12.12.2008<br />

(87) WO 2009/082437 2009/27 02.07.2009<br />

(88) 03.09.2009<br />

(30) 21.12.2007 US 8731<br />

(54) • SELEKTIVE ANDROGENREZEPTORMODU-<br />

LATOREN (SARMS) UND IHRE VERWEN-<br />

DUNG<br />

• SELECTIVE ANDROGEN RECEPTOR MOD-<br />

ULATORS (SARMS) AND USES THEREOF<br />

• MODULATEURS SÉLECTIFS DU RÉCEP-<br />

TEUR ANDROGÈNE (SARM) ET LEURS<br />

UTILISATIONS<br />

(71) Ligand Pharmaceuticals Inc., 11085 North<br />

Torrey Pines Road Suite 300, San Diego, CA<br />

92037, US<br />

(72) ZHI, Lin, San Diego, CA 92130, US<br />

(74) Baldock, Sharon Claire, Boult Wade Tennant<br />

Verulam Gardens 70 Gray's Inn Road,<br />

London WC1X 8BT, GB<br />

83<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>35</strong>/<strong>2010</strong>) 01.09.<strong>2010</strong><br />

C07D 207/09 → (51) C07D 207/08<br />

(51) C07D 207/12 (11) 2 222 637 A1*<br />

C07D 211/58 C07D 409/12<br />

C07D 295/195 A61K 31/40<br />

A61K 31/4468 A61K 31/495<br />

A61K 31/496 A61P 11/06<br />

A61P 11/08<br />

(25) En (26) En<br />

(21) 08863026.4 (22) 12.12.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/086645 12.12.2008<br />

(87) WO 2009/079392 2009/26 25.06.2009<br />

(30) 14.12.2007 US 7750<br />

(54) • AMIDINHALTIGE VERBINDUNGEN ALS<br />

MUSCARINREZEPTOR-ANTAGONISTEN<br />

• AMIDINE-CONTAINING COMPOUNDS<br />

USEFUL AS MUSCARINIC RECEPTOR<br />

ANTAGONISTS<br />

• COMPOSÉS CONTENANT DE L'AMIDINE<br />

UTILES COMME ANTAGONISTES DU<br />

RÉCEPTEUR MUSCARINIQUE<br />

(71) Theravance, Inc., 901 Gateway Boulevard,<br />

South San Francisco, CA 94080, US<br />

(72) JI, Yu-Hua, Redwood City California 94065,<br />

US<br />

HUSFELD, Craig, Redwood City California<br />

94061, US<br />

LEE, Rick, Daly City California 94015, US<br />

MU, Yongqi, Los Altos California 94022, US<br />

SMITH, Cameron, Burlingame California<br />

94010, US<br />

(74) Scott, Susan Margaret, et al, Abel & Imray 20<br />

Red Lion Street, London WC1R 4PQ, GB<br />

(51) C07D 207/16 (11) 2 222 638 A2*<br />

C07D 213/64 C07D 213/79<br />

C07D 231/12 C07D 239/42<br />

C07D 401/06 C07D 471/04<br />

C07D 473/18 C07D 473/40<br />

C07D 285/1<strong>35</strong> C07D 213/06<br />

C07D 213/74 C07D 213/75<br />

C07D 213/84 C07D 401/04<br />

C07D 233/90<br />

(25) En (26) En<br />

(21) 08851045.8 (22) 20.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/084193 20.11.2008<br />

(87) WO 2009/067600 2009/22 28.05.2009<br />

(88) 30.07.2009<br />

(30) 21.11.2007 US 989551 P<br />

(54) • BIARYLE ALS PDE4-INHIBITOREN ZUR<br />

BEHANDLUNG VON ENTZÜNDUNGEN<br />

• BIARYL PDE4 INHIBITORS FOR TREATING<br />

INFLAMMATION<br />

• INHIBITEURS DE PDE4 BIARYLE POUR<br />

TRAITER UNE INFLAMMATION<br />

(71) Decode Genetics EHF, Sturlugata 8, 101<br />

Reykjavik, IS<br />

(72) SINGH, Jasbir, Naperville Illinois 60564, US<br />

GURNEY, Mark E., Grand Rapids Michigan<br />

49506, US<br />

BURGIN, Alex, Kingston Washington 98346,<br />

US<br />

SANDANAYAKA, Vincent, Northboro Massachusetts<br />

01532, US<br />

KISELYOV, Alexander, San Diego California<br />

92130, US<br />

MOTTA, Adalie, Naperville Illinois 60564, US<br />

SCHULTZ, Gary, Naperville Illinois 60540, US

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